Melting of nanostructured drugs embedded into a polymeric matrix

Journal of Physical Chemistry B

Volumn 108, Issue 40, 2004, Pages 15488-15493

  Bergese, P ^a   Colombo, I ^b   Gervasoni, D ^b   Depero, Laura E ^a  

^a UNIVERSITY OF BRESCIA   (Italy)

^b Eurand SpA   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

ABSORPTION; CRYSTAL STRUCTURE; CRYSTALLINE MATERIALS; DIFFUSION; MICROSTRUCTURE; MOLECULAR DYNAMICS; NANOSTRUCTURED MATERIALS; PHASE TRANSITIONS; THERMODYNAMICS; X RAY DIFFRACTION ANALYSIS;

MOLECULAR DIFFUSION; NANOCRYSTALS; NANOSTRUCTURED DRUGS; POLYMERIC MATRIX; THERMODYNAMIC MELTING MODEL;

DRUG DOSAGE;

EID: 6444239981     PISSN: 15206106     EISSN: None     Source Type: Journal    
DOI: 10.1021/jp048762u     Document Type: Article

References (68)

1. Devane, J. Pharm. Technol. 1998, Nov., 68.
2. Waiver of in vivo bioavailability and bioequtvalence studies for immaediate-release solid oral dosage forms based on a biopharmacutics classification system, U.S. Department of Health and Human Services, Food and Drug Administration, Center for Drug Evaluation and Research: Washington, DC, 2000. Also available at: http://www.fda.gov/cder/guidance/index.htm.
3. Amidon, G. L.; Lennearnas, H.; Shah, V. P.; Crison, R. Pharm. Res. 1995, 12, 413.
4. Hsia, D. C.; Kim, C. K.; Kildsig, D. O. J. Pharm. Sci. 1977, 66, 961.
5. Bergese, P. Ph.D. Thesis, Pharmaceutical nanocomposites generated by microwave induced diffusion. Università degli studi di Brescia: Brescia, Italy, 2002; pp 12-19.
6. Zhao, M.; Zhou, X. H.; Jiang, Q. J. Mater. Res. 2001, 16, 3304.
7. Liang, L. H.; Zhao, M.; Jiang, Q. J. Mater. Sci. Lett 2002, 21, 1843.
8. Liu, R., Ed. Water-Insoluble Drug Formulation; Interpharm Press: Denver, CO, 2000.
9. Carli, F.; Colombo, I.; Magarotto, L. In 13th International Symposium on controlled release of bioactive materials; Nortfolk, Chaudy, I., Ed.; The Controlled Release Society: Minneapolis, MN, 1986; p 193.
10. Carli, F.; Colombo, I. Acta Pharm. Jugosl. 1988, 38, 361.
11. Button, G.; Beezer, A. E. Int. J. Pharm. 1992, 82, R7.
12. Mosharraf, M.; Sebhatu, T.; Nystrom, C. Int. J. Pharm. 1999, 777, 29.
13. Burt, H. M.; Mitchell, A. O. Int. J. Pharm. 1981, 9, 137.
14. Allen, G. L.; Gile, W. W.; Jesser, W. A. Acta Metall. 1980, 28, 1695.
15. Shi, F. G. J. Mater. Res. 1994, 9, 1307.
16. Lu, K.; Jin, Z. H. Curr. Opin. Solid State. Mater. 2001, 5, 39.
17. Sanz, N.; Boudet, A.; Ibanez, A. J. Nanop. Res. 2002, 4, 99.
18. Takagi, M. J. Phys. Soc. Jpn. 1954, 9, 359.
19. Couchman, P. R.; Jesser, W. A. Nature (London) 1977, 269, 481.
20. Lu, K.; Sui, M. L. Acta Metall. Mater. 1995, 43, 3325.
21. Peters, K. F.; Cohen, J. B.; Chung, Y. W. Phys. Rev. B 1998, 57, 13430.
22. Sheng, H. W.; Lu, K.; Ma, E. Acta Mater. 1998, 46, 5195.
23. Zhang, M.; Efremov, M. Y.; Schiettekatte, F.; Olson, E. A.; Kwan, A. T.; Lai, S. L.; Wisleder, T.; Greene, J. E.; Allen, L. H. Phys. Rev. B 2000, 62, 10548.
24. Bottani, C. E.; Li Bassi, A.; Stella, A.; Cheyssac, P.; Kofman, R. Europhys. Lett. 2001, 56, 386.
25. Liang, L. H.; Li, J. C.; Jiang, Q. Physica B 2003, 334, 49.
26. Depero, L. E.; Bontempi, E.; Sangaletti, L.; Pagliara, S. J. Chem. Phys. 2003, 118, 1400.
27. Goldstain, A. N.; Echer, C. M.; Alivisatos. A. P. Science 1992, 256, 1425.
28. Zhang, Z.; Zhao, M.; Jiang, Q. Semicond. Sci. Technol. 2001, 16, L33.
29. Liang, L. H.; Li, J. C.; Jiang. Q. Phys. Status Solidi B 2003, 236, 583.
30. Jackson. C. L.; McKenna, G. B. J. Chem. Phys. 1990, 93, 9002.
31. Zhang, J.; Liu, G.; Jonas, J. J. Phys. Chem. 1992, 96, 3478.
32. Jiang, Q.; Shi, H. X.; Zhao, M. J. Chem. Phys. 1999, 111, 2176.
33. Sliwinska-Bartkowiak, M.; Dudziak, G.; Sikorski, R.; Gras, R. J. Chem. Phys. 2001, 114, 950.
34. Rottele, A.; Thurn-Albrecht, T.; Sommer, J. U.; Reiter, G. Macromolecules 2003, 36, 1257.
35. Handa, Y. P.; Zakrzewski, M.; Fairbridge, C. J. Phys. Chem. 1992, 96, 8594.
36. Brun, M.; Lallemand, A.; Quinson, J. F.; Eyraud, C. J. Chim. Phys. 1973, 70, 979.
37. Brun, M.; Lallemand, A.; Quinson, J. F.; Eyraud, C. Thermochim. Acta 1977, 21, 59.
38. Homshaw, L. G. J. Colloid Interface Sci. 1981, 84, 141.
39. Ishikiriyama, K.; Todoki, M.; Min, K. H.; Yonemori, S.; Noshiro, M. J. Therm. Anal. 1996, 46, 1177.
40. Adamson, A. W.; Gast, A. P. Physical Chemistry of Surfaces; Wiley: New York, 2000.
41. Bertsch, G. Science 1997, 277, 1619.
42. Zhao, S. J.; Wang, S. Q.; Cheng, D. Y.; Ye, H. Q. J. Phys. Chem. B 2001, 105, 12857.
43. Cheng, H. P.; Berry, R. S. Phys. Rev. A. 1992, 45, 7969.
44. Huang, S. P.; Balbuena, P. B. J. Phys. Chem. B 2002, 106, 7225.
45. Rastogi, S.; Zakrzewski, M.; Suryanarayanan, R. Pharm. Res. 2001, 18. 267.
46. Rastogi, S.; Zakrzewski, M.; Suryanarayanan, R. Pharm. Res. 2002, 19. 1265.
47. Bergese, P.; Colombo, I.; Gervasoni, D.; Depero, L. E. J. Appl. Crystallogr. 2003, 36, 74.
48. Lovrecich, M. Supported drugs with increased dissolution rate, and a process for their preparation. US Patent 5 449 521, 1995.
49. Dobetti, L.; Cadelli, G.; Furlani, D.; Zotti, M.; Ceschia, D.; Grassi, M. Proc. 28th Int. Symp. Contr. Relat. Bioact. Mater. 2001, 6059.
50. Meriani, F.; Coceani, N.; Sirotti, C.; Voinovich, D.; Grassi, M. J. Pharm. Sci. 2004, 93, 540.
51. Grassi, M. Proc. AAPS Conf. Phanna. Drug Deliv. 2004.
52. Alexander, L.; Klug, H. P. Anal. Chem. 1948, 20, 886.
53. Yu, L. Adv. Drug Del. Rew 2001, 48, 27.
54. Craig, D. Q. M.; Kett, V. L.; Murphy, J. R.; Price, D. M. Pharm. Res. 2001, 75, 1081.
55. Boutonnet-Fagegaltier, N.; Menegotto, J.; Lamure, A.; Duplaa, H.; Caron, A.; Lacabanne, C.; Bauer, M. J. Pharm. Sci. 2002, 91, 1548.
56. Saito, Y.; Saito, K.; Atake, T. Themochim. Acta 1986, 107, 279.
57. Sauders, M.; Podluii, K.; Shergill, S.; Bukton, G.; Royall, P. Int. J. Pharm. 2004, 274, 35.
58. Theeuwes, F.; Hussain, A.; Higuchi, T. J. Pharm. Sci. 1974, 63, 427.
59. Balzar, D. In Voight-function model in diffraction line-broadening ananlysis; in Defect and Microstructure analysis by diffraction; Snyder, R. L., Bunge, H. J., Fiala, J.; Eds.; International Union of Crystallography, Oxford University Press: New York, 1999.
60. Cheary, R. W.; Coelho, A. A. J. Appl. Crystallogr. 1992, 25, 109.
61. Bruker AXS; TOPAS V2.0: General profile and structure ananlysis software for powder diffraction data; User manual, Bruker AXS: Karlsruhe, Germany, 2000.
62. Enzo, S.; Fagherazzi, F.; Benedetti, A.; Polizzi, S. J. Appl. Crystallogr. 1988, 21, 536.
63. Delogu, F.; Cocco, G. J. Mater. Synth. Process. 2000, 8, 271.
64. Fedors, R. F. Polym. Eng. Sci. 1974, 14, 147.
65. Wu, S. J. Polym. Sci. C 1971, 34, 19.
66. Van Krevelen, D. W. Properties of polymers; Elsevier Science: Amsterdam, 1997.
67. Langford, J. I.; Louer, D.; Scardi, P. J. Appl. Crystallogr. 2000, 33, 964.
68. Balzar, D. Report on the first size-strain round-robin of CPD; IUCr; http://www.boulder.nist.gov/div853/balzar/s - s_rr.htm.