Antitumor activity and COMPARE analysis of bis-indole derivatives

Bioorganic and Medicinal Chemistry

Volumn 18, Issue 9, 2010, Pages 3004-3011

  Andreani, Aldo ^a   Burnelli, Silvia ^a   Granaiola, Massimiliano ^a   Leoni, Alberto ^a   Locatelli, Alessandra ^a   Morigi, Rita ^a   Rambaldi, Mirella ^a   Varoli, Lucilla ^a   Landi, Laura ^a   Prata, Cecilia ^a   Sega, Francesco Vieceli Dalla ^a   Caliceti, Cristiana ^a   Shoemaker, Robert H ^b  

^a UNIVERSITY OF BOLOGNA   (Italy)

^b Screening Technologies Branch   (United States)

Author keywords

Antitumor; COMPARE; Hollow fiber assay; Indole; NQO1; Pyridine

Indexed keywords

INDOLE DERIVATIVE; OXIDOREDUCTASE; PYRIDINE; REDUCED NICOTINAMIDE ADENINE DINUCLEOTIDE QUINONE OXIDOREDUCTASE 1; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER INHIBITION; DRUG DESIGN; DRUG SYNTHESIS; HUMAN; HUMAN CELL; LC 50; STRUCTURE ACTIVITY RELATION;

ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CELL PROLIFERATION; DRUG SCREENING ASSAYS, ANTITUMOR; HUMANS; INDOLES; INHIBITORY CONCENTRATION 50; MOLECULAR STRUCTURE; NEOPLASMS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 77951203766     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2010.03.063     Document Type: Article

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