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Volumn 51, Issue 21, 2010, Pages 2909-2913

An efficient synthesis of sulfamides

Author keywords

[No Author keywords available]

Indexed keywords

AMIDE; CHLORINE; DORIPENEM; FAMOTIDINE; FK 506 BINDING PROTEIN; JNJ 26990990; MACITENTAN; PROLINE; PYRIDINE; QUINAGOLIDE; SOLVENT; SULFAMIDE DERIVATIVE; UNCLASSIFIED DRUG;

EID: 77950930457     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2010.03.106     Document Type: Article
Times cited : (14)

References (31)
  • 1
    • 77950943253 scopus 로고    scopus 로고
    • note
    • 2NHCONHR.
  • 7
    • 77950943887 scopus 로고    scopus 로고
    • Bender, J. A.; Ding, M.; Gentles, R. G.; Hewawasam, P. 'Cyclopropyl Fused Indolobenzazepine HCV NS5B Inhibitors', WO2009/067108 A1.
    • Bender, J. A.; Ding, M.; Gentles, R. G.; Hewawasam, P. 'Cyclopropyl Fused Indolobenzazepine HCV NS5B Inhibitors', WO2009/067108 A1.
  • 13
    • 34948846564 scopus 로고    scopus 로고
    • 10.1021/jm070435y
    • Parrish C.A., et al. J. Med. Chem. 50 (2007) 4939 10.1021/jm070435y
    • (2007) J. Med. Chem. , vol.50 , pp. 4939
    • Parrish, C.A.1
  • 19
  • 27
    • 77950932393 scopus 로고    scopus 로고
    • Preparation of various sulfamoyl chlorides have been previously reported in following patent publication. Guo, C, Dong, L, Hou, X, Vanderpool, D. L, Villafranca, J. E. PCT Int. Appl. WO 01/40185 A1, 2001
    • Preparation of various sulfamoyl chlorides have been previously reported in following patent publication. Guo, C.; Dong, L.; Hou, X.; Vanderpool, D. L.; Villafranca, J. E. PCT Int. Appl. WO 01/40185 A1, 2001.
  • 28
    • 77950949571 scopus 로고    scopus 로고
    • note
    • 2 in deuterated DMSO) consistent with unlabeled product.
  • 29
    • 77950949798 scopus 로고    scopus 로고
    • note
    • 15N-labeled product.
  • 30
    • 77950946757 scopus 로고    scopus 로고
    • note
    • Nucleophilic addition to either ortho or para position of the pyridinium ring can lead to the same terminal sulfamide side product (21). Ortho addition is shown as an example in the proposed mechanism.
  • 31
    • 77950958056 scopus 로고    scopus 로고
    • Synthetic procedure and analytical data of all compounds listed herein have been previously reported in following patent publication. Guo, C, Dong, L, Hou, X, Vanderpool, D. L, Villafranca, J. E. PCT Int. Appl. WO 01/40185 A1, 2001
    • Synthetic procedure and analytical data of all compounds listed herein have been previously reported in following patent publication. Guo, C.; Dong, L.; Hou, X.; Vanderpool, D. L.; Villafranca, J. E. PCT Int. Appl. WO 01/40185 A1, 2001.


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.