Characterization of the potent gonadotropin-releasing activity of RF9, a selective antagonist of RF-amide-related peptides and neuropeptide FF receptors: Physiological and pharmacological implications

Endocrinology

Volumn 151, Issue 4, 2010, Pages 1902-1913

  Pineda, R ^a,b   Garcia Galiano, D ^a   Sanchez Garrido, M A ^a,b   Romero, M ^a   Ruiz Pino, F ^a   Aguilar, E ^a,b,c   Dijcks, F A ^d   Blomenrohr M ^d   Pinilla, L ^b   Van Noort, P I ^d   Tena Sempere, Manuel ^a,b,c  

^a UNIVERSITY OF CÓRDOBA   (Spain)

^b Instituto de Salud Carlos III   (Spain)

^c Instituto de Salud Carlos III   (Spain)

^d MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ESTRADIOL; ESTROGEN RECEPTOR ALPHA; FOLLITROPIN; GONADOTROPIN; KISSPEPTIN; LUTEINIZING HORMONE; NEUROPEPTIDE AF RECEPTOR; NEUROPEPTIDE FF RECEPTOR; NEUROPEPTIDE RECEPTOR; PEPTIDE; RECEPTOR BLOCKING AGENT; RF 9; RF AMIDE RELATED PEPTIDE; TESTOSTERONE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DOSE RESPONSE; DRUG POTENCY; FEMALE; GONADOTROPIN RELEASE; HORMONE RELEASE; IN VITRO STUDY; IN VIVO STUDY; MALE; MOUSE; NONHUMAN; PRIORITY JOURNAL; RAT;

ADAMANTANE; ANALYSIS OF VARIANCE; ANIMALS; DIPEPTIDES; DOSE-RESPONSE RELATIONSHIP, DRUG; ESTRADIOL; ESTROGEN RECEPTOR ALPHA; ESTROUS CYCLE; FEMALE; FOLLICLE STIMULATING HORMONE; HYPOTHALAMO-HYPOPHYSEAL SYSTEM; LUTEINIZING HORMONE; MALE; MICE; PITUITARY GLAND; PROTEINS; RADIOIMMUNOASSAY; RATS; RATS, WISTAR; TIME FACTORS;

EID: 77950268600     PISSN: 00137227     EISSN: 00137227     Source Type: Journal    
DOI: 10.1210/en.2009-1259     Document Type: Article

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