메뉴 건너뛰기




Volumn 12, Issue 7, 2009, Pages 62-65

Developing an appropriate salt form for an active pharmaceutical ingredient

Author keywords

[No Author keywords available]

Indexed keywords

BASE; FAMOTIDINE; SALICYLIC ACID; SODIUM CHLORIDE;

EID: 74749083749     PISSN: 10998012     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (8)

References (17)
  • 2
    • 0001056344 scopus 로고    scopus 로고
    • Preparation of Water-Soluble Compounds Through Salt Formation
    • Chapter 34 in The, CG Wermuth, ed. Academic Press, New York
    • BD Anderson and KP Flora. Preparation of Water-Soluble Compounds Through Salt Formation. Chapter 34 in The Practice of Medicinal Chemistry, CG Wermuth, ed. Academic Press, New York, 1996, pp. 739-754.
    • (1996) Practice of Medicinal Chemistry , pp. 739-754
    • Anderson, B.D.1    Flora, K.P.2
  • 4
  • 5
    • 1642457350 scopus 로고    scopus 로고
    • Automated Approach to Salt Selection for New Unique Trazodone Salts
    • EC Ware and DR Lu. An Automated Approach to Salt Selection for New Unique Trazodone Salts. Pharm. Res., 21: 177-184 (2004).
    • (2004) Pharm. Res , vol.21 , pp. 177-184
    • Ware, E.C.1    An, D.L.2
  • 6
    • 27944487022 scopus 로고    scopus 로고
    • Occurrence of Pharmaceutically Acceptable Anions and Cations in the Cambridge Structural Database
    • DA Haynes, W Jones, and WDS Motherwell. Occurrence of Pharmaceutically Acceptable Anions and Cations in the Cambridge Structural Database. J. Pharm. Sci., 94: 2111-2120 (2005).
    • (2005) J. Pharm. Sci , vol.94 , pp. 2111-2120
    • Haynes, D.A.1    Jones, W.2    Motherwell, W.D.S.3
  • 7
    • 0023032232 scopus 로고
    • Salt Selection for Basic Drugs
    • PL Gould. Salt Selection for Basic Drugs. Int. J. Pharm., 33: 201-217 (1986).
    • (1986) Int. J. Pharm , vol.33 , pp. 201-217
    • Gould, P.L.1
  • 9
    • 0031806352 scopus 로고    scopus 로고
    • In Situ Salt Screening - A Useful Technique for Discovery Support and Preformulation Studies
    • W-Q Tong and G Whitesell. In Situ Salt Screening - A Useful Technique for Discovery Support and Preformulation Studies. Pharm. Dev. Tech., 3: 215-223 (1998).
    • (1998) Pharm. Dev. Tech , vol.3 , pp. 215-223
    • Tong, W.-Q.1    Whitesell, G.2
  • 10
    • 0033671441 scopus 로고    scopus 로고
    • General Equations for In Situ Salt Screening of Multibasic Drugs in Multiprotic Acids
    • M Sacchetti. General Equations for In Situ Salt Screening of Multibasic Drugs in Multiprotic Acids. Pharm. Dev. Tech., 5: 579-582 (2000).
    • (2000) Pharm. Dev. Tech , vol.5 , pp. 579-582
    • Sacchetti, M.1
  • 11
    • 0034345216 scopus 로고    scopus 로고
    • Salt Selection and Optimization Procedures for Pharmaceutical New Chemical Entities
    • RJ Bastin, MJ Bowker, and BJ Slater. Salt Selection and Optimization Procedures for Pharmaceutical New Chemical Entities. Org. Proc. Res. Dev., 4: 427-435 (2000).
    • (2000) Org. Proc. Res. Dev , vol.4 , pp. 427-435
    • Bastin, R.J.1    Bowker, M.J.2    Slater, B.J.3
  • 12
    • 1042284960 scopus 로고    scopus 로고
    • Handbook of Pharmaceutical Salts, and, eds. Wiley-VCH, Weinheim, Germany
    • ATM Serajuddin and M Pudipeddi. Salt-Selection Strategies, chapter 6 in Handbook of Pharmaceutical Salts, PH Stahl and CG Wermuth, eds. Wiley-VCH, Weinheim, Germany, 2002, pp. 135-160.
    • (2002) Salt-Selection Strategies , pp. 135-160
    • Serajuddin, A.T.M.1    Pudipeddi, M.2
  • 13
    • 1042284962 scopus 로고    scopus 로고
    • Handbook of Pharmaceutical Salts, and, eds. Wiley-VCH, Weinheim, Germany
    • MJ Bowker. A Procedure for Salt Selection and Optimization. chapter 7 in Handbook of Pharmaceutical Salts, PH Stahl and CG Wermuth, eds. Wiley-VCH, Weinheim, Germany, 2002, pp. 161-189.
    • (2002) A Procedure for Salt Selection and Optimization , pp. 161-189
    • Bowker, M.J.1
  • 14
    • 33750904749 scopus 로고    scopus 로고
    • RB Hammond, RS Hashim, C Ma, and KJ Roberts. Grid-Based Molecular Modeling for Pharmaceutical Salt Screening: Case Example of 3,4,5,7,8,9- hexahydro-2H-pyrimido-(1,2-a)-primidinium acetate. J. Pharm. Sci., 95: 2361-2372 (2006).
    • RB Hammond, RS Hashim, C Ma, and KJ Roberts. Grid-Based Molecular Modeling for Pharmaceutical Salt Screening: Case Example of 3,4,5,7,8,9- hexahydro-2H-pyrimido-(1,2-a)-primidinium acetate. J. Pharm. Sci., 95: 2361-2372 (2006).
  • 15
    • 40149094922 scopus 로고    scopus 로고
    • Strategy for the Prediction and Selection of Drug Substance Salt Forms
    • HG Brittain. Strategy for the Prediction and Selection of Drug Substance Salt Forms. Pharm. Tech., 31(10): 78-88 (2007).
    • (2007) Pharm. Tech , vol.31 , Issue.10 , pp. 78-88
    • Brittain, H.G.1
  • 16
    • 36048986392 scopus 로고    scopus 로고
    • Critical Compilation of pKA Values for Pharmaceutical Substances
    • HG Brittain, ed. Elsevier-Academic Press, Amsterdam
    • RJ Prankerd. Critical Compilation of pKA Values for Pharmaceutical Substances. in Profiles of Drug Substances Excipients, and Related Methodology, HG Brittain, ed. Elsevier-Academic Press, Amsterdam, 2007, p 191.
    • (2007) Profiles of Drug Substances Excipients, and Related Methodology , pp. 191
    • Prankerd, R.J.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.