Tetrahydroisoquinoline derivatives as melatonin MT 2 receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 23, 2004, Pages 5881-5884

  Karageorge, George N ^a   Bertenshaw, Stephen ^a   Iben, Lawrence ^a   Xu, Cen ^a   Sarbin, Nathan ^a   Gentile, Anthony ^a   Dubowchik, Gene M ^a  

^a BRISTOL MYERS SQUIBB   (United States)

Author keywords

Antagonist; Melatonin

Indexed keywords

HORMONE RECEPTOR BLOCKING AGENT; MELATONIN RECEPTOR; MELATONIN RECEPTOR BLOCKING AGENT; TETRAHYDROISOQUINOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG POTENCY; DRUG RECEPTOR BINDING; EMBRYO; MOUSE; NONHUMAN;

HUMANS; PROTEIN BINDING; RECEPTOR, MELATONIN, MT2; TETRAHYDROISOQUINOLINES;

EID: 7044254907     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.09.024     Document Type: Article

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