SCOPUS 정보 검색 플랫폼

Volumn 5, Issue 3, 2010, Pages 428-435

Fragmenting the S100B-p53 interaction: Combined virtual/biophysical screening approaches to identify ligands

(8) Agamennone, Mariangela a Cesari, Lucia b,c Lalli, Daniela d Turlizzi, Elisa b Del Conte, Rebecca d Turano, Paola d Mangani, Stefano c Padova, Alessandro b

a UNIVERSITY OF CHIETI (Italy)

b Siena Biotech SpA (Italy)

c UNIVERSITY OF SIENA (Italy)

d UNIVERSITY OF FLORENCE (Italy)

Author keywords

Fragment based drug design; NMR spectroscopy; Protein protein interactions; X ray diffraction

Indexed keywords

LIGAND; PROTEIN; PROTEIN INHIBITOR; PROTEIN P53; PROTEIN S100B; SEN 205 A; SEN 683 A; SEN 684 A; SEN 728 A; SEN 829; TRTK 12 PROTEIN; UNCLASSIFIED DRUG;

ARTICLE; BINDING SITE; BIOPHYSICS; COMPUTER MODEL; CONTROLLED STUDY; CRYSTAL STRUCTURE; DRUG ABSORPTION; DRUG BINDING; DRUG DISTRIBUTION; DRUG ELIMINATION; DRUG IDENTIFICATION; DRUG METABOLISM; DRUG SCREENING; MOLECULAR DOCKING; MOLECULAR INTERACTION; NUCLEAR MAGNETIC RESONANCE; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PHARMACOPHORE; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN CONFORMATION; PROTEIN PROTEIN INTERACTION; X RAY CRYSTALLOGRAPHY;

CRYSTALLOGRAPHY, X-RAY; DRUG DESIGN; LIGANDS; MODELS, MOLECULAR; NERVE GROWTH FACTORS; NUCLEAR MAGNETIC RESONANCE, BIOMOLECULAR; PROTEIN BINDING; PROTEIN CONFORMATION; S100 PROTEINS; TUMOR SUPPRESSOR PROTEIN P53;

EID: 77249087753 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.200900393 Document Type: Article

Times cited : (21)

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