-
1
-
-
0019236427
-
Medicinal chemistry of tetrazoles
-
(a) Singh, H.; Chawla, A. S.; Kapoor, V. K.; Paul, D.; Malhotra, R. K. Medicinal chemistry of tetrazoles. Prog. Med. Chem. 1980, 17, 151;
-
(1980)
Prog. Med. Chem
, vol.17
, pp. 151
-
-
Singh, H.1
Chawla, A.S.2
Kapoor, V.K.3
Paul, D.4
Malhotra, R.K.5
-
2
-
-
0014233779
-
Preparation and antiinflammatory properties of some 5-(2-anilinophenyl)tetrazoles
-
(b) Juby, P. F.; Hudyma, T. W.; Brown, M. Preparation and antiinflammatory properties of some 5-(2-anilinophenyl)tetrazoles. J. Med. Chem. 1968, 11, 111-117.
-
(1968)
J. Med. Chem
, vol.11
, pp. 111-117
-
-
Juby, P.F.1
Hudyma, T.W.2
Brown, M.3
-
3
-
-
33748832377
-
Ring transformations in tetrazole chemistry
-
Moderhack, D. Ring transformations in tetrazole chemistry. J. Prakt. Chem. 1998, 340, 687-709.
-
(1998)
J. Prakt. Chem
, vol.340
, pp. 687-709
-
-
Moderhack, D.1
-
4
-
-
84884197352
-
Recent development in tetrazole chemistry: A review
-
(a) Wittenberger, S. J. Recent development in tetrazole chemistry: A review. Org. Prep. Proced. Int. 1994, 26, 499-531;
-
(1994)
Org. Prep. Proced. Int
, vol.26
, pp. 499-531
-
-
Wittenberger, S.J.1
-
5
-
-
33750689149
-
Discovery and in vitro=in vivo studies of tetrazole derivatives as Kv1.5 blockers
-
(b) Wu, S.; Fluxe, A.; Sheffer, J.; Janusz, J. M.; Blass, B. E.; White, R.; Jackson, C.; Hedges, R.; Muawsky, M.; Fang, B.; Fadayel, G. M.; Hare, M.; Djandjighian, L. Discovery and in vitro=in vivo studies of tetrazole derivatives as Kv1.5 blockers. Bioorg. Med. Chem. Lett. 2006, 16, 6213-6218;
-
(2006)
Bioorg. Med. Chem. Lett
, vol.16
, pp. 6213-6218
-
-
Wu, S.1
Fluxe, A.2
Sheffer, J.3
Janusz, J.M.4
Blass, B.E.5
White, R.6
Jackson, C.7
Hedges, R.8
Muawsky, M.9
Fang, B.10
Fadayel, G.M.11
Hare, M.12
Djandjighian, L.13
-
6
-
-
0037171833
-
Investigation of potential bioisosteric replacements for the carboxyl groups of peptidomimetic inhibitors of protein tyrosine phosphatase 1B: Identification of a tetrazole-containing inhibitor with cellular activity
-
(c) Liljebris, C.; Larsen, S. D.; Ogg, D.; Palazuk, B. J.; Bleasdale, J. E. Investigation of potential bioisosteric replacements for the carboxyl groups of peptidomimetic inhibitors of protein tyrosine phosphatase 1B: Identification of a tetrazole-containing inhibitor with cellular activity. J. Med. Chem. 2002, 45, 1785-1798.
-
(2002)
J. Med. Chem
, vol.45
, pp. 1785-1798
-
-
Liljebris, C.1
Larsen, S.D.2
Ogg, D.3
Palazuk, B.J.4
Bleasdale, J.E.5
-
7
-
-
11844253794
-
Organocatalysis with proline derivatives: Improved catalysts for the asymmetric Mannich, nitro-Michael, and aldol reactions
-
(a) Cobb, A. J. A.; Shaw, D. M.; Longbottom, D. A.; Gold, J. B.; Ley, S. V. Organocatalysis with proline derivatives: improved catalysts for the asymmetric Mannich, nitro-Michael, and aldol reactions. Org. Biomol. Chem. 2005, 3, 84-96;
-
(2005)
Org. Biomol. Chem
, vol.3
, pp. 84-96
-
-
Cobb, A.J.A.1
Shaw, D.M.2
Longbottom, D.A.3
Gold, J.B.4
Ley, S.V.5
-
8
-
-
33746157422
-
Expedient synthesis of chiral 1,2- and 1,4-diamines: Protecting group dependent regioselectivity in direct organocatalytic asymmetric Mannich reactions
-
(b) Chowdari, N. S.; Ahmad, M.; Albertshofer, K.; Tanaka, F.; Barbas, III. C. F. Expedient synthesis of chiral 1,2- and 1,4-diamines: Protecting group dependent regioselectivity in direct organocatalytic asymmetric Mannich reactions. Org. Lett. 2006, 8, 2839-2842.
-
(2006)
Org. Lett
, vol.8
, pp. 2839-2842
-
-
Chowdari, N.S.1
Ahmad, M.2
Albertshofer, K.3
Tanaka, F.4
Barbas III, C.F.5
-
10
-
-
0010604237
-
Synthesis of iminotetrazoline derivatives as trichomonacidal and fungicidal agents
-
(b) Herbst, R. M.; Froberger, C. F. Synthesis of iminotetrazoline derivatives as trichomonacidal and fungicidal agents. J. Org. Chem. 1957, 22, 1050-1053.
-
(1957)
J. Org. Chem
, vol.22
, pp. 1050-1053
-
-
Herbst, R.M.1
Froberger, C.F.2
-
11
-
-
0034680614
-
Fast microwave-assisted preparation of aryl and vinyl nitriles and the corresponding tetrazoles from organo-halides
-
(a) Alterman, M.; Hallberg, A. Fast microwave-assisted preparation of aryl and vinyl nitriles and the corresponding tetrazoles from organo-halides. J. Org. Chem. 2000, 65, 7984-7989;
-
(2000)
J. Org. Chem
, vol.65
, pp. 7984-7989
-
-
Alterman, M.1
Hallberg, A.2
-
12
-
-
0010114968
-
An improved synthesis of 5-substituted tetrazoles
-
(b) Finnegan, W. G.; Henry, R. A.; Lofquist, R. An improved synthesis of 5-substituted tetrazoles. J. Am. Chem. Soc. 1958, 80, 3908-3911;
-
(1958)
J. Am. Chem. Soc
, vol.80
, pp. 3908-3911
-
-
Finnegan, W.G.1
Henry, R.A.2
Lofquist, R.3
-
13
-
-
0023620309
-
Improved conditions for the formation of tetrazoles
-
(c) Bernstein, P. R.; Vacek, E. P. Improved conditions for the formation of tetrazoles. Synthesis 1987, 1133-1134.
-
(1987)
Synthesis
, pp. 1133-1134
-
-
Bernstein, P.R.1
Vacek, E.P.2
-
14
-
-
0017334524
-
Studies on antianaphylactic agents, 5: Synthesis of 3-(1H-tetrazol-5-yl) chromones, a new series of antiallergic substances
-
(a) Nohara, A.; Kuriki, H.; Saijo, T.; Sugihara, H.; Kanno, M.; Sanno, Y. Studies on antianaphylactic agents, 5: Synthesis of 3-(1H-tetrazol-5-yl) chromones, a new series of antiallergic substances. J. Med.Chem. 1977, 20, 141-145;
-
(1977)
J. Med.Chem
, vol.20
, pp. 141-145
-
-
Nohara, A.1
Kuriki, H.2
Saijo, T.3
Sugihara, H.4
Kanno, M.5
Sanno, Y.6
-
15
-
-
1842688821
-
TBAF-catalyzed synthesis of 5-substituted 1H-tetrazoles under solventless conditions
-
(b) Amantini, D.; Beleggia, R.; Fringuelli, F.; Pizzo, F.; Vaccaro, L. TBAF-catalyzed synthesis of 5-substituted 1H-tetrazoles under solventless conditions. J. Org. Chem. 2004, 69, 2896-2898;
-
(2004)
J. Org. Chem
, vol.69
, pp. 2896-2898
-
-
Amantini, D.1
Beleggia, R.2
Fringuelli, F.3
Pizzo, F.4
Vaccaro, L.5
-
16
-
-
14844344119
-
Efficient syntheses of 5-aminoalkyl-1H-tetrazoles and of polyamines incorporating tetrazole rings
-
(c) Athanassopoulos, C. M.; Garnelis, T.; Vahliotis, D.; Papaioannou, D. Efficient syntheses of 5-aminoalkyl-1H-tetrazoles and of polyamines incorporating tetrazole rings. Org. Lett. 2005, 7, 561-564.
-
(2005)
Org. Lett
, vol.7
, pp. 561-564
-
-
Athanassopoulos, C.M.1
Garnelis, T.2
Vahliotis, D.3
Papaioannou, D.4
-
17
-
-
0000096835
-
Click chemistry: Diverse chemical function from a few good reactions
-
Kolb, H. C.; Finn, M. G.; Sharpless, K. B. Click chemistry: diverse chemical function from a few good reactions. Angew. Chem. Int. Ed. 2001, 40, 2004-2021.
-
(2001)
Angew. Chem. Int. Ed
, vol.40
, pp. 2004-2021
-
-
Kolb, H.C.1
Finn, M.G.2
Sharpless, K.B.3
-
18
-
-
0038042134
-
An expedient route to the tetrazole analogues of a-amino acids
-
Demko, Z. P.; Sharpless, K. B. An expedient route to the tetrazole analogues of a-amino acids. Org. Lett. 2002, 4, 2525-2527.
-
(2002)
Org. Lett
, vol.4
, pp. 2525-2527
-
-
Demko, Z.P.1
Sharpless, K.B.2
-
19
-
-
34548354905
-
Synthesis of tetrazole analogues of amino acids using Fmoc chemistry: Isolation of amino free tetrazoles and their incorporation into peptides
-
Sureshbabu, V. V.; Venkataramanarao, R.; Naik, S. A.; Chennakrishnareddy, G. Synthesis of tetrazole analogues of amino acids using Fmoc chemistry: Isolation of amino free tetrazoles and their incorporation into peptides. Tetrahedron Lett. 2007, 48, 7038-7041.
-
(2007)
Tetrahedron Lett
, vol.48
, pp. 7038-7041
-
-
Sureshbabu, V.V.1
Venkataramanarao, R.2
Naik, S.A.3
Chennakrishnareddy, G.4
-
20
-
-
0001081264
-
Tetrazole analogues of amino acids and peptides, part I: Preparation of tetrazole analogues of amino acids from amino acids
-
(a) Grzonka, Z.; Liberek, B. Tetrazole analogues of amino acids and peptides, part I: Preparation of tetrazole analogues of amino acids from amino acids. Roczniki Chem. 1971, 45, 967-980;
-
(1971)
Roczniki Chem
, vol.45
, pp. 967-980
-
-
Grzonka, Z.1
Liberek, B.2
-
21
-
-
0010567592
-
Tetrazole analogues of amino acids and peptides, V: Synthesis of peptide derivatives containing tetrazoles analogues of amino acids in C-terminal position
-
(b) Grzonka, Z.; Rekowska, E.; Liberek, B. Tetrazole analogues of amino acids and peptides, V: Synthesis of peptide derivatives containing tetrazoles analogues of amino acids in C-terminal position. Tetrahedron 1971, 27, 2317-2322.
-
(1971)
Tetrahedron
, vol.27
, pp. 2317-2322
-
-
Grzonka, Z.1
Rekowska, E.2
Liberek, B.3
-
22
-
-
0027524045
-
Tetrazole amino acids as competitive NMDA antagonists
-
Ornstein, P. L.; Arnold, M. B.; Evrard, D.; Leander, J. D.; Lodge, D.; Darryle, D. Tetrazole amino acids as competitive NMDA antagonists. Bioorg. Med. Chem. Lett. 1993, 3, 43-48.
-
(1993)
Bioorg. Med. Chem. Lett
, vol.3
, pp. 43-48
-
-
Ornstein, P.L.1
Arnold, M.B.2
Evrard, D.3
Leander, J.D.4
Lodge, D.5
Darryle, D.6
-
23
-
-
0029076025
-
Activation of carboxylic acids by pyrocarbonates: Application of di-tert-butyl pyrocarbonate as condensing agent in the synthesis of amides of protected amino acids and peptides
-
Pozdnev, V. F. Activation of carboxylic acids by pyrocarbonates: Application of di-tert-butyl pyrocarbonate as condensing agent in the synthesis of amides of protected amino acids and peptides. Tetrahedron Lett. 1995, 36, 7115-7118.
-
(1995)
Tetrahedron Lett
, vol.36
, pp. 7115-7118
-
-
Pozdnev, V.F.1
-
24
-
-
0000355144
-
A convenient synthesis of versatile side-chain intermediates for carbapenem antibiotics
-
Kawamoto, I.; Endo, R.; Ishikawa, K.; Kojima, K.; Miyauchi, M.; Nakayama, E. A convenient synthesis of versatile side-chain intermediates for carbapenem antibiotics. Synlett 1995, 575-577.
-
(1995)
Synlett
, pp. 575-577
-
-
Kawamoto, I.1
Endo, R.2
Ishikawa, K.3
Kojima, K.4
Miyauchi, M.5
Nakayama, E.6
-
25
-
-
0345508076
-
A convenient synthesis of nitriles from primary amides under mild conditions
-
(a) Campagna, F.; Carotti, A.; Casini, G. A convenient synthesis of nitriles from primary amides under mild conditions. Tetrahedron Lett. 1977, 21, 1813-1816;
-
(1977)
Tetrahedron Lett
, vol.21
, pp. 1813-1816
-
-
Campagna, F.1
Carotti, A.2
Casini, G.3
-
26
-
-
0030972839
-
A simple preparation of N-protected chiral α-aminonitriles from N-protected α-amino acid amides
-
(b) Maetz, P.; Rodriguez, M. A simple preparation of N-protected chiral α-aminonitriles from N-protected α-amino acid amides. Tetrahedron Lett. 1997, 38, 4221-4222;
-
(1997)
Tetrahedron Lett
, vol.38
, pp. 4221-4222
-
-
Maetz, P.1
Rodriguez, M.2
-
27
-
-
0000223138
-
An efficient chemoselective synthesis of nitriles from primary amides
-
(c) Claremon, D. A.; Phillips, B. T. An efficient chemoselective synthesis of nitriles from primary amides. Tetrahedron Lett. 1988, 29, 2155-2158.
-
(1988)
Tetrahedron Lett
, vol.29
, pp. 2155-2158
-
-
Claremon, D.A.1
Phillips, B.T.2
|