Optimization of peptide-based inhibitors of prostate-specific antigen (PSA) as targeted imaging agents for prostate cancer

Bioorganic and Medicinal Chemistry

Volumn 17, Issue 14, 2009, Pages 4888-4893

  LeBeau, Aaron M ^a   Banerjee, Sangeeta R ^a   Pomper, Martin G ^a,b   Mease, Ronnie C ^a   Denmeade, Samuel R ^a,b  

^a JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE   (United States)

^b JOHNS HOPKINS UNIVERSITY   (United States)

Author keywords

Boronic acid; Chelate; Imaging; Prostate cancer; Prostate specific antigen; Protease inhibitor

Indexed keywords

BORONIC ACID DERIVATIVE; ENZYME INHIBITOR; PEPTIDE DERIVATIVE; PROSTATE SPECIFIC ANTIGEN;

AMINO ACID SUBSTITUTION; ARTICLE; CANCER DIAGNOSIS; ENZYME INHIBITION; HUMAN; POSITRON EMISSION TOMOGRAPHY; PROSTATE CANCER; PROTEIN SYNTHESIS; SINGLE PHOTON EMISSION COMPUTER TOMOGRAPHY;

AMINO ACID SEQUENCE; BORONIC ACIDS; DIAGNOSTIC IMAGING; HUMANS; MALE; PEPTIDE LIBRARY; PEPTIDES; PROSTATE-SPECIFIC ANTIGEN; PROSTATIC NEOPLASMS; SEMEN; SUBSTRATE SPECIFICITY;

EID: 67650067463     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2009.06.012     Document Type: Article

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