Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: Potential PET imaging agents for tumor detection

Bioorganic and Medicinal Chemistry Letters

Volumn 19, Issue 16, 2009, Pages 4873-4877

  Qiao, Yali ^a   He, Yong ^a   Zhang, Shuting ^a   Li, Guixia ^a   Liu, Hang ^a   Xu, Jingli ^a   Wang, Xiao ^a   Qi, Chuanmin ^a   Peng, Cheng ^b  

^a BEIJING NORMAL UNIVERSITY   (China)

^b CAPITAL MEDICAL UNIVERSITY   (China)

Author keywords

Amino acids; F 18 labeled; Fluoroarylvaline derivatives; PET imaging agents; Tumor detection

Indexed keywords

FLUORINE 18; FLUORODEOXYGLUCOSE F 18; FLUOROVALINE DERIVATIVE; METHYL 2 ( 2 FLUORO 4 NITROBENZAMIDO) 3 METHYLBUTANOIC ACID F 18; O 2 FLUOROETHYLTYROSINE F 18; UNCLASSIFIED DRUG; VALINE;

ANIMAL TISSUE; ARTICLE; BRAIN BLOOD FLOW; CANCER DIAGNOSIS; DIAGNOSTIC VALUE; DOSE TIME EFFECT RELATION; DRUG DISTRIBUTION; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; FEMALE; MOUSE; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; TUMOR BLOOD FLOW;

ANIMALS; BENZAMIDES; BUTYRATES; CELL LINE, TUMOR; FLUORINE RADIOISOTOPES; FLUORODEOXYGLUCOSE F18; MICE; NEOPLASMS; POSITRON-EMISSION TOMOGRAPHY; RADIOPHARMACEUTICALS; TISSUE DISTRIBUTION; TYROSINE;

MUS;

EID: 67651095992     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2009.03.027     Document Type: Article

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