-
1
-
-
33644886821
-
First inhibitors of the steroidogenic enzyme type 7 17β-hydroxysteroid dehydrogenase
-
Bellavance E., Luu-The V., and Poirier D. First inhibitors of the steroidogenic enzyme type 7 17β-hydroxysteroid dehydrogenase. Lett. Drug Des. Discov. 1 (2004) 194-197
-
(2004)
Lett. Drug Des. Discov.
, vol.1
, pp. 194-197
-
-
Bellavance, E.1
Luu-The, V.2
Poirier, D.3
-
3
-
-
60149084693
-
-
Bydal, P., Luu-The, V., Poirier, P., in press. Steroidal lactones as inhibitors of 17β-hydroxysteroid dehydrogenase type 5: chemical synthesis, enzyme inhibitory activity, and assessment of estrogenic and androgenic activities. Eur. J. Med. Chem., doi:10.1016/j.ejmech.2008.03.020.
-
Bydal, P., Luu-The, V., Poirier, P., in press. Steroidal lactones as inhibitors of 17β-hydroxysteroid dehydrogenase type 5: chemical synthesis, enzyme inhibitory activity, and assessment of estrogenic and androgenic activities. Eur. J. Med. Chem., doi:10.1016/j.ejmech.2008.03.020.
-
-
-
-
4
-
-
33845336541
-
C6-(N,N-butyl-methyl-heptanamide) derivatives of estrone and estradiol as inhibitors of type 1 17β-hydroxysteroid dehydrogenase: chemical synthesis and biological evaluation
-
Cadot C., Laplante Y., Kamal F., Luu-The V., and Poirier D. C6-(N,N-butyl-methyl-heptanamide) derivatives of estrone and estradiol as inhibitors of type 1 17β-hydroxysteroid dehydrogenase: chemical synthesis and biological evaluation. Bioorg. Med. Chem. 15 (2007) 714-726
-
(2007)
Bioorg. Med. Chem.
, vol.15
, pp. 714-726
-
-
Cadot, C.1
Laplante, Y.2
Kamal, F.3
Luu-The, V.4
Poirier, D.5
-
5
-
-
0141919555
-
Inhibition of estrone sulphate-induced uterine growth by potent nonestrogenic steroidal inhibitors of steroid sulfatase
-
Ciobanu L.C., Luu-The V., Martel C., Labrie F., and Poirier D. Inhibition of estrone sulphate-induced uterine growth by potent nonestrogenic steroidal inhibitors of steroid sulfatase. Cancer Res. 63 (2003) 6442-6446
-
(2003)
Cancer Res.
, vol.63
, pp. 6442-6446
-
-
Ciobanu, L.C.1
Luu-The, V.2
Martel, C.3
Labrie, F.4
Poirier, D.5
-
7
-
-
60249090183
-
Relative involvement of three 17β-hydroxysteroid dehydrogenases (types 1, 7 and 12) in the formation of estradiol in various breast cancer cell lines using selective inhibitors
-
Laplante Y., Rancourt C., and Poirier D. Relative involvement of three 17β-hydroxysteroid dehydrogenases (types 1, 7 and 12) in the formation of estradiol in various breast cancer cell lines using selective inhibitors. Mol. Cell. Endocrinol. 301 (2009) 146-153
-
(2009)
Mol. Cell. Endocrinol.
, vol.301
, pp. 146-153
-
-
Laplante, Y.1
Rancourt, C.2
Poirier, D.3
-
8
-
-
0034993363
-
Analysis and characteristics of multiple types of human 17beta-hydroxysteroid dehydrogenase
-
Luu-The V. Analysis and characteristics of multiple types of human 17beta-hydroxysteroid dehydrogenase. J. Steroid Biochem. Mol. Biol. 76 (2001) 143-151
-
(2001)
J. Steroid Biochem. Mol. Biol.
, vol.76
, pp. 143-151
-
-
Luu-The, V.1
-
9
-
-
31444432288
-
Characterization of type 12 17beta-hydroxysteroid dehydrogenase, an isoform of type 3 17beta-hydroxysteroid dehydrogenase responsible for estradiol formation in women
-
Luu-The V., Tremblay P., and Labrie F. Characterization of type 12 17beta-hydroxysteroid dehydrogenase, an isoform of type 3 17beta-hydroxysteroid dehydrogenase responsible for estradiol formation in women. Mol. Endocrinol. 20 (2006) 437-443
-
(2006)
Mol. Endocrinol.
, vol.20
, pp. 437-443
-
-
Luu-The, V.1
Tremblay, P.2
Labrie, F.3
-
10
-
-
33644894458
-
Multifunctionality of human 17β-hydroxysteroid dehydrogenases
-
Moeller G., and Adamski J. Multifunctionality of human 17β-hydroxysteroid dehydrogenases. Mol. Cell. Endocrinol. 248 (2006) 47-55
-
(2006)
Mol. Cell. Endocrinol.
, vol.248
, pp. 47-55
-
-
Moeller, G.1
Adamski, J.2
-
11
-
-
33644881888
-
Aldo-keto reductase (AKR) 1C3: role in prostate disease and the development of specific inhibitors
-
Penning T., Steckelbroeck S., Bauman D.R., Miller M.W., Jin Y., Peehl D.M., Fung K.M., and Lin H.K. Aldo-keto reductase (AKR) 1C3: role in prostate disease and the development of specific inhibitors. Mol. Cell. Endocrinol. 248 (2006) 182-191
-
(2006)
Mol. Cell. Endocrinol.
, vol.248
, pp. 182-191
-
-
Penning, T.1
Steckelbroeck, S.2
Bauman, D.R.3
Miller, M.W.4
Jin, Y.5
Peehl, D.M.6
Fung, K.M.7
Lin, H.K.8
-
12
-
-
0037277521
-
Inhibitors of 17β-hydroxysteroid dehydrogenases
-
Poirier D. Inhibitors of 17β-hydroxysteroid dehydrogenases. Curr. Med. Chem. 10 (2003) 453-477
-
(2003)
Curr. Med. Chem.
, vol.10
, pp. 453-477
-
-
Poirier, D.1
-
13
-
-
17044428337
-
Steroid sulfatase: molecular biology, regulation, and inhibition
-
Reed M.J., Purohit A., Woo L.W.L., Newman S.P., and Potter B.V.L. Steroid sulfatase: molecular biology, regulation, and inhibition. Endocr. Rev. 26 (2005) 171-202
-
(2005)
Endocr. Rev.
, vol.26
, pp. 171-202
-
-
Reed, M.J.1
Purohit, A.2
Woo, L.W.L.3
Newman, S.P.4
Potter, B.V.L.5
-
14
-
-
0035019952
-
Inhibitors of steroidogenesis as agents for the treatment of hormone-dependent cancers
-
Smith H.J., Nicholls P.J., Simons C., and Le Lain R. Inhibitors of steroidogenesis as agents for the treatment of hormone-dependent cancers. Expert Opin. Ther. Patents 11 (2001) 789-824
-
(2001)
Expert Opin. Ther. Patents
, vol.11
, pp. 789-824
-
-
Smith, H.J.1
Nicholls, P.J.2
Simons, C.3
Le Lain, R.4
-
15
-
-
33644898089
-
Expression analysis of estrogen-metabolizing enzymes in human endometrial cancer
-
Smuc T., Rupreht R., Sinkovec J., Adamski J., and Lanisnik-Rizner T. Expression analysis of estrogen-metabolizing enzymes in human endometrial cancer. Mol. Cell. Endocrinol. 248 (2006) 114-117
-
(2006)
Mol. Cell. Endocrinol.
, vol.248
, pp. 114-117
-
-
Smuc, T.1
Rupreht, R.2
Sinkovec, J.3
Adamski, J.4
Lanisnik-Rizner, T.5
-
16
-
-
60249103491
-
Aberrant pre-receptor regulation of estrogen and progesterone action in endometrial cancer
-
Smuc T., and Lanisnik-Rizner T. Aberrant pre-receptor regulation of estrogen and progesterone action in endometrial cancer. Mol. Cell. Endocrinol. 301 (2009) 74-82
-
(2009)
Mol. Cell. Endocrinol.
, vol.301
, pp. 74-82
-
-
Smuc, T.1
Lanisnik-Rizner, T.2
-
17
-
-
18444369971
-
Inhibitors of type 1 17β-hydroxysteroid dehydrogenase with reduced estrogenic activity: modifications of the positions 3 and 6 of estradiol
-
Tremblay M.R., Boivin R., Luu-The V., and Poirier D. Inhibitors of type 1 17β-hydroxysteroid dehydrogenase with reduced estrogenic activity: modifications of the positions 3 and 6 of estradiol. J. Enzyme Inhib. Med. Chem. 20 (2005) 153-163
-
(2005)
J. Enzyme Inhib. Med. Chem.
, vol.20
, pp. 153-163
-
-
Tremblay, M.R.1
Boivin, R.2
Luu-The, V.3
Poirier, D.4
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