-
2
-
-
0034518876
-
Recent advances in the Biginelli dihydropyrimidine synthesis. New tricks from an old dog
-
DOI 10.1021/ar000048h
-
Kappe, C. O. Acc. Chem. Res. 2000, 33, 879-888. doi:10.1021/ar000048h. (Pubitemid 32056773)
-
(2000)
Accounts of Chemical Research
, vol.33
, Issue.12
, pp. 879-888
-
-
Kappe, C.O.1
-
3
-
-
4644324512
-
Demonstration of the feasibility of a direct solid-phase split-pool Biginelli synthesis of 3,4-dihydropyrimidinones
-
DOI 10.1021/ol048946r
-
Lusch, M. J.; Tallarico, J. A. Org. Lett. 2004, 6, 3237-3240. doi:10.1021/ol048946r. (Pubitemid 39297308)
-
(2004)
Organic Letters
, vol.6
, Issue.19
, pp. 3237-3240
-
-
Lusch, M.J.1
Tallarico, J.A.2
-
4
-
-
17144366282
-
-
doi:10.1002/anie.200460548
-
Ramón, D. J.; Yus, M. Angew. Chem., Int. Ed. 2005, 44, 1602-1634. doi:10.1002/anie.200460548.
-
(2005)
Angew. Chem., Int. Ed.
, vol.44
, pp. 1602-1634
-
-
Ramón, D.J.1
Yus, M.2
-
6
-
-
0038203081
-
The first catalytic, asymmetric -additions of isocyanides. Lewis-base-catalyzed, enantioselective Passerini-type reactions
-
DOI 10.1021/ja035410c
-
Denmark, S. E.; Fan, Y. J. Am. Chem. Soc. 2003, 125, 7825-7827. doi:10.1021/ja035410c. (Pubitemid 36782158)
-
(2003)
Journal of the American Chemical Society
, vol.125
, Issue.26
, pp. 7825-7827
-
-
Denmark, S.E.1
Fan, Y.2
-
7
-
-
9444230492
-
-
doi:10.1021/ol0482893
-
Andreana, P. R.; Liu, C. C.; Schreiber, S. L. Org. Lett. 2004, 6, 4231-4233. doi:10.1021/ol0482893.
-
(2004)
Org. Lett.
, vol.6
, pp. 4231-4233
-
-
Andreana, P.R.1
Liu, C.C.2
Schreiber, S.L.3
-
8
-
-
20644448209
-
Highly enantioselective one-pot, three-component imino-reformatsky reaction
-
DOI 10.1002/anie.200462757
-
Cozzi, P. G.; Rivalta, E. Angew. Chem., Int. Ed. 2005, 44, 3600-3603. doi:10.1002/anie.200462757. (Pubitemid 40831824)
-
(2005)
Angewandte Chemie - International Edition
, vol.44
, Issue.23
, pp. 3600-3603
-
-
Cozzi, P.G.1
Rivalta, E.2
-
9
-
-
0000512227
-
-
doi:10.1021/ar9502083
-
Armstrong, R. W.; Combs, A. P.; Tempest, P. A.; Brown, S. D.; Keating, T. A. Acc. Chem. Res. 1996, 29, 123-131. doi:10.1021/ar9502083.
-
(1996)
Acc. Chem. Res.
, vol.29
, pp. 123-131
-
-
Armstrong, R.W.1
Combs, A.P.2
Tempest, P.A.3
Brown, S.D.4
Keating, T.A.5
-
10
-
-
3042799070
-
A Planning Strategy for Diversity-Oriented Synthesis
-
DOI 10.1002/anie.200300626
-
Burke, M. D.; Schreiber, S. L. Angew. Chem., Int. Ed. 2004, 43, 46-58. doi:10.1002/anie.200300626. (Pubitemid 38063470)
-
(2004)
Angewandte Chemie - International Edition
, vol.43
, Issue.1
, pp. 46-58
-
-
Burke, M.D.1
Schreiber, S.L.2
-
11
-
-
0026065919
-
-
doi:10.1021/jm00106a048 Dihydropyrimidine calcium channel modulators
-
Atwal, K. S.; Swanson, B. N.; Unger, S. E.; Floyd, D. M.; Moreland, S.; Hedberg, A.; O'Reilly, B. C. J. Med. Chem. 1991, 34, 806-811. doi:10.1021/jm00106a048 Dihydropyrimidine calcium channel modulators.
-
(1991)
J. Med. Chem.
, vol.34
, pp. 806-811
-
-
Atwal, K.S.1
Swanson, B.N.2
Unger, S.E.3
Floyd, D.M.4
Moreland, S.5
Hedberg, A.6
O'Reilly, B.C.7
-
12
-
-
0034519777
-
Biologically active dihydropyrimidones of the Biginelli-type - A literature survey
-
DOI 10.1016/S0223-5234(00)01189-2
-
Kappe, C. O. Eur. J. Med. Chem. 2000, 35, 1043-1052. doi:10.1016/S0223- 5234(00)01189-2. (Pubitemid 32050011)
-
(2000)
European Journal of Medicinal Chemistry
, vol.35
, Issue.12
, pp. 1043-1052
-
-
Kappe, C.O.1
-
13
-
-
0042469059
-
-
doi:10.1002/qsar.200320001
-
Kappe, C. O. QSAR Comb. Sci. 2003, 22, 630-645. doi:10.1002/qsar. 200320001.
-
(2003)
QSAR Comb. Sci.
, vol.22
, pp. 630-645
-
-
Kappe, C.O.1
-
14
-
-
0027205552
-
-
doi:10.1016/S0040-4020(01)87971-0 For review
-
Kappe, C. O. Tetrahedron 1993, 49, 6937-6963. doi:10.1016/S0040-4020(01) 87971-0 For review.
-
(1993)
Tetrahedron
, vol.49
, pp. 6937-6963
-
-
Kappe, C.O.1
-
15
-
-
0030732273
-
A reexamination of the mechanism of the Biginelli dihydropyrimidine synthesis. Support for an N-acyliminium ion intermediate
-
DOI 10.1021/jo971010u
-
Kappe, C. O. J. Org. Chem. 1997, 62, 7201-7204. doi:10.1021/jo971010u. (Pubitemid 27463078)
-
(1997)
Journal of Organic Chemistry
, vol.62
, Issue.21
, pp. 7201-7204
-
-
Kappe, C.O.1
-
16
-
-
0032854156
-
-
Kappe, C. O.; Falsone, S. F.; Fabian, W. M. F.; Belaj, F. Heterocycles 1999, 51, 77-84.
-
(1999)
Heterocycles
, vol.51
, pp. 77-84
-
-
Kappe, C.O.1
Falsone, S.F.2
Fabian, W.M.F.3
Belaj, F.4
-
17
-
-
0032524801
-
Unprecedented catalytic three component one-pot condensation reaction: An efficient synthesis of 5-alkoxycarbonyl-4-aryl-3,4-dihydropyrimidin- 2(1H)-ones
-
DOI 10.1021/jo970846u
-
Hu, E. H.; Sidler, D. R.; Dolling, U.-H. J. Org. Chem. 1998, 63, 3454-3457. doi:10.1021/jo970846u. (Pubitemid 28269630)
-
(1998)
Journal of Organic Chemistry
, vol.63
, Issue.10
, pp. 3454-3457
-
-
Hu, E.H.1
Sidler, D.R.2
Dolling, U.-H.3
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