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Volumn 20, Issue 4, 2009, Pages 303-311

Penile erection and yawning induced by dopamine D2-like receptor agonists in rats: Influence of strain and contribution of dopamine D2, but not D3 and D4 receptors

Author keywords

Apomorphine; Dopamine D2 receptor; Penile erection; Rats; Yawning

Indexed keywords

2 DIPROPYLAMINO 7 HYDROXYTETRALIN; 3 [[4 (4 CHLOROPHENYL) 1 PIPERAZINYL]METHYL] 1H PYRROLO[2,3 B]PYRIDINE; 3,4,4A,10B TETRAHYDRO 4 PROPYL 2H,5H [1]BENZOPYRANO[4,3 B][1,4]OXAZIN 9 OL; ABT 724; APOMORPHINE; CP 226 269; DOPAMINE 2 RECEPTOR; DOPAMINE 2 RECEPTOR STIMULATING AGENT; DOPAMINE 3 RECEPTOR; DOPAMINE 3 RECEPTOR BLOCKING AGENT; DOPAMINE 4 RECEPTOR; DOPAMINE RECEPTOR BLOCKING AGENT; DOPAMINE RECEPTOR STIMULATING AGENT; L 741626; N [4 (2 CYANOPHENYL) 1 PIPERAZINYLMETHYL] 3 METHYLBENZAMIDE; N [4 [2 (6 CYANO 1,2,3,4 TETRAHYDRO 2 ISOQUINOLINYL)ETHYL]CYCLOHEXYL] 4 QUINOLINECARBOXAMIDE; QUINELORANE; RBI 257; RO 10 5824; S 33084; UNCLASSIFIED DRUG;

EID: 68449090716     PISSN: 09558810     EISSN: None     Source Type: Journal    
DOI: 10.1097/FBP.0b013e32832ec5aa     Document Type: Article
Times cited : (26)

References (39)
  • 2
    • 17944369889 scopus 로고    scopus 로고
    • 3 receptor antagonist SB-277011 in rat, dog and monkey: In vitro/in vivo correlation and the role of aldehydeoxidase
    • 3 receptor antagonist SB-277011 in rat, dog and monkey: in vitro/in vivo correlation and the role of aldehydeoxidase. Xenobiotica 31:677-686.
    • (2001) Xenobiotica , vol.31 , pp. 677-686
    • Austin, N.E.1    Baldwin, S.J.2    Cutler, L.3    Deeks, N.4    Kelly, P.J.5    Nash, M.6
  • 5
  • 6
    • 0033023938 scopus 로고    scopus 로고
    • Intracavernous pressure during erection in rats: Anintegrative approach based on telemetric recording
    • Bernabe J, Rampin O, Sachs BD, Giuliano F (1999). Intracavernous pressure during erection in rats: anintegrative approach based on telemetric recording. Am JPhysiol 276:441-449.
    • (1999) Am JPhysiol , vol.276 , pp. 441-449
    • Bernabe, J.1    Rampin, O.2    Sachs, B.D.3    Giuliano, F.4
  • 8
    • 41649104487 scopus 로고    scopus 로고
    • Commentary on apomorphine versus sildenafil for erectiledysfunction
    • CarsonCC
    • CarsonCC (2008). Commentary on apomorphine versus sildenafil for erectiledysfunction. J Urol 179:S95-96.
    • (2008) J Urol , vol.179
  • 11
    • 68449090705 scopus 로고    scopus 로고
    • 4, receptor in the rat. SanDiego: Society for Neurosciences.710.11.
    • 4, receptor in the rat. SanDiego: Society for Neurosciences.710.11.
  • 13
    • 3142582454 scopus 로고    scopus 로고
    • Discovery of2-(4-pyridin-2-ylpiperazin-1-ylmethyl)-1 H-benzimidazole (ABT-724), adopaminergic agent with a novel mode of action for the potentialtreatment of erectile dysfunction
    • Cowart M, Latshaw SP, Bhatia P, Daanen JF, Rohde J, Nelson SL, et al. (2004). Discovery of2-(4-pyridin-2-ylpiperazin-1-ylmethyl)-1 H-benzimidazole (ABT-724), adopaminergic agent with a novel mode of action for the potentialtreatment of erectile dysfunction. J Med Chem 47:3853-3864.
    • (2004) J Med Chem , vol.47 , pp. 3853-3864
    • Cowart, M.1    Latshaw, S.P.2    Bhatia, P.3    Daanen, J.F.4    Rohde, J.5    Nelson, S.L.6
  • 16
    • 0021181775 scopus 로고
    • The yawningpenile erection syndrome as a model forputative dopamine autoreceptor activity
    • BroekkampCL
    • Gower AJ, Berendsen HG, Princen MM, BroekkampCL (1984). The yawningpenile erection syndrome as a model forputative dopamine autoreceptor activity. Eur J Pharmacol 103:81-89.
    • (1984) Eur J Pharmacol , vol.103 , pp. 81-89
    • Gower, A.J.1    Berendsen, H.G.2    Princen, M.M.3
  • 17
    • 0022550085 scopus 로고
    • Antagonism of drug-induced yawning and penile erections in rats
    • Gower AJ, Berendsen HH, Broekkamp CL (1986). Antagonism of drug-induced yawning and penile erections in rats. Eur J Pharmacol 122:239-244.
    • (1986) Eur J Pharmacol , vol.122 , pp. 239-244
    • Gower, A.J.1    Berendsen, H.H.2    Broekkamp, C.L.3
  • 19
    • 9144229084 scopus 로고    scopus 로고
    • Central mechanismsregulating penile erection in conscious rats: The dopaminergicsystems related to the proerectile effect of apomorphine
    • Hsieh GC, Hollingsworth PR, Martino B, Chang R, Terranova MA, O'Neill AB, et al. (2004). Central mechanismsregulating penile erection in conscious rats: the dopaminergicsystems related to the proerectile effect of apomorphine. JPharmacol Exp Ther 308:330-338.
    • (2004) JPharmacol Exp Ther , vol.308 , pp. 330-338
    • Hsieh, G.C.1    Hollingsworth, P.R.2    Martino, B.3    Chang, R.4    Terranova, M.A.5    O'Neill, A.B.6
  • 26
    • 0034047204 scopus 로고    scopus 로고
    • Millan MJ, Dekeyne A, Rivet JM, Dubuffet T, Lavielle G, Brocco M (2000). S33084, a novel, potent, selective, and competitiveantagonist at dopamine D(3)-receptors: II. Functional and behavioralprofile compared with GR218,231 and L741,626. J Pharmacol ExpTher 293:1063-1073.
    • Millan MJ, Dekeyne A, Rivet JM, Dubuffet T, Lavielle G, Brocco M (2000). S33084, a novel, potent, selective, and competitiveantagonist at dopamine D(3)-receptors: II. Functional and behavioralprofile compared with GR218,231 and L741,626. J Pharmacol ExpTher 293:1063-1073.
  • 27
    • 0036827811 scopus 로고    scopus 로고
    • Differential actions of antiparkinson agents at multiple classes of monoaminergicreceptor. I. A multivariate analysis of the binding profiles of 14drugs at 21 native and cloned human receptor subtypes
    • Millan MJ, Maiofiss L, Cussac D, Audinot V, Boutin JA, Newman-Tancredi A (2002). Differential actions of antiparkinson agents at multiple classes of monoaminergicreceptor. I. A multivariate analysis of the binding profiles of 14drugs at 21 native and cloned human receptor subtypes. J PharmacolExp Ther 303:791-804.
    • (2002) J PharmacolExp Ther , vol.303 , pp. 791-804
    • Millan, M.J.1    Maiofiss, L.2    Cussac, D.3    Audinot, V.4    Boutin, J.A.5    Newman-Tancredi, A.6
  • 28
    • 33846841096 scopus 로고    scopus 로고
    • 2 receptorsenhances frontocortical cholinergic transmission and social memory inrats: A parallel neurochemical and behavioural analysis
    • 2 receptorsenhances frontocortical cholinergic transmission and social memory inrats: a parallel neurochemical and behavioural analysis. JNeurochem 100:1047-1061.
    • (2007) JNeurochem , vol.100 , pp. 1047-1061
    • Millan, M.J.1    Di Cara, B.2    Dekeyne, A.3    Panayi, F.4    De Groote, L.5    Sicard, D.6
  • 29
    • 0017759072 scopus 로고
    • Drugs affecting dopamine neurons and yawning behavior
    • Mogilnicka E, Klimek V (1977). Drugs affecting dopamine neurons and yawning behavior. PharmacolBiochem Behav 7:303-305.
    • (1977) PharmacolBiochem Behav , vol.7 , pp. 303-305
    • Mogilnicka, E.1    Klimek, V.2
  • 34
    • 0033838517 scopus 로고    scopus 로고
    • Pharmacological actions of a novel, high-affinity, and selectivehuman dopamine D(3) receptor antagonist, SB-277011-A
    • Reavill C, Taylor SG, Wood MD, Ashmeade T, Austin NE, Avenell KY, et al. (2000). Pharmacological actions of a novel, high-affinity, and selectivehuman dopamine D(3) receptor antagonist, SB-277011-A. J PharmacolExp Ther 294:1154-1165.
    • (2000) J PharmacolExp Ther , vol.294 , pp. 1154-1165
    • Reavill, C.1    Taylor, S.G.2    Wood, M.D.3    Ashmeade, T.4    Austin, N.E.5    Avenell, K.Y.6
  • 35
    • 0025744944 scopus 로고
    • Effect of apomorphine on penile tumescence inmen with psychogenic impotence
    • Segraves RT, Bari M, Segraves K, Spirnak P (1991). Effect of apomorphine on penile tumescence inmen with psychogenic impotence. J Urol 145:1174-1175.
    • (1991) J Urol , vol.145 , pp. 1174-1175
    • Segraves, R.T.1    Bari, M.2    Segraves, K.3    Spirnak, P.4
  • 37
    • 0034066880 scopus 로고    scopus 로고
    • Design and synthesis oftrans-N-[4-[2-(6-cyano-1,2,3,4- tetrahydroi-soquinolin-2-yl)ethyl]cyclohexyl]-4-quinolinecarboxamide(SB-277011): A potent and selective dopamine D(3) receptor antagonistwith high oral bioavailability and CNS penetration in the rat
    • Stemp G, Ashmeade T, Branch CL, Hadley MS, Hunter AJ, Johnson CN, et al. (2000). Design and synthesis oftrans-N-[4-[2-(6-cyano-1,2,3,4- tetrahydroi-soquinolin-2-yl)ethyl]cyclohexyl]-4-quinolinecarboxamide(SB-277011): a potent and selective dopamine D(3) receptor antagonistwith high oral bioavailability and CNS penetration in the rat. JMed Chem 43:1878-1885.
    • (2000) JMed Chem , vol.43 , pp. 1878-1885
    • Stemp, G.1    Ashmeade, T.2    Branch, C.L.3    Hadley, M.S.4    Hunter, A.J.5    Johnson, C.N.6
  • 38
    • 0026575051 scopus 로고
    • Age-related changes in apomorphine-induced erections
    • Varrin S, Heaton JP (1992). Age-related changes in apomorphine-induced erections. NeurobiolAging 13:175-177.
    • (1992) NeurobiolAging , vol.13 , pp. 175-177
    • Varrin, S.1    Heaton, J.P.2


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