Investigation of β2-adrenoceptor subtype selectivity and organ specificity for bedoradrine (KUR-1246), a novel tocolytic beta-adrenergic receptor stimulant

Journal of Obstetrics and Gynaecology Research

Volumn 35, Issue 3, 2009, Pages 405-413

  Inoue, Yoshihito ^a   Yoshizato, Toshiyuki ^a   Kawarabayashi, Tatsuhiko ^a  

^a FUKUOKA UNIVERSITY   (Japan)

Author keywords

Bedoradrine; Beta adrenergic receptor; Organ specificity; Ritodrine; Tocolytic agent

Indexed keywords

2 [1,2,3,4 TETRAHYDRO 2 [2 HYDROXY 2 [4 HYDROXY 3 (2 HYDROXYETHYL)PHENYL]ETHYLAMINO] 7 NAPHTHYLOXY] N,N DIMETHYLACETAMIDE; BETA 1 ADRENERGIC RECEPTOR; BETA 2 ADRENERGIC RECEPTOR; BETA 3 ADRENERGIC RECEPTOR; CYCLIC AMP; ISOPRENALINE; RITODRINE;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; ASCENDING COLON; CHO CELL; CONTROLLED STUDY; DOSE RESPONSE; DRUG DOSE COMPARISON; DRUG EFFICACY; DRUG SELECTIVITY; DRUG SPECIFICITY; FEMALE; HEART ATRIUM CONTRACTION; IN VIVO STUDY; MUSCLE CONTRACTION; NONHUMAN; NUCLEOTIDE METABOLISM; ORGAN CULTURE TECHNIQUE; PROTEIN EXPRESSION; PROTEIN SYNTHESIS INHIBITION; RAT; TRACHEA; UTERUS;

ACETAMIDES; ANIMALS; CHO CELLS; CRICETINAE; CRICETULUS; CYCLIC AMP; DRUG EVALUATION, PRECLINICAL; FEMALE; MUSCLE CONTRACTION; NAPHTHALENES; OBSTETRIC LABOR, PREMATURE; ORGAN SPECIFICITY; PREGNANCY; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, ADRENERGIC, BETA-2; TOCOLYTIC AGENTS; UTERINE CONTRACTION; UTERUS;

EID: 67650434095     PISSN: 13418076     EISSN: 14470756     Source Type: Journal    
DOI: 10.1111/j.1447-0756.2008.01001.x     Document Type: Article

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