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1
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57549112701
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Presented at the 235th National Meeting of the American Chemical Society, New Orleans, LA; April 6-10, 2008.
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Presented at the 235th National Meeting of the American Chemical Society, New Orleans, LA; April 6-10, 2008.
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2
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0033614947
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Jimonet P., Audiau F., Barreau M., Blanchard J.-C., Boireau A., Bour Y., Coleno M.-A., Doble A., Doerflinger G., Huu C.D., Donat M.H., Duchesne J.M., Ganul P., Gueremy C., Honore R., Just B., Kerpherique R., Gontier S., Hubert P., Laduron P.M., LeBlevec J., Meunier M., Miquet J.-M., Nemecek C., Pasquet M., Piot O., Pratt J., Rataud J., Reibaud M., Stutzman J.-M., and Mignani S. J. Med. Chem. 42 (1999) 2828-2843
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(1999)
J. Med. Chem.
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Jimonet, P.1
Audiau, F.2
Barreau, M.3
Blanchard, J.-C.4
Boireau, A.5
Bour, Y.6
Coleno, M.-A.7
Doble, A.8
Doerflinger, G.9
Huu, C.D.10
Donat, M.H.11
Duchesne, J.M.12
Ganul, P.13
Gueremy, C.14
Honore, R.15
Just, B.16
Kerpherique, R.17
Gontier, S.18
Hubert, P.19
Laduron, P.M.20
LeBlevec, J.21
Meunier, M.22
Miquet, J.-M.23
Nemecek, C.24
Pasquet, M.25
Piot, O.26
Pratt, J.27
Rataud, J.28
Reibaud, M.29
Stutzman, J.-M.30
Mignani, S.31
more..
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3
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0037171819
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Hauel N.H., Nar H., Priepke H., Ries U., Stassen J.-M., and Wienen W. J. Med. Chem. 45 (2002) 1757-1766
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(2002)
J. Med. Chem.
, vol.45
, pp. 1757-1766
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Hauel, N.H.1
Nar, H.2
Priepke, H.3
Ries, U.4
Stassen, J.-M.5
Wienen, W.6
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5
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43449104720
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Thiel O.R., Bernard C., King T., Dilmeghani-Seran M., Bostick T., Larsen R.D., and Faul M.M. J. Org. Chem. 73 (2008) 3508-3515
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(2008)
J. Org. Chem.
, vol.73
, pp. 3508-3515
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Thiel, O.R.1
Bernard, C.2
King, T.3
Dilmeghani-Seran, M.4
Bostick, T.5
Larsen, R.D.6
Faul, M.M.7
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6
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0033577574
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Suzuki H., Shindo K., Ueno A., Miura T., Takei M., Sakakibara M., Fukamachi H., Tanaka J., and Higa T. Bioorg. Med. Chem. Lett. 9 (1999) 1361-1364
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Suzuki, H.1
Shindo, K.2
Ueno, A.3
Miura, T.4
Takei, M.5
Sakakibara, M.6
Fukamachi, H.7
Tanaka, J.8
Higa, T.9
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7
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0032480820
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Bonnert R.V., Brown R.C., Chapman D., Cheshire D.R., Dixon J., Ince F., Kinchin E.C., Lyons A.J., Davis A.M., Hallam C., Harper S.T., Unitt J.F., Dougall I.G., Jackson D.M., McKechnie K., Young A., and Simpson W.T. J. Med. Chem. 41 (1998) 4915
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J. Med. Chem.
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Bonnert, R.V.1
Brown, R.C.2
Chapman, D.3
Cheshire, D.R.4
Dixon, J.5
Ince, F.6
Kinchin, E.C.7
Lyons, A.J.8
Davis, A.M.9
Hallam, C.10
Harper, S.T.11
Unitt, J.F.12
Dougall, I.G.13
Jackson, D.M.14
McKechnie, K.15
Young, A.16
Simpson, W.T.17
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10
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57549104470
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See also: Pansegrau, P. D. U.S. 6013841 (1998), WO2000006527, 1999.
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See also: Pansegrau, P. D. U.S. 6013841 (1998), WO2000006527, 1999.
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11
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0001340433
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For a representative protocol for preparing an N,N-di-tert-butoxycarbonyl (i.e, the N,N-diBoc) derivative of an amine see:
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For a representative protocol for preparing an N,N-di-tert-butoxycarbonyl (i.e, the N,N-diBoc) derivative of an amine see:. Kokotos G., Padrón M., Martín T., Gibbons W.A., and Martín V.S. J. Org. Chem. 63 (1998) 3741-3744
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(1998)
J. Org. Chem.
, vol.63
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Kokotos, G.1
Padrón, M.2
Martín, T.3
Gibbons, W.A.4
Martín, V.S.5
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13
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0005986596
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For early references on the conversion of arylmethyl groups to dibromides en route to the corresponding aldehydes see:
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For early references on the conversion of arylmethyl groups to dibromides en route to the corresponding aldehydes see:. Gilman H., Brannen C., and Ingham R.K. J. Am. Chem. Soc. 78 (1956) 1689-1692
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(1956)
J. Am. Chem. Soc.
, vol.78
, pp. 1689-1692
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Gilman, H.1
Brannen, C.2
Ingham, R.K.3
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14
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33044495162
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Baraldi P.G., Budriesi R., Cacciari B., Chiarini A., Garuti L., Giovannineti G., Leoni A., and Roberti M. Collect. Czech. Chem. Commun. 57 (1992) 169-178
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(1992)
Collect. Czech. Chem. Commun.
, vol.57
, pp. 169-178
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Baraldi, P.G.1
Budriesi, R.2
Cacciari, B.3
Chiarini, A.4
Garuti, L.5
Giovannineti, G.6
Leoni, A.7
Roberti, M.8
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15
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39149102658
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Ma D., Ding Ke., Tian H., Wang B., and Cheng D. Tetrahedron: Asymmetry 13 (2002) 961-969
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(2002)
Tetrahedron: Asymmetry
, vol.13
, pp. 961-969
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Ma, D.1
Ding, Ke.2
Tian, H.3
Wang, B.4
Cheng, D.5
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17
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0942268076
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For a procedure where the conversion of a methyl group to an aldehyde or a carboxylic acid is facilitated through a monobromide see:
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For a procedure where the conversion of a methyl group to an aldehyde or a carboxylic acid is facilitated through a monobromide see:. Deady L.W., Devine S.M., and Rogers M.L. Org. Prep. Proced. Int. 35 (2003) 627-630
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(2003)
Org. Prep. Proced. Int.
, vol.35
, pp. 627-630
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Deady, L.W.1
Devine, S.M.2
Rogers, M.L.3
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18
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33947460144
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For the related Kornblum oxidation of alkyl and benzyl halides and tosylates to aldehydes see:
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For the related Kornblum oxidation of alkyl and benzyl halides and tosylates to aldehydes see:. Kornblum N., Jones W.J., and Anderson G.J. J. Am. Chem. Soc. 81 (1959) 4113-4114
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(1959)
J. Am. Chem. Soc.
, vol.81
, pp. 4113-4114
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Kornblum, N.1
Jones, W.J.2
Anderson, G.J.3
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19
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57549095552
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Seemuth, P. D. U. S. Patent 4,317,934, 1982.
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Seemuth, P. D. U. S. Patent 4,317,934, 1982.
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20
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57549117009
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Smutny, E. J.; Colby, T. H. U. S. Patent 4,229,380, 1980.
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Smutny, E. J.; Colby, T. H. U. S. Patent 4,229,380, 1980.
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21
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0032005225
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Jones C.W., Carter N.G., Oakes S.C., Wilson S.L., and Johnstone A. J. Chem. Technol. Biotechnol. 71 (1998) 111-120
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(1998)
J. Chem. Technol. Biotechnol.
, vol.71
, pp. 111-120
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Jones, C.W.1
Carter, N.G.2
Oakes, S.C.3
Wilson, S.L.4
Johnstone, A.5
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22
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22744453841
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Tishkov A.A., Schmidhammer U., Roth S., Riedle E., and Mayr H. Angew. Chem., Int. Ed. Engl. 44 (2005) 4623-4626
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(2005)
Angew. Chem., Int. Ed. Engl.
, vol.44
, pp. 4623-4626
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Tishkov, A.A.1
Schmidhammer, U.2
Roth, S.3
Riedle, E.4
Mayr, H.5
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24
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57549094600
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note
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The preparation of S1319 analogues, using the scheme described herein will be communicated separately.
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