Design and synthesis of novel delta opioid receptor agonists and their pharmacologies

Bioorganic and Medicinal Chemistry Letters

Volumn 19, Issue 10, 2009, Pages 2792-2795

  Nagase, Hiroshi ^a   Osa, Yumiko ^a   Nemoto, Toru ^a   Fujii, Hideaki ^a   Imai, Masayuki ^b   Nakamura, Takashi ^b   Kanemasa, Toshiyuki ^b   Kato, Akira ^b   Gouda, Hiroaki ^a   Hirono, Shuichi ^a  

^a KITASATO UNIVERSITY   (Japan)

^b SHIONOGI AND CO LTD   (Japan)

Author keywords

Receptor; Analgesics; Naltrexone; Opioid

Indexed keywords

1,2,3,4,4A,5,12,12AALPHA OCTAHYDRO 4AALPHA (3 HYDROXYPHENYL) 2 METHYLQUINOLINO[2,3 G]ISOQUINOLINE; DELTA OPIATE RECEPTOR AGONIST; SN 11; SN 23; SN 28; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; DRUG CONFORMATION; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS;

DRUG DESIGN; MORPHINANS; NALTREXONE; RECEPTORS, OPIOID, DELTA;

EID: 65349183593     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2009.03.099     Document Type: Article

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