Stabilizing dispersions of hydrophobic drug molecules using cellulose ethers during anti-solvent synthesis of micro-particulates

Colloids and Surfaces B: Biointerfaces

Volumn 70, Issue 1, 2009, Pages 7-14

  Meng, Xiangxin ^a   Chen, Yuhong ^a   Chowdhury, Subhendu R ^a   Yang, Dachuan ^b   Mitra, Somenath ^a  

^a NEW JERSEY INSTITUTE OF TECHNOLOGY   (United States)

^b ETHICON INC   (United States)

Author keywords

Anti solvent; Colloid; Drug delivery; Drug particles; Micronization of API

Indexed keywords

ANTI-SOLVENT; AVERAGE PARTICLE SIZES; CELLULOSE ETHERS; DRUG MOLECULES; DRUG PARTICLES; FENOFIBRATE; HYDROPHOBIC DRUGS; LOW-POWER; MEAN DIAMETERS; MICRO-SCALE; MICRONIZATION OF API; PARTICLE SHAPES; PARTICLE SIZE DISTRIBUTIONS; POINT MEASUREMENTS; SEDIMENTATION RATES; SMALL PARTICLES; STABLE SUSPENSIONS; THERMODYNAMICALLY STABLES; ZETA POTENTIAL MEASUREMENTS;

AGGLOMERATION; CELLULOSE; DIFFUSERS (OPTICAL); DRUG DELIVERY; ETHERS; MELTING POINT; ORGANIC COMPOUNDS; PARTICLE SIZE; SCANNING ELECTRON MICROSCOPY; SOLVENTS; SURFACE ACTIVE AGENTS; ZETA POTENTIAL;

SUSPENSIONS (FLUIDS);

CELLULOSE; ETHER; FENOFIBRATE; GRISEOFULVIN; SURFACTANT;

ARTICLE; CHEMICAL REACTION; DRUG STRUCTURE; HYDROPHOBICITY; PARTICLE SIZE; PRIORITY JOURNAL;

CELLULOSE; COLLOIDS; DRUG COMPOUNDING; DRUG DELIVERY SYSTEMS; ETHER, ETHYL; GRISEOFULVIN; HYDROPHOBICITY; MICROSCOPY, ELECTRON, SCANNING; MODELS, CHEMICAL; PARTICLE SIZE; PROCETOFEN; SOLVENTS; SPECTRUM ANALYSIS, RAMAN; SUSPENSIONS; THERMODYNAMICS;

AGGLOMERATION; CELLULOSE; COLLOIDS; DIFFUSERS; DISPERSIONS; ETHERS; MELTING POINT; ORGANIC COMPOUNDS; PARTICLE SIZE; SCANNING ELECTRON MICROSCOPY; SOLVENTS; SURFACTANTS; ZETA POTENTIAL;

EID: 61449085466     PISSN: 09277765     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.colsurfb.2008.12.002     Document Type: Article

References (40)

1. Mehta S.K., Kaur G., and Bhasin K.K. Colloids Surf. B: Biointerf. 60 (2007) 95-104
2. Yuan H., Huang L., Du Y., Ying X., You J., Hu F., and Zeng S. Colloids Surf. B: Biointerf. 61 (2008) 132-137
3. Gao Y., Li L., and Zhai G. Colloids Surf. B: Biointerf. 64 (2008) 194-199
4. Perrut M., Jung J., and Leboeuf F. Int. J. Pharm. 288 (2005) 3-10
5. Wong S.M., Kellaway I.W., and Murdan S. Int. J. Pharm. 317 (2006) 61-68
6. Gioannis B.D., Jestin P., and Subra P. J. Cryst. Growth 262 (2004) 519-526
7. Zimmermann A., Elema M.R., Hansen T., Mullertz A., and Hovgaard L. J. Pharmaceut. Biomed. 44 (2007) 874-880
8. Helfgen B., Hils P., Holzknecht C., Turk M., and Schaber K. J. Aerosol Sci. 32 (2001) 295-319
9. Weber M., Russell L.M., and Debenedetti P.G. J. Supercrit. Fluid 23 (2002) 65-80
10. Young T.J., Johnston K.P., Pace G.W., and Mishra A.K. AAPS PharmSciTech. 5 (2003) 1-16
11. Marchisio D.L., Rivautella L., and Barresi A.A. AIChE J. 52 (2006) 1877-1887
12. M. Weber, M.C. Thies, Understanding the RESS process, in: Y.P. Sun, (Ed.), Supercritical Fluid Technology in Materials Science and Engineering: Synthesis, Properties, and Applications, Marcel Dekker, New York, 2002, pp. 387-437.
13. Matteucci M.E., Hotze M.A., Johnston K.P., and William R.O. Langmuir 22 (2006) 8951-8959
14. Zili Z., Sfar S., and Fessi H. Int. J. Pharm. 294 2005 (2005) 261-267
15. Dreis S., Rothweiler F., Michaelis M., Cinatl J.J., Kreuter J., and Langer K. Int. J. Pharm. 341 (2007) 207-214
16. Muller R.H., Moschwitzer J., and Bushrab F.N. In: Gupta R.B., and Kompella U.B. (Eds). Manufacturing of Nanoparticles by Milling and Homogenization Techniques (2006), Nanoparticle Technology for Drug Delivery, New York 21-52
17. Duro R., Alvarez C., Martinez-Pacheco R., Gomez-Amoza J.L., Concheiro A., and Souto C. Eur. J. Pharm. Biopharm. 45 (1998) 181-188
18. Chacon M., Molpeceres L., Berges L., Guzman M., and Aberturas M.R. Eur. J. Pharm. Sci. 8 (1999) 99-107
19. Martinac A., Filipovic-Grcic J., Voinovich D., Perissutti B., and Franceschinis E. Int. J. Pharm. 291 (2005) 69-77
20. Tantishaiyakul V., Kaewnopparat N., and Ingkatawornwong S. Int. J. Pharm. 181 (1999) 143-151
21. Broman E., Khoo C., and Taylor L.S. Int. J. Pharm. 222 (2001) 139-151
22. Yagi N., Terashima Y., Kenmotsu H., Sekikawa H., and Takada M. Chem. Pharm. Bull. 44 (1996) 241-244
23. Pongpeerapat A., Itoh K., Tozuka Y., Moribe K., Oguchi T., and Yamamoto K. J. Drug Del. Sci. Technol. 14 (2004) 441-447
24. Terayama H., Funakoshi M., Torigoe K., and Esumi K. Colloids Surf. B: Biointerf. 23 (2002) 65-71
25. Terayama H., Hirota K., Yoshimura T., and Esumi K. Colloids Surf. B: Biointerf. 27 (2002) 177-180
26. Terayama H., Okumura K., Sakai K., Torigoe K., and Esumi K. Colloids Surf. B: Biointerf. 20 (2001) 73-77
27. Itoh K., Pongpeerapat A., Tozuka Y., Oguchi T., and Yamamoto K. Chem. Pharm. Bull. 51 (2003) 171-174
28. Yasueda S., Inada K., Matsuhisa K., Terayama H., and Ohtori A. Eur. J. Pharm. Sci. 57 (2004) 377-382
29. Ain-Ai A., and Gupta P.K. Int. J. Pharm. 351 (2008) 282-288
30. Yalkowsky S.H., and Valvani S.C. J. Pharm. Sci. 69 (1980) 912-922
31. Vippagunta S.R., Wang Z., Hornung S., and Krill S.L. J. Pharm. Sci. 96 (2007) 294-304
32. C.F. Rodriguez, N. Bruneau, J. Barra, D. Alfonso, E. Doelker, Hydrophilic cellulose derivatives as drug delivery carriers: Influence of substitution type on the properties of compressed matrix tablets, in: D.L. Wise (Ed.), Handbook of Pharmaceutical Controlled Release Technology, Marcel Dekker, New York, 2000, pp. 1-30.
33. Gun'ko V.M., Klyueva A.V., Levchuk Y.N., and Leboda R. Adv. Colloid Interf. 105 (2003) 201-328
34. Eerdenbrugha B., Froyenb L., Humbeeckb J., Martensc J.A., Augustijnsa P., and Mootera G. Eur. J. Pharm. Sci. 35 (2008) 127-135
35. J.R. Larson, G.A. Gibson, S.P. Schmidt, Liquid toner materials, in: A.S. Diamond, D.S. Weiss (Eds.), Handbook of Imaging Materials, Marcel Dekker, New York, 2002, pp. 239-264.
36. Daniels R., and Barta A. Eur. J. Pharm. Sci. 40 (1994) 128-133
37. Rasenack N., and Muller B.W. Pharm. Res. 19 (2002) 1894-1900
38. L.V. Allen, N.G. Popvich, H.C. Ansel, Section VI. Liquid dosage forms, in: Ansel's Pharmaceutical Dosage Forms and Drug Delivery Systems, 8th ed., Lippincott Williams & Wilkins, Baltimore, 2005, pp. 336-384.
39. Terayama H., Inada K., Nakayama H., Yasueda S., and Esumi K. Colloids Surf. B: Biointerf. 39 (2004) 159-164
40. Bolton B.A., and Prasad P.N. J. Pharm. Sci. 70 (1981) 789-793