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Volumn 14, Issue 3, 2009, Pages 233-239

Dry mixing transformed micro-particles of a drug from a highly crystalline to a highly amorphous state

Author keywords

Activation; Crystallinity; Mixing; Solubility

Indexed keywords

CRYSTALLIN; GLASS; GRISEOFULVIN;

EID: 70350654533     PISSN: 10837450     EISSN: 10979867     Source Type: Journal    
DOI: 10.1080/10837450802585252     Document Type: Article
Times cited : (8)

References (34)
  • 1
    • 0022347683 scopus 로고
    • Mechanical activation of pharmaceutical systems
    • Hüttenrauch R, Fricke S, Zielke P. Mechanical activation of pharmaceutical systems. Pharm Res. 1985;6:302-306.
    • (1985) Pharm Res. , vol.6 , pp. 302-306
    • Hüttenrauch, R.1    Fricke, S.2    Zielke, P.3
  • 2
    • 0036173405 scopus 로고    scopus 로고
    • The effect of disorder on the chemical reactivity of an organic solid, tetraglycine methyl ester: Change of the reaction mechanism
    • Shalaev E, Shalaeva M, Zografi G. The effect of disorder on the chemical reactivity of an organic solid, tetraglycine methyl ester: change of the reaction mechanism. J Pharm Sci. 2002;91:584-593.
    • (2002) J Pharm Sci. , vol.91 , pp. 584-593
    • Shalaev, E.1    Shalaeva, M.2    Zografi, G.3
  • 5
    • 0037026338 scopus 로고    scopus 로고
    • Investigation of the effects of grinding and co-grinding on physicochemical properties of glisentide
    • Mura P, Cirri M, Faucci MT, Gines-Dorado JM, Bettinetti GP. Investigation of the effects of grinding and co-grinding on physicochemical properties of glisentide. J Pharm Biomed Anal. 2002;30:227-237.
    • (2002) J Pharm Biomed Anal. , vol.30 , pp. 227-237
    • Mura, P.1    Cirri, M.2    Faucci, M.T.3    Gines-Dorado, J.M.4    Bettinetti, G.P.5
  • 7
    • 0037043106 scopus 로고    scopus 로고
    • Comparison of the mechanical properties of the crystalline and amorphous forms of a drug substance
    • Hancock BC, Carlson GT, Ladipo DD, Langdon BA, Mullarney MP. Comparison of the mechanical properties of the crystalline and amorphous forms of a drug substance. Int. J. Pharm. 2002;241:73-85.
    • (2002) Int. J. Pharm. , vol.241 , pp. 73-85
    • Hancock, B.C.1    Carlson, G.T.2    Ladipo, D.D.3    Langdon, B.A.4    Mullarney, M.P.5
  • 8
    • 0037074121 scopus 로고    scopus 로고
    • The impact of low levels of amorphous material (5%) on the blending characteristics of a direct compression formulation
    • Mackin L, Sartnurak S, Thomas I, Moore S. The impact of low levels of amorphous material
    • (2002) Int J Pharm. , vol.231 , pp. 213-226
    • MacKin, L.1    Sartnurak, S.2    Thomas, I.3    Moore, S.4
  • 9
    • 0002611989 scopus 로고
    • Molekulargalenik als grundlage moderner arzneiformung
    • Hüttenrauch R. Molekulargalenik als grundlage moderner arzneiformung. Acta Pharm Technol. 1978;(Suppl. 6):55-127.
    • (1978) Acta Pharm Technol , Issue.SUPPL. 6 , pp. 55-127
    • Hüttenrauch, R.1
  • 10
    • 0033460251 scopus 로고    scopus 로고
    • The effect of dry mixing on the apparent solubility of hydrophobic, sparingly soluble drugs
    • Mosharraf M, Nyström C. The effect of dry mixing on the apparent solubility of hydrophobic, sparingly soluble drugs. Eur J Pharm Sci. 1999;9:145-156.
    • (1999) Eur J Pharm Sci. , vol.9 , pp. 145-156
    • Mosharraf, M.1    Nyström, C.2
  • 11
    • 0343651819 scopus 로고
    • The impossibility of comminuting small particles by compression
    • (London)
    • Kendall K. The impossibility of comminuting small particles by compression. Nature (London) 1978;272:710-711.
    • (1978) Nature , vol.272 , pp. 710-711
    • Kendall, K.1
  • 12
    • 0023260056 scopus 로고
    • Brittle/ductile behaviour in pharmaceutical materials used in tabletting
    • Roberts RJ, Rowe RC. Brittle/ductile behaviour in pharmaceutical materials used in tabletting. Int J Pharm. 1987;36:205-209.
    • (1987) Int J Pharm. , vol.36 , pp. 205-209
    • Roberts, R.J.1    Rowe, R.C.2
  • 13
    • 0022103712 scopus 로고
    • Studies on direct compression of tablets XIV. the effect of powder fineness on the relation between tablet permeametry surface area and compaction pressure
    • Alderborn G, Nyström C. Studies on direct compression of tablets XIV. The effect of powder fineness on the relation between tablet permeametry surface area and compaction pressure. Powder Technol. 1985;44:37-42.
    • (1985) Powder Technol. , vol.44 , pp. 37-42
    • Alderborn, G.1    Nyström, C.2
  • 14
    • 2942579233 scopus 로고    scopus 로고
    • 5th ed. Council of Europe Strasbourg
    • European Pharmacopoeia. 5th ed. Council of Europe, Strasbourg; 2005.
    • (2005) European Pharmacopoeia
  • 15
    • 0026594756 scopus 로고
    • Physicochemical aspects of drug release. XV. Investigation of diffusional transport in dissolution of suspended, sparingly soluble drugs
    • Bisrat M, Anderberg EK, Barnett MI, Nyström C. Physicochemical aspects of drug release. XV. Investigation of diffusional transport in dissolution of suspended, sparingly soluble drugs. Int J Pharm. 1992;80:191-201.
    • (1992) Int J Pharm. , vol.80 , pp. 191-201
    • Bisrat, M.1    Anderberg, E.K.2    Barnett, M.I.3    Nyström, C.4
  • 16
    • 0032103736 scopus 로고    scopus 로고
    • Crystallisation of partially amorphous griseofulvin in water vapour: Determination of kinetic parameters using isothermal heat conduction microcalorimetry
    • Ahmed H, Buckton G, Rawlins DA. Crystallisation of partially amorphous griseofulvin in water vapour: Determination of kinetic parameters using isothermal heat conduction microcalorimetry. Int J Pharm. 1998;167:139-145.
    • (1998) Int J Pharm. , vol.167 , pp. 139-145
    • Ahmed, H.1    Buckton, G.2    Rawlins, D.A.3
  • 17
    • 0026525409 scopus 로고
    • Evaluation of heat- conduction microcalorimetry in pharmaceutical stability studies. V. A new approach for continuous measurements in abundant water vapour
    • Angberg M, Nyström C, Castensson S. Evaluation of heat- conduction microcalorimetry in pharmaceutical stability studies. V. A new approach for continuous measurements in abundant water vapour. Int J Pharm. 1992;81:153-167.
    • (1992) Int J Pharm. , vol.81 , pp. 153-167
    • Angberg, M.1    Nyström, C.2    Castensson, S.3
  • 18
    • 0026734782 scopus 로고
    • Evaluation of heat- conduction microcalorimetry in pharmaceutical stability studies. VI. Continuous monitoring of the interaction of water vapour with powders and powder mixtures at various relative humidities
    • Angberg M, Nyström C, Castensson S. Evaluation of heat- conduction microcalorimetry in pharmaceutical stability studies. VI. Continuous monitoring of the interaction of water vapour with powders and powder mixtures at various relative humidities. Int J Pharm. 1992;83:11-23.
    • (1992) Int J Pharm. , vol.83 , pp. 11-23
    • Angberg, M.1    Nyström, C.2    Castensson, S.3
  • 19
    • 0009438882 scopus 로고
    • Quantitative X-ray investigations on the crystallinity of cellulose fibers. A background analysis
    • Hermans PH, Weidinger A. Quantitative X-ray investigations on the crystallinity of cellulose fibers. A background analysis. J Appl Phys. 1948;19:491-506.
    • (1948) J Appl Phys. , vol.19 , pp. 491-506
    • Hermans, P.H.1    Weidinger, A.2
  • 20
    • 0021916412 scopus 로고
    • Evaluation of two concepts of crystallinity using calcium gluceptate as a model compound
    • Suryanarayanan R, Mitchell AG. Evaluation of two concepts of crystallinity using calcium gluceptate as a model compound. Int J Pharm. 1985;24:1-17.
    • (1985) Int J Pharm. , vol.24 , pp. 1-17
    • Suryanarayanan, R.1    Mitchell, A.G.2
  • 21
    • 0022652390 scopus 로고
    • True density and thermal expansivity of pharmaceutical solids: Comparison of methods and assessment of crystallinity
    • Duncan-Hewitt WC, Grant DJW. True density and thermal expansivity of pharmaceutical solids: Comparison of methods and assessment of crystallinity. Int J Pharm. 1986;28:75-84.
    • (1986) Int J Pharm. , vol.28 , pp. 75-84
    • Duncan-Hewitt, W.C.1    Grant, D.J.W.2
  • 22
    • 0017857869 scopus 로고
    • Quantitative crystallinity determinations for β-lactam antibiotics by solution calorimetry: Correlations with stability
    • Pikal MJ, Lukes AL, Lang JE, Gaines K. Quantitative crystallinity determinations for β-lactam antibiotics by solution calorimetry: correlations with stability. J Pharm Sci. 1978;67:767-773.
    • (1978) J Pharm Sci. , vol.67 , pp. 767-773
    • Pikal, M.J.1    Lukes, A.L.2    Lang, J.E.3    Gaines, K.4
  • 23
    • 0025293878 scopus 로고
    • Characterization of calcium fenoprofen 1. Powder dissolution rate and degree of crystallinity
    • Hendriksen BA. Characterization of calcium fenoprofen 1. Powder dissolution rate and degree of crystallinity. Int J Pharm. 1990;60:243-252.
    • (1990) Int J Pharm. , vol.60 , pp. 243-252
    • Hendriksen, B.A.1
  • 24
    • 0017727218 scopus 로고
    • Estimation of the degree of crystallinity in digoxin by X-ray and infrared methods
    • Black DB, Lovering EG. Estimation of the degree of crystallinity in digoxin by X-ray and infrared methods. J Pharm Pharmacol. 1977;29:684-687.
    • (1977) J Pharm Pharmacol. , vol.29 , pp. 684-687
    • Black, D.B.1    Lovering, E.G.2
  • 25
    • 0031792334 scopus 로고    scopus 로고
    • Comparison of solid-state NMR and isothermal microcalorimetry in the assessment of the amorphous component of lactose
    • Gustafsson C, Lennholm H, Iversen T, Nyström C. Comparison of solid-state NMR and isothermal microcalorimetry in the assessment of the amorphous component of lactose. Int J Pharm. 1998;174:243-252.
    • (1998) Int J Pharm. , vol.174 , pp. 243-252
    • Gustafsson, C.1    Lennholm, H.2    Iversen, T.3    Nyström, C.4
  • 26
    • 0028215092 scopus 로고
    • Assessment of the degree of disorder in crystalline solids by isothermal microcalorimetry
    • Sebhatu T, Angberg M, Ahlneck C. Assessment of the degree of disorder in crystalline solids by isothermal microcalorimetry. Int J Pharm. 1994;104:135-144.
    • (1994) Int J Pharm. , vol.104 , pp. 135-144
    • Sebhatu, T.1    Angberg, M.2    Ahlneck, C.3
  • 28
    • 0036171845 scopus 로고    scopus 로고
    • Cryogenic grinding of indomethacin polymorphs and solvates: Assessment of amorphous phase formation and amorphous phase physical stability
    • Crowley KJ, Zografi G. Cryogenic grinding of indomethacin polymorphs and solvates: assessment of amorphous phase formation and amorphous phase physical stability. J Pharm Sci. 2002;91:492-507.
    • (2002) J Pharm Sci. , vol.91 , pp. 492-507
    • Crowley, K.J.1    Zografi, G.2
  • 29
    • 0032980269 scopus 로고    scopus 로고
    • Differences in crystallisation behaviour between quenched and ground amorphous ursodeoxycholic acid
    • Yonemochi E, Inoue Y, Buckton G, Moffat A, Oguchi T, Yamamoto K. Differences in crystallisation behaviour between quenched and ground amorphous ursodeoxycholic acid. Pharm Res. 1999;16:835-840.
    • (1999) Pharm Res. , vol.16 , pp. 835-840
    • Yonemochi, E.1    Inoue, Y.2    Buckton, G.3    Moffat, A.4    Oguchi, T.5    Yamamoto, K.6
  • 31
    • 0037479923 scopus 로고    scopus 로고
    • Apparent solubility of drugs in partially crystalline systems
    • Mosharraf M, Nyström C. Apparent solubility of drugs in partially crystalline systems. Drug Dev Ind Pharm. 2003;29:603-622.
    • (2003) Drug Dev Ind Pharm. , vol.29 , pp. 603-622
    • Mosharraf, M.1    Nyström, C.2
  • 32
    • 1142303337 scopus 로고    scopus 로고
    • What is the true solubility advantage for amorphous pharmaceuticals?
    • Hancock BC, Parks M. What is the true solubility advantage for amorphous pharmaceuticals? Pharm Res. 2000;17:397-404.
    • (2000) Pharm Res. , vol.17 , pp. 397-404
    • Hancock, B.C.1    Parks, M.2
  • 33
    • 33749431861 scopus 로고    scopus 로고
    • Amorphization of indomethacin by cogrinding with neusilin US2: Amorphization kinetics, physical stability and mechanism
    • Bahl D, Bogner RH. Amorphization of indomethacin by cogrinding with neusilin US2: Amorphization kinetics, physical stability and mechanism. Pharm Res. 2006;23:2317-2325.
    • (2006) Pharm Res. , vol.23 , pp. 2317-2325
    • Bahl, D.1    Bogner, R.H.2
  • 34


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.