Melatonin receptor antagonists that differentiate hetween the human Mel(1a) and Mel(1b) recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML(1) presynaptic heteroreceptor

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 355, Issue 3, 1997, Pages 365-375

  Dubocovich, Margarita L ^a   Masana, Monica I ^a   Iacob, Stanca ^a   Sauri, Daniel M ^a  

^a NORTHWESTERN UNIVERSITY   (United States)

Author keywords

2 125I iodomelatonin binding; COS 7 cells; Dopamine release; Human Mel(1a) and Mel(1b) recombinant receptors; Melatonin receptor antagonists; ML(1B) melatonin receptor; Rabbit retina

Indexed keywords

6 CHLOROMELATONIN; 6 METHOXYMELATONIN; 6,7 DICHLORO 2 METHYLMELATONIN; LUZINDOLE; MELATONIN; MELATONIN DERIVATIVE; MELATONIN RECEPTOR; N ACETYLTRYPTAMINE; RECEPTOR SUBTYPE; RECOMBINANT PROTEIN; TETRALIN DERIVATIVE;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CELL STRAIN COS1; CONTROLLED STUDY; DOPAMINE RELEASE; DRUG RECEPTOR BINDING; GENE EXPRESSION; HUMAN; IN VITRO STUDY; NONHUMAN; RABBIT; RETINA; STRUCTURE ACTIVITY RELATION;

ANIMALS; CELL LINE; HUMANS; IODINE RADIOISOTOPES; KINETICS; MELATONIN; RABBITS; RECEPTORS, CELL SURFACE; RECEPTORS, CYTOPLASMIC AND NUCLEAR; RECEPTORS, MELATONIN; RECEPTORS, PRESYNAPTIC; RECOMBINANT PROTEINS; RETINA;

EID: 0030964398     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/PL00004956     Document Type: Article

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