메뉴 건너뛰기




Volumn 24, Issue 2, 2009, Pages 209-214

Synthesis and assessment of 99mTc chelate-conjugated alendronate for development of specific radiopharmaceuticals

Author keywords

Biodistribution; Bisphosphonates; Radiochemistry; Scintigraphy

Indexed keywords

3 INDOLECARBALDEHYDE; ALDEHYDE DERIVATIVE; ALENDRONIC ACID TECHNETIUM TC 99M; MEDRONATE TECHNETIUM TC 99M; RADIOPHARMACEUTICAL AGENT; SOLVENT; UNCLASSIFIED DRUG; ALENDRONIC ACID; DIAGNOSTIC AGENT; DRUG DERIVATIVE; INDOLE DERIVATIVE; INDOLE-3-CARBALDEHYDE; TECHNETIUM;

EID: 66249135975     PISSN: 10849785     EISSN: None     Source Type: Journal    
DOI: 10.1089/cbr.2008.0551     Document Type: Article
Times cited : (10)

References (38)
  • 1
    • 0002767351 scopus 로고    scopus 로고
    • Structure and development of the skeleton
    • In: eds. Principles of Bone Biology, ed., San Diego
    • Marks SC, Jr, Odgren PR. Structure and development of the skeleton. In: Bilezikian JP, Raisz LG, Rodan EA, eds. Principles of Bone Biology, 2nd ed., 2-vol set. San Diego: Academic Press, 2002: 3.
    • (2002) Academic Press , vol.2 , Issue.2 , pp. 3
    • Marks, S.C.1    Jr Odgren, P.R.2    Bilezikian, J.P.3    Raisz, L.G.4    Rodan, E.A.5
  • 2
    • 0034284550 scopus 로고    scopus 로고
    • Therapeutic approaches to bone diseases
    • Odgren PR, Martin TJ. Therapeutic approaches to bone diseases. Science 2000; 289: 1508.
    • (2000) Science , vol.289 , pp. 1508
    • Odgren, P.R.1    Martin, T.J.2
  • 3
    • 0030678549 scopus 로고    scopus 로고
    • Osf2/Cbfa1: A transcriptional activator of osteoblast differentiation
    • Ducy P, Zhang R, Geoffroy V, et al. A transcriptional activator of osteoblast differentiation. Cell 1997; 89: 747. (Pubitemid 27516177)
    • (1997) Cell , vol.89 , Issue.5 , pp. 747-754
    • Ducy, P.1    Zhang, R.2    Geoffroy, V.3    Ridall, A.L.4    Karsenty, G.5
  • 5
    • 0032468984 scopus 로고    scopus 로고
    • Bisphosphonates: Mechanisms of action
    • Fleisch H. Bisphosphonates: Mechanisms of action. Endocr Rev 1998; 19: 80. (Pubitemid 29122075)
    • (1998) Endocrine Reviews , vol.19 , Issue.1 , pp. 80-100
    • Fleisch, H.1
  • 6
    • 0028851590 scopus 로고
    • Effect of oral alendronate on bone mineral density and the incidence of fractures in postmenopausal osteoporosis: The Alendronate Phase III Osteoporosis Treatment Study Group
    • Liberman UA, Weiss SR, Broll J, et al. Effect of oral alendronate on bone mineral density and the incidence of fractures in postmenopausal osteoporosis: The Alendronate Phase III Osteoporosis Treatment Study Group. NEMJ 1995; 333: 1437.
    • (1995) NEMJ , vol.333 , pp. 1437
    • Liberman, U.A.1    Weiss, S.R.2    Broll, J.3
  • 8
    • 6844266291 scopus 로고    scopus 로고
    • Alendronate prevents postmenopausal bone loss in women without osteoporosis: A double-blind randomized, controlled trial. Alendronate Osteoporosis Prevention Study Group
    • McClung M, Clemmesen B, Daifotis A, et al. Alendronate prevents postmenopausal bone loss in women without osteoporosis: A double-blind randomized, controlled trial. Alendronate Osteoporosis Prevention Study Group. Ann Intern Med 1998; 128: 253.
    • (1998) Ann Intern Med , vol.128 , pp. 253
    • McClung, M.1    Clemmesen, B.2    Daifotis, A.3
  • 10
    • 0028846051 scopus 로고
    • Effects of oral alendronate and intranasal salmon calcitonin on bone mass and biochemical markers of bone turnover in postmenopausal women with osteoporosis
    • Adami S, Passeri M, Orolani S, et al. Effects of oral alendronate and intranasal salmon calcitonin on bone mass and biochemical markers of bone turnover in postmenopausal women with osteoporosis. Bone 1995; 17: 383.
    • (1995) Bone , vol.17 , pp. 383
    • Adami, S.1    Passeri, M.2    Orolani, S.3
  • 11
    • 0029116697 scopus 로고
    • Alendronate treatment of the postmenopausal osteoporotic woman: Effect of multiple dosages on bone mass and bone remodeling
    • Chesnut CH, McClung MR, Ensrud KE, et al. Alendronate treatment of the postmenopausal osteoporotic woman: Effect of multiple dosages on bone mass and bone remodeling. Am J Med 1995; 99: 144.
    • (1995) Am J Med , vol.99 , pp. 144
    • Chesnut, C.H.1    McClung, M.R.2    Ensrud, K.E.3
  • 14
    • 0031006598 scopus 로고    scopus 로고
    • Prevention of nonvertebral fractures by alendronate: A meta-analysis. the Alendronate Osteoporosis Treatment Study Groups
    • Karpf DB, Shapiro DR, Seeman E, et al. Prevention of nonvertebral fractures by alendronate: A meta-analysis. The Alendronate Osteoporosis Treatment Study Groups. JAMA 1997; 277: 1159.
    • (1997) JAMA , vol.277 , pp. 1159
    • Karpf, D.B.1    Shapiro, D.R.2    Seeman, E.3
  • 17
    • 0017891632 scopus 로고
    • Uptake by bone of pyrophosphate, diphosphonates and their technetium derivatives
    • Bisaz S, Jung A, Fleisch H. Uptake by boul of pyrophosphate, diphosphonates, and their technetium derivatives. Clin Sci Mol Med 1978; 54; 265. (Pubitemid 8286494)
    • (1978) Clinical Science and Molecular Medicine , vol.54 , Issue.3 , pp. 265-272
    • Bisaz, S.1    Jung, A.2    Fleisch, H.3
  • 18
    • 0015939609 scopus 로고
    • The binding of pyrophosphate and two diphosphonates by hydroxyapatite crystals
    • Jung A, Bisaz S, Fleisch H. The binding of pyrophosphate and two diphosphonates by hydroxyapatite crystals. Calcif Tissue Res 1973; 11: 269.
    • (1973) Calcif Tissue Res , vol.11 , pp. 269
    • Jung, A.1    Bisaz, S.2    Fleisch, H.3
  • 19
    • 0016262325 scopus 로고
    • 99mTc-polyphosphate
    • 99mTc-polyphosphate. Nucl Med 1974; 15: 1057.
    • (1974) Nucl Med , vol.15 , pp. 1057
    • Richards, A.G.J.1
  • 20
    • 0026064309 scopus 로고
    • Pamidronate: A review of its pharmacological properties and therapeutic efficacy in resorptive bone disease
    • Fitton A, McTavish D. Pamidronate: A review of its pharmacological properties and therapeutic efficacy in resorptive bone disease. Drugs 1991; 41: 289. (Pubitemid 121000771)
    • (1991) Drugs , vol.41 , Issue.2 , pp. 289-318
    • Fitton, A.1    McTavish, D.2
  • 21
    • 0019214294 scopus 로고
    • Comparative evaluation of three diphosphonates: In vitro adsorption (C-14 labeled) and in vivo osteogenic uptake (Tc-99m complexed)
    • Francis MD, Ferguson DL, Tofe AJ, et al. Comparative evaluation of three diphosphonates: In-vitro adsorption (C- 14 labeled) and in-vivo osteogenic uptake (Tc-99m complexed). Nucl Med 1980; 21: 1185. (Pubitemid 11196766)
    • (1980) Journal of Nuclear Medicine , vol.21 , Issue.12 , pp. 1185-1189
    • Francis, M.D.1    Ferguson, D.L.2    Tofe, A.J.3
  • 26
    • 7544241450 scopus 로고    scopus 로고
    • Complexes of divalent transitional met al.s with bis (amino methyl) phosphonic acid in aqueous solution and in solid state
    • Kubicek V, Vojtísek P, Rudovsky J, et al. Complexes of divalent transitional met al.s with bis (amino methyl) phosphonic acid in aqueous solution and in solid state. Dalton Trans 2003; 20: 3927.
    • (2003) Dalton Trans , vol.20 , pp. 3927
    • Kubicek, V.1    Vojtiacute2    Sek, P.3    Rudovsky, J.4
  • 27
    • 0017106182 scopus 로고
    • 99mTc-labeled phosphate and phosphonate agents for skelet al. imaging
    • 99mTc-labeled phosphate and phosphonate agents for skelet al. imaging. Semin Nucl Med 1976; 6: 19.
    • (1976) Semin Nucl Med , vol.6 , pp. 19
    • Davis, M.1    Jones, A.G.2
  • 30
    • 0020585468 scopus 로고
    • 99mTc-DPD, and 99mTc-HDP for the detection of bone metastases
    • 99mTc-DPD, and 99mTc-HDP for the detection of bone metastases. Eur J Nucl Med 1983; 8: 118.
    • (1983) Eur J Nucl Med , vol.8 , pp. 118
    • Pauwels, E.K.1    Blom, J.2    Camps, J.A.3
  • 31
    • 0020972241 scopus 로고
    • A clinical comparison of Tc- 99m DPD and two Tc-99m MDP agents
    • Vorne M, Vahatalo S, Lantto T. A clinical comparison of Tc- 99m DPD and two Tc-99m MDP agents. Eur J Nucl Med 1983; 8: 395.
    • (1983) Eur J Nucl Med , vol.8 , pp. 395
    • Vorne, M.1    Vahatalo, S.2    Lantto, T.3
  • 32
    • 0001719707 scopus 로고    scopus 로고
    • Rhenium-188 hydroxyethylidene diphosphonate: A new generator-produced radiotherapeutic drug of potential value for the treatment of bone metastases
    • Lin WY, Lin CP, Yeh SJ, et al. Rhenium-188 hydroxyethylidene diphosphonate: A new generator-produced radiotherapeutic drug of potential value for the treatment of bone metastases. Eur J Nucl Med 1997; 24: 590.
    • (1997) Eur J Nucl Med , vol.24 , pp. 590
    • Lin, W.Y.1    Lin, C.P.2    Yeh, S.J.3
  • 33
    • 0023228018 scopus 로고
    • Skeletal localization of samarium-153 chelates: Potential therapeutic bone agents
    • Goeckeler WF, Edwards B, Volkert WA, et al. Skelet al. localization of samarium-153 chelates: Potential therapeutic bone agents. J Nucl Med 1987; 28: 495. (Pubitemid 17074172)
    • (1987) Journal of Nuclear Medicine , vol.28 , Issue.4 , pp. 495-504
    • Goeckeler, W.F.1    Edwards, B.2    Volkert, W.A.3
  • 34
    • 0035176708 scopus 로고    scopus 로고
    • The palliative management of skeletal metastases in prostate cancer: Use of bone-seeking radionuclides and bisphosphonates
    • Hamdy NA, Papapoulos SE. The palliative management of skelet al. metastases in prostate cancer: Use of bone-seeking radionuclides and bisphosphonates. Semin Nucl Med 2001; 31: 62. (Pubitemid 32060653)
    • (2001) Seminars in Nuclear Medicine , vol.31 , Issue.1 , pp. 62-68
    • Hamdy, N.A.T.1    Papapoulos, S.E.2
  • 35
    • 0001575017 scopus 로고
    • Pharmacokinetics of rhenium-186 after administration of Re-186-HEDP to patients with bone metastases
    • De Klerk JMH, Van Dijk A, Van Rijk PP, et al. Pharmacokinetics of rhenium-186 after administration of Re-186-HEDP to patients with bone metastases. Nucl Med 1991; 32: 1082.
    • (1991) Nucl Med , vol.32 , pp. 1082
    • De Klerk, J.M.H.1    Van Dijk, A.2    Van Rijk, P.P.3
  • 36
    • 0023875466 scopus 로고
    • Re-186 (Sn) HEDP for treatment of multiple metastatic foci in bone: Human biodistribution and dosimetric studies [published erratum appears in Radiology]
    • III
    • Maxon HR, III, Deutsch EA, Thomas SR, et al. Re-186 (Sn) HEDP for treatment of multiple metastatic foci in bone: Human biodistribution and dosimetric studies [published erratum appears in Radiology]. Radiology 1988; 166: 501.
    • (1988) Radiology , vol.166 , pp. 501
    • Maxon, H.R.1    Deutsch, E.A.2    Thomas, S.R.3
  • 37
    • 38149007203 scopus 로고    scopus 로고
    • Synthesis, characterization, and biological activiy of Schiff base analogues of indole-3-carboxaldehyde
    • Sinha D, Tiwari AK, Singh S, et al. Synthesis, characterization, and biological activiy of Schiff base analogues of indole-3-carboxaldehyde. Eur J Med Chem 2007; 43: 160.
    • (2007) Eur J Med Chem , vol.43 , pp. 160
    • Sinha, D.1    Tiwari, A.K.2    Singh, S.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.