Ratiometric Ca+2 measurement in human recombinant muscarinic receptor subtypes using the flexstation scanning fluorometer

Journal of Receptors and Signal Transduction

Volumn 29, Issue 2, 2009, Pages 100-106

  Gupta, Suman ^a   Singh, Rakesh Kumar ^a   Nanda, Kamna ^a   Chatterjee, Mou ^a   Sundaram, Sindhuja ^a   Gupta, Dikshi ^a   Dastidar, Sunanda ^a   Ray, Abhijit ^a  

^a RANBAXY RESEARCH LABORATORIES   (India)

Author keywords

Affinity; Calcium mobilization; Fold selectivity; Muscarinic receptor; Receptor binding

Indexed keywords

ATROPINE; CALCIUM ION; FURA 2 ACETOXYMETHYL ESTER; G PROTEIN COUPLED RECEPTOR; MUSCARINIC M1 RECEPTOR; MUSCARINIC M3 RECEPTOR; MUSCARINIC M5 RECEPTOR; OXYBUTYNIN; RECOMBINANT RECEPTOR; TOLTERODINE; BENZHYDRYL DERIVATIVE; CALCIUM; CRESOL; DRUG DERIVATIVE; FLUORESCENT DYE; FURA 2; FURA-2-AM; MANDELIC ACID DERIVATIVE; MUSCARINIC RECEPTOR BLOCKING AGENT; PHENYLPROPANOLAMINE; SCOPOLAMINE DERIVATIVE;

ANIMAL CELL; ARTICLE; BINDING ASSAY; CALCIUM MOBILIZATION; CHO CELL; CONTROLLED STUDY; DRUG POTENCY; DRUG RECEPTOR BINDING; FLUOROMETER; GENE OVEREXPRESSION; IC 50; NONHUMAN; RADIOASSAY; RECEPTOR AFFINITY; ANIMAL; COMPARATIVE STUDY; CRICETULUS; DRUG ANTAGONISM; FLUORESCENCE; FLUOROMETRY; GENETIC TRANSFECTION; HAMSTER; HUMAN; INSTRUMENTATION; METABOLISM; METHODOLOGY;

ANIMALS; ATROPINE; BENZHYDRYL COMPOUNDS; CALCIUM; CHO CELLS; CRESOLS; CRICETINAE; CRICETULUS; FLUORESCENCE; FLUORESCENT DYES; FLUOROMETRY; FURA-2; HUMANS; MANDELIC ACIDS; MUSCARINIC ANTAGONISTS; PHENYLPROPANOLAMINE; RADIOLIGAND ASSAY; RECEPTOR, MUSCARINIC M1; RECEPTOR, MUSCARINIC M3; RECEPTOR, MUSCARINIC M5; SCOPOLAMINE DERIVATIVES; TRANSFECTION;

EID: 68949190920     PISSN: 10799893     EISSN: 15324281     Source Type: Journal    
DOI: 10.1080/10799890902802634     Document Type: Article

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