Pseudoephedrine hydrochloride sustained-release pellets prepared by a combination of hot-melt subcoating and polymer coating

Drug Development and Industrial Pharmacy

Volumn 34, Issue 12, 2008, Pages 1323-1330

  Yang, Zi Yi ^a   Lu, Yan ^a   Tang, Xing ^a  

^a SHENYANG PHARMACEUTICAL UNIVERSITY   (China)

Author keywords

Fluidized bed; Hot melt subcoating; Polymer coating; Pseudoephedrine hydrochloride; Sustained release pellets

Indexed keywords

EUDRAGIT; POLYMER; PSEUDOEPHEDRINE;

ARTICLE; DENSITY; DRUG PELLET; DRUG SOLUBILITY; FLUIDIZED BED; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; PARTICLE SIZE; SURFACE PROPERTY; SUSTAINED RELEASE PREPARATION;

DELAYED-ACTION PREPARATIONS; MICROSCOPY, ELECTRON, SCANNING; PSEUDOEPHEDRINE; SOLUBILITY; TECHNOLOGY, PHARMACEUTICAL;

EID: 57349091773     PISSN: 03639045     EISSN: 15205762     Source Type: Journal    
DOI: 10.1080/03639040802084938     Document Type: Article

References (21)

1. Allen, L. V., Jr., Popovich, N. G., & Ansel, H. C. (2005). Ansel's pharmaceutical dosage forms and drug delivery systems (8th ed., pp. 265-266). Lippincott Williams & Wilkins.
2. Barthelemya, P., Laforêta, J. P., Faraha, N., & Joachimb, J. (1999). Compritol® 888 ATO: An innovative hot-melt coating agent for prolonged-release drug formulations. Eur. J. Pharm. Biopharm., 47, 87-90.
3. Bruce, L. D., Koleng, J. J., & McGinity, J. W. (2003). The influence of polymeric subcoats and pellet formulation on the release of chlorpheniramine maleate from enteric coated pellets. Drug Dev. Ind. Pharm., 29, 909-924.
4. Bruce, L. D., Petereit, H. J., Beckert, T., & McGinty, J. W. (2003). Properties of enteric coated sodium valproate pellets. Int. J. Pharm., 264, 85-96.
5. Crotts, G., Sheth, A., Twist, J., & Ghebre-Sellassie, I. (2001). Development of an enteric coating formulation and process for tablets primarily composed of a highly water-soluble organic acid. Eur. J. Pharm. Biopharm., 51, 71-76.
6. Felton, L. A., Haase, M. M., Shah, N. H., Zhang, G., Infeld, M. H., Malick, A. W., et al. (1995). Physical and enteric properties of soft gelatin capsules coated with Eudragit L30D-55. Int. J. Pharm., 113, 17-24.
7. Frenning, G., Tunón, Å., & Alderborn, G. (2003). Modelling of drug release from coated granular pellets. J. Control. Release, 92, 113-123.
8. Garcia, A. M., & Ghaly, E. S. (1996). Preliminary spherical agglomerates of water soluble drug using natural polymer and cross-linking technique. J. Control. Release, 40, 179-186.
9. Guo, H. X., Heinamaki, J., & Yliruusi, J. (2002). Amylopectin as a subcoating material improves the acidic resistance of enteric-coated pellets containing a freely soluble drug. Int. J. Pharm., 235, 79-86.
10. Hamdani, J., Moës, A. J., & Amighi, K. (2002). Development and evaluation of prolonged release pellets obtained by the melt pelletization process. Int. J. Pharm., 245, 167-177.
11. Heng, P. W. S., Hao, J., Chan, L. W., & Chew, S. H. (2007). Influences of osmotic agents in diffusion layer on drug release from multilayer coated pellets. Drug Dev. Ind. Pharm., 30, 213-220.
12. Lehmann, K. (1997). Chemistry and application properties of polymethacrylate coating systems. In J. W. McGinity, (Ed.), Aqueous polymeric coatings for pharmaceutical dosage forms (2nd ed., pp. 101-176). New York, Basel, Hong Kong: Marcel Dekker, Inc.
13. Li, S. P., & Feld, K. M. (1997). The effect of polymer coating systems on the preparation, tableting, and dissolution properties of sustained-release drug pellets. Drug Dev. Ind. Pharm., 23, 623-631.
14. Matthews, J. W., & Vergilio, G. (1989). Process for coating gelatin capsules, US Patent Issued on March, 28.
15. Ozturk, A. G., Ozturk, S. S., Palsson, B. O., Wheatley, T. A., & Dressman, J. B. (1990). Mechanism of release from pellets coated with an ethylcellulose-based film. J. Control. Release, 14, 203-213.
16. Phaechamud, T., & Ritthidej, G. C. (2007). Sustained-release from layered matrix system comprising chitosan and xanthan gum. Drug Dev. Ind. Pharm., 33, 595-605.
17. Sadeghi, F., Ford, J. L., Rubinstein, M. H., & Rajabi-Siahboomi, A. R. (2000). Comparative study of drug release from pellets coated with HPMC or surelease. Drug Dev. Ind. Pharm., 26, 651-660.
18. Sinchaipanid, N., Junyaprasert, V., & Mitrevej, A. (2004). Application of hotmelt coating for controlled release of propranolol hydrochloride pellets. Powder Tech., 141, 203-209.
19. Umprayn, K., Chitropas, P., & Amarekajorn, S. (1999). Development of terbutaline sulfate sustained-release coated pellets. Drug Dev. Ind. Pharm., 25, 477-491.
20. Zeng, H.-X., Cheng, G., Pan, W. -S., Zhong, G.-P., & Huang, M. (2007). Preparation of codeine-resinate and chlorpheniramine-resinate sustained-release suspension and its pharmacokinetic evaluation in beagle dogs. Drug Dev. Ind. Pharm., 33, 649-665.
21. Zheng, W. J., & James, W. (2003). Influence of Eudragit® NE30D blended with Eudragit L30 D-55 on the release of phenylpropanolamine hydrochloride from coated pellets. Drug Dev. Ind. Pharm., 29, 357-366.