Physicochemical interactions between drugs and superdisintegrants

Journal of Pharmacy and Pharmacology

Volumn 60, Issue 12, 2008, Pages 1583-1589

  Fransén, Nelly ^a   Morin, Malin ^a   Björk, Erik ^a   Edsman, Katarina ^a,b  

^a UPPSALA UNIVERSITY   (Sweden)

^b Q Med AB   (Sweden)

Author keywords

[No Author keywords available]

Indexed keywords

ALPRENOLOL; AMITRIPTYLINE; ATENOLOL; CETYLPYRIDINIUM SALT; CROSCARMELLOSE SODIUM; CROSPOVIDONE; DIPHENHYDRAMINE; DISINTEGRATING AGENT; ETHYL PARABEN; METHYL PARABEN; NAPROXEN; PROPYL PARABEN; SALICYLATE SODIUM; STARCH GLYCOLATE SODIUM; VERAPAMIL;

ARTICLE; BINDING AFFINITY; CHEMICAL STRUCTURE; DIFFUSION COEFFICIENT; DRUG ABSORPTION; DRUG BIOAVAILABILITY; DRUG CROSS REACTIVITY; DRUG RELEASE; HYDRATION; HYDROGEL; HYDROPHILICITY; IONIC STRENGTH; LIPOPHILICITY; PHYSICAL CHEMISTRY; SPECTROPHOTOMETRY;

EID: 56849084972     PISSN: 00223573     EISSN: None     Source Type: Journal    
DOI: 10.1211/jpp.60.12.0003     Document Type: Article

References (18)

1. Attwood, D. (1995) The mode of association of amphiphilic drugs in aqueous solution. Adv. Colloid. Interface Sci. 55: 271-303
2. Björk, E., Edman, P. (1990) Characterization of degradable starch microspheres as a nasal delivery system for drugs. Int. J. Pharm. 62: 187-192
3. Bramer, T., Paulsson, M., Edwards, K., Edsman, K. (2003) Cationic drug-surfactant mixtures: phase behavior and sustained release from gels. Pharm. Res. 20: 1661-1667
4. Bredenberg, S., Duberg, M., Lennernäs, B., Lennernäs, H., Pettersson, A., Westerberg, M., Nystrom, C. (2003) In vitro and in vivo evaluation of a new sublingual tablet system for rapid oromucosal absorption using fentanyl citrate as the active substance. Eur. J. Pharm. Sci. 20: 327-334
5. Chien, Y. W., Van Nostrand, P., Hurwitz, A. R., Shami, E. G. (1981) Drug-disintegrant interactions: binding of oxymorphone derivatives. J. Pharm. Sci. 70: 709-710
6. Edge, S., Belu, A. M., Potter, U. J., Steele, D. F., Young, P. M., Price, R., Staniforth, J. N. (2002) Chemical characterisation of sodium starch glycolate particles. Int. J. Pharm. 240: 67-78
7. Fransén, N., Björk, E., Nyström, C. (2007) Development and characterisation of interactive mixtures with a fine-particulate mucoadhesive carrier for nasal drug delivery. Eur. J. Pharm. Biopharm. 67: 370-376
8. Garcia-Mateos, I., Pérez, S., Velázquez, M. M. (1997) Interaction between cetyl pyridinium chloride and water-soluble polymers in aqueous solutions. J. Colloid. Interface. Sci. 194: 356-363
9. Hansson, P. (2006) Interaction between polyelectrolyte gels and surfactants of opposite charge. Curr. Opin. Colloid. Interface Sci. 11: 351-362
10. Higuchi, W. I. (1962) Analysis of data on the medicament release from ointments. J. Pharm. Sci. 51: 802-804
11. Hollenbeck, R. G. (1988) Bioavailability of phenylpropanolamine HCl from tablet dosage forms containing croscarmellose sodium. Int. J. Pharm. 47: 89-93
12. Hollenbeck, R. G., Mitrevej, K. T., Fan, A. C. (1983) Estimation of the extent of drug-excipient interactions involving croscarmellose sodium. J. Pharm. Sci. 72: 325-327
13. Huang, W. X., Desai, M., Tang, Q., Yang, R., Vivilecchia, R. V., Joshi, Y. (2006) Elimination of metformin-croscarmellose sodium interaction by competition. Int. J. Pharm. 311: 33-39
14. Paulsson, M., Edsman, K. (2002) Controlled drug release from gels using lipophilic interactions of charged substances with surfactants and polymers. J. Colloid. Interface Sci. 248: 194-200
15. Ritger, P. L., Peppas, N. A. (1987) A simple equation for description of solute release I. Fickian and non-Fickian release from non-swellable devices in the form of slabs, spheres, cylinders or discs. J. Control. Release 5: 23-36
16. th edn, Pharmaceutical Press, London, UK
17. SciFinder (2008) Property values were calculated using advanced chemistry development (ACD/Labs) software V8.14 for solaris ((c) 1994-2008 ACD/Labs) and delivered through SciFinder Scholar; reproduced with permission of CAS
18. Taboada, P., Pérez-Rodriguez, M., Attwood, D., Varela, L. M., Ruso, J. M., Mosquera, V. (2001) Self-association of verapamil in aqueous electrolyte solution. J. Colloid. Interface Sci. 241: 459-464