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Volumn 35, Issue 3, 2009, Pages 337-351

Formulation and characterization of a compacted multiparticulate system for modified release of water-soluble drugs - Part 1 acetaminophen

Author keywords

Ethylcellulose; Extrusion spheronization; Matrix tablets; Modified release; Multiparticulate delivery systems; Segregation

Indexed keywords

ALCOHOL; CALCIUM SILICATE; ETHYL CELLULOSE; LACTOSE; MICROCRYSTALLINE CELLULOSE; PARACETAMOL; PLACEBO; POVIDONE; WATER;

EID: 61649097748     PISSN: 03639045     EISSN: 15205762     Source Type: Journal    
DOI: 10.1080/03639040802360502     Document Type: Article
Times cited : (15)

References (39)
  • 1
    • 2942737072 scopus 로고    scopus 로고
    • Extruded and spheronized beads containing no microcrystalline cellulose: Influence of formulation and process variables
    • Agrawal, A., Howard, M. A., & Neau, S. H. (2004). Extruded and spheronized beads containing no microcrystalline cellulose: Influence of formulation and process variables. Pharm. Dev. Tech., 9(2), 197-217.
    • (2004) Pharm. Dev. Tech , vol.9 , Issue.2 , pp. 197-217
    • Agrawal, A.1    Howard, M.A.2    Neau, S.H.3
  • 2
    • 0028948839 scopus 로고
    • A theoretical basis for a biopharmaceutic drug classification: The correlation of in vitro drug product dissolution and in vivo bioavailability
    • Amidon, G. L., Lennernas, H., Shah, V. P., & Crison, J. R. (1995). A theoretical basis for a biopharmaceutic drug classification: The correlation of in vitro drug product dissolution and in vivo bioavailability. Pharm. Res., 12(3), 413-420.
    • (1995) Pharm. Res , vol.12 , Issue.3 , pp. 413-420
    • Amidon, G.L.1    Lennernas, H.2    Shah, V.P.3    Crison, J.R.4
  • 3
    • 0030909662 scopus 로고    scopus 로고
    • Changes in volume and compression energy upon compression of calcium silicate tablets
    • Asano, T., Tsubuku, S., Sugawara, S., Miyajima, M., Sato, H., Yuasa, H., & Kanaya, Y. (1997). Changes in volume and compression energy upon compression of calcium silicate tablets. Drug Dev. Ind. Pharm., 23(7), 679-685.
    • (1997) Drug Dev. Ind. Pharm , vol.23 , Issue.7 , pp. 679-685
    • Asano, T.1    Tsubuku, S.2    Sugawara, S.3    Miyajima, M.4    Sato, H.5    Yuasa, H.6    Kanaya, Y.7
  • 4
    • 0027984295 scopus 로고
    • The strength and compaction of millispheres
    • Aulton, M., Dyer, A. M., & Khan, K. A. (1994). The strength and compaction of millispheres. Drug Dev. Ind. Pharm., 20(20), 3069-3104.
    • (1994) Drug Dev. Ind. Pharm , vol.20 , Issue.20 , pp. 3069-3104
    • Aulton, M.1    Dyer, A.M.2    Khan, K.A.3
  • 5
    • 0035927222 scopus 로고    scopus 로고
    • Drying behavior of two sets of microcrystalline cellulose pellets
    • Berggren, J., & Alderborn, G. (2001). Drying behavior of two sets of microcrystalline cellulose pellets. Int. J. Pharm., 219, 113-126.
    • (2001) Int. J. Pharm , vol.219 , pp. 113-126
    • Berggren, J.1    Alderborn, G.2
  • 6
    • 2942616956 scopus 로고    scopus 로고
    • Compaction of enteric-coated pellets: Influence of formulation and process parameters on tablet properties and in vivo evaluation
    • Debunne, A., Vervaet, C., Mangelings, D., & Remon, J. P. (2004). Compaction of enteric-coated pellets: influence of formulation and process parameters on tablet properties and in vivo evaluation. Eur. J. Pharm. Sci., 22, 305-314.
    • (2004) Eur. J. Pharm. Sci , vol.22 , pp. 305-314
    • Debunne, A.1    Vervaet, C.2    Mangelings, D.3    Remon, J.P.4
  • 7
    • 0029093378 scopus 로고    scopus 로고
    • Dyer, A. M., Khan, K. A, & Aulton, M. E. (1995). Effect of polymer loading on drug release from film-coated Ibuprofen pellets prepared by extrusion-spheronization. Drug Dev. Ind. Pharm., 21(16), 1841-1858.
    • Dyer, A. M., Khan, K. A, & Aulton, M. E. (1995). Effect of polymer loading on drug release from film-coated Ibuprofen pellets prepared by extrusion-spheronization. Drug Dev. Ind. Pharm., 21(16), 1841-1858.
  • 8
    • 0031950145 scopus 로고    scopus 로고
    • Microcrystalline cellulose as a sponge as an alternative concept to the crystalline-gel model for extrusion and spheronization
    • Ek, R., & Newton, J. M. (1998). Microcrystalline cellulose as a sponge as an alternative concept to the crystalline-gel model for extrusion and spheronization. Pharm. Res., 15, 509-510.
    • (1998) Pharm. Res , vol.15 , pp. 509-510
    • Ek, R.1    Newton, J.M.2
  • 9
    • 0026554835 scopus 로고
    • Effect of amount and composition of granulation liquid on mixing, extrusion, and spheronization
    • Elbers, J., Bakkenes, H. W., & Fokkens, J. G. (1992). Effect of amount and composition of granulation liquid on mixing, extrusion, and spheronization. Drug Dev. Ind. Pharm., 18, 501-517.
    • (1992) Drug Dev. Ind. Pharm , vol.18 , pp. 501-517
    • Elbers, J.1    Bakkenes, H.W.2    Fokkens, J.G.3
  • 10
    • 42749084495 scopus 로고    scopus 로고
    • Cellulose swelling by protic solvents: Which properties of the biopolymer and the solvent matter?
    • El Seoud, O. A., Fidale, L. C., Ruiz, N., D'Almeida, M. L. O., & Frollini, E. (2008). Cellulose swelling by protic solvents: Which properties of the biopolymer and the solvent matter? Cellulose, 15, 371-392.
    • (2008) Cellulose , vol.15 , pp. 371-392
    • El Seoud, O.A.1    Fidale, L.C.2    Ruiz, N.3    D'Almeida, M.L.O.4    Frollini, E.5
  • 11
  • 12
    • 0021879828 scopus 로고
    • Formulation of sustained release promethazine hydrochloride tablets using hydroxypropylmethylcellulose matrices
    • Ford, J. L., Rubinstein, M. H., & Hogan, J. E. (1985). Formulation of sustained release promethazine hydrochloride tablets using hydroxypropylmethylcellulose matrices. Int. J. Pharm., 24, 327-338.
    • (1985) Int. J. Pharm , vol.24 , pp. 327-338
    • Ford, J.L.1    Rubinstein, M.H.2    Hogan, J.E.3
  • 13
    • 0034960479 scopus 로고    scopus 로고
    • A study of the effects of the physical characteristics of microcrystalline cellulose on performance in extrusion spheronization
    • Heng, P. W., & Koo, O. M. Y. (2001). A study of the effects of the physical characteristics of microcrystalline cellulose on performance in extrusion spheronization. Pharm. Res., 18(4), 480-487.
    • (2001) Pharm. Res , vol.18 , Issue.4 , pp. 480-487
    • Heng, P.W.1    Koo, O.M.Y.2
  • 14
    • 0030317409 scopus 로고    scopus 로고
    • Extrusion spheronization - Effect of moisture content and spheronization time on pellet characteristics
    • Iyer, R., Augsburger, L. L., Pope, D. G., & Shah, R. D. (1996). Extrusion spheronization - Effect of moisture content and spheronization time on pellet characteristics. Pharm. Dev. Tech., 1(4), 325-331.
    • (1996) Pharm. Dev. Tech , vol.1 , Issue.4 , pp. 325-331
    • Iyer, R.1    Augsburger, L.L.2    Pope, D.G.3    Shah, R.D.4
  • 15
    • 0028872408 scopus 로고
    • Compression behavior and compactibility of microcrystalline cellulose pellets in relation to their pore structure and mechanical properties
    • Johansson, B., Wickberg, M., Ek, R., & Alderborn, G. (1995). Compression behavior and compactibility of microcrystalline cellulose pellets in relation to their pore structure and mechanical properties. Int. J. Pharm., 117, 57-73.
    • (1995) Int. J. Pharm , vol.117 , pp. 57-73
    • Johansson, B.1    Wickberg, M.2    Ek, R.3    Alderborn, G.4
  • 16
    • 0029052299 scopus 로고
    • Ethylcellulose matrix controlled release tablets of a water soluble drug
    • August
    • Katikaneni, P., Upadrashta, S. M., Neau, S. H., & Mitra, A. K. (1995a). Ethylcellulose matrix controlled release tablets of a water soluble drug. Int. J. Pharm., 123(August), 119-125.
    • (1995) Int. J. Pharm , vol.123 , pp. 119-125
    • Katikaneni, P.1    Upadrashta, S.M.2    Neau, S.H.3    Mitra, A.K.4
  • 17
    • 0028896830 scopus 로고
    • Consolidation of ethylcellulose: Effect of particle size, press speed, and lubricants
    • April
    • Katikaneni, P. R., Upadrashta, S. M., Rowlings, C. E., Neau, S. H., Hileman, G. A. (1995b). Consolidation of ethylcellulose: effect of particle size, press speed, and lubricants. Int. J. Pharm., 117(April), 13-21.
    • (1995) Int. J. Pharm , vol.117 , pp. 13-21
    • Katikaneni, P.R.1    Upadrashta, S.M.2    Rowlings, C.E.3    Neau, S.H.4    Hileman, G.A.5
  • 18
    • 34447127532 scopus 로고    scopus 로고
    • Drug release kinetics from tablet matrices based upon ethylcellulose ether-derivatives: A comparison between different formulations
    • Khan, G., & Meidan, V.M. (2007). Drug release kinetics from tablet matrices based upon ethylcellulose ether-derivatives: A comparison between different formulations. Drug Dev. Ind. Pharm., 33(6), 627-639.
    • (2007) Drug Dev. Ind. Pharm , vol.33 , Issue.6 , pp. 627-639
    • Khan, G.1    Meidan, V.M.2
  • 19
    • 0031001487 scopus 로고    scopus 로고
    • The crystallite-gel-model for microcrystalline cellulose in wet-granulation, extrusion, and spheronization
    • Kleinebudde, P. (1997). The crystallite-gel-model for microcrystalline cellulose in wet-granulation, extrusion, and spheronization. Pharm. Res., 14(6), 804-809.
    • (1997) Pharm. Res , vol.14 , Issue.6 , pp. 804-809
    • Kleinebudde, P.1
  • 23
    • 33749666655 scopus 로고    scopus 로고
    • Once-daily tablet formulation and in vitro release evaluation of Cefpodoxime using hydroxypropyl methylcellulose: A technical note
    • Article
    • Merchant, H. A., Shoaib, H. M., Tazeen, J., & Yousuf, R. I. (2006). Once-daily tablet formulation and in vitro release evaluation of Cefpodoxime using hydroxypropyl methylcellulose: A technical note. AAPS PharmSciTech, 7(3), Article 78.
    • (2006) AAPS PharmSciTech , vol.7 , Issue.3 , pp. 78
    • Merchant, H.A.1    Shoaib, H.M.2    Tazeen, J.3    Yousuf, R.I.4
  • 24
    • 0025294139 scopus 로고
    • The strength of microcrystalline cellulose pellets: The effect of granulating with water/ethanol mixtures
    • Millili, G., & Schwartz, J. B. (1990). The strength of microcrystalline cellulose pellets: The effect of granulating with water/ethanol mixtures. Drug Development and Industrial Pharmacy, 16, 1411-1426.
    • (1990) Drug Development and Industrial Pharmacy , vol.16 , pp. 1411-1426
    • Millili, G.1    Schwartz, J.B.2
  • 25
    • 61649106803 scopus 로고    scopus 로고
    • Martindale: The complete drug reference. Paracetamol
    • Parfitt, K, Ed, London: Pharmaceutical Press
    • Parfitt, K. (Ed.). (1999). Martindale: The complete drug reference. Paracetamol. In Analgesics, antiinflammatory drugs and antipyretics (pp. 1-91). London: Pharmaceutical Press.
    • (1999) Analgesics, antiinflammatory drugs and antipyretics , pp. 1-91
  • 26
    • 0023909986 scopus 로고
    • Influence of liquid bonding strength on power consumption during granulation in a high shear mixer
    • Ritala, M., Holm, P., Schaefer, T., & Kristensen, H. G. (1988). Influence of liquid bonding strength on power consumption during granulation in a high shear mixer. Drug Development and Industrial Pharmacy, 14(8), 1041-1060.
    • (1988) Drug Development and Industrial Pharmacy , vol.14 , Issue.8 , pp. 1041-1060
    • Ritala, M.1    Holm, P.2    Schaefer, T.3    Kristensen, H.G.4
  • 27
    • 0034690967 scopus 로고    scopus 로고
    • Effects of liquid phase migration on extrusion of microcrystalline cellulose pastes
    • Rough, S. L., Bridgwater, J., & Wilson, D. I., (2000). Effects of liquid phase migration on extrusion of microcrystalline cellulose pastes. International Journal of Pharmaceutics, 204, 117-126.
    • (2000) International Journal of Pharmaceutics , vol.204 , pp. 117-126
    • Rough, S.L.1    Bridgwater, J.2    Wilson, D.I.3
  • 28
    • 0029921644 scopus 로고    scopus 로고
    • Investigation of ethylcellulose as a matrix former and a new method to regard and evaluate the compaction data
    • Shlieout, G., & Zessin, G. (1996). Investigation of ethylcellulose as a matrix former and a new method to regard and evaluate the compaction data. Drug Development and Industrial Pharmacy, 22(4), 313-319.
    • (1996) Drug Development and Industrial Pharmacy , vol.22 , Issue.4 , pp. 313-319
    • Shlieout, G.1    Zessin, G.2
  • 29
    • 33750606941 scopus 로고    scopus 로고
    • Micromeritics
    • D. Troy Ed, Philadelphia, PA: Lippincott Williams and Wilkins
    • Sinko, P. J. (2006). Micromeritics. In D. Troy (Ed.), Martin's physical pharmacy and pharmaceutical sciences (pp. 533-560). Philadelphia, PA: Lippincott Williams and Wilkins.
    • (2006) Martin's physical pharmacy and pharmaceutical sciences , pp. 533-560
    • Sinko, P.J.1
  • 31
    • 23144461821 scopus 로고    scopus 로고
    • Controlled release formulation of tramadol hydrochloride using hydrophilic and hydrophobic matrix system
    • Article
    • Tiwari, S., Murthy, T. M., Pai, M. R., Mehta, P. R., & Chowdary, P. B. (2003). Controlled release formulation of tramadol hydrochloride using hydrophilic and hydrophobic matrix system. AAPS PharmSciTech, 4(3), Article 31.
    • (2003) AAPS PharmSciTech , vol.4 , Issue.3 , pp. 31
    • Tiwari, S.1    Murthy, T.M.2    Pai, M.R.3    Mehta, P.R.4    Chowdary, P.B.5
  • 33
    • 0036637718 scopus 로고    scopus 로고
    • Formulation and optimization of a sustained-release tablet of ketorolac tromethamine
    • Vatsaraj, N., Zia, H., & Needham, T. (2002). Formulation and optimization of a sustained-release tablet of ketorolac tromethamine. Drug Delivery, 9, 153-159.
    • (2002) Drug Delivery , vol.9 , pp. 153-159
    • Vatsaraj, N.1    Zia, H.2    Needham, T.3
  • 37
    • 61649096236 scopus 로고    scopus 로고
    • Xie, L., Wu, H., Shen, M., Augsburger, L. L., Lyon, R. C., Khan, M. A., Hussain, A. S., & Hoag, S. W. (2007) Quality-by-design: Effects of testing parameters and formulation variables on the segregation tendency of pharmaceutical powder measured by the ASTM D 6940-04 segregation tester. Journal of Pharmaceutical Sciences.
    • Xie, L., Wu, H., Shen, M., Augsburger, L. L., Lyon, R. C., Khan, M. A., Hussain, A. S., & Hoag, S. W. (2007) Quality-by-design: Effects of testing parameters and formulation variables on the segregation tendency of pharmaceutical powder measured by the ASTM D 6940-04 segregation tester. Journal of Pharmaceutical Sciences.
  • 38
    • 0029997330 scopus 로고    scopus 로고
    • Studies on internal structure of tablets VI. Stress dispersion in tablets by excipients
    • Yuasa, H., Akutagawa, M., Hashizume, T., & Kanaya, Y. (1996). Studies on internal structure of tablets VI. Stress dispersion in tablets by excipients. Chemical and Pharmaceutical Bulletin, 44(2), 378-382.
    • (1996) Chemical and Pharmaceutical Bulletin , vol.44 , Issue.2 , pp. 378-382
    • Yuasa, H.1    Akutagawa, M.2    Hashizume, T.3    Kanaya, Y.4
  • 39
    • 0034948965 scopus 로고    scopus 로고
    • Studies on stress dispersion in tablets III. Suppression of fracture of coated film by an excipient during the preparation of tablets containing coated particles
    • Yuasa, H., Takashima, Y., Omata, T., & Kanaya, Y. (2001). Studies on stress dispersion in tablets III. Suppression of fracture of coated film by an excipient during the preparation of tablets containing coated particles. STP Pharma Sciences, 11(3), 221-227.
    • (2001) STP Pharma Sciences , vol.11 , Issue.3 , pp. 221-227
    • Yuasa, H.1    Takashima, Y.2    Omata, T.3    Kanaya, Y.4


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