Catanionic Drug-Surfactant Mixtures: Phase Behavior and Sustained Release from Gels

Pharmaceutical Research

Volumn 20, Issue 10, 2003, Pages 1661-1667

  Bramer, Tobias ^a   Paulsson, Mattias ^a   Edwards, Katarina ^a   Edsman, Katarina ^a  

^a UPPSALA UNIVERSITY   (Sweden)

Author keywords

Catanionic mixtures; Gel; Phase diagram; Slow release; Surfactant

Indexed keywords

AMITRIPTYLINE; CARBOPOL 940; DIPHENHYDRAMINE; TETRACAINE;

ARTICLE; CONTROLLED RELEASE FORMULATION; DRUG RELEASE; FLOW KINETICS; GEL; MICELLE; PRIORITY JOURNAL; SUSTAINED RELEASE PREPARATION; TRANSMISSION ELECTRON MICROSCOPY;

AMITRIPTYLINE; ANIONS; CATIONS; DELAYED-ACTION PREPARATIONS; DIPHENHYDRAMINE; DRUG CARRIERS; DRUG COMPOUNDING; GELS; HYDROGEN-ION CONCENTRATION; MICELLES; PHARMACEUTICAL PREPARATIONS; PHASE TRANSITION; RHEOLOGY; SODIUM CHLORIDE; SODIUM DODECYL SULFATE; SURFACE-ACTIVE AGENTS; TEMPERATURE; TETRACAINE; TIME FACTORS;

EID: 0142042432     PISSN: 07248741     EISSN: None     Source Type: Journal    
DOI: 10.1023/A:1026103805283     Document Type: Article

References (27)

1. H. Fukuda, K. Kawata, and H. Okuda. Bilayer-forming ion-pair amphiphiles from single-chain surfactants. J. Am. Chem. Soc. 112: 1635-1637 (1990).
2. P. Jokela, B. Jönsson, and A. Kahn. Equilibria of catanionic surfactant-water systems. J. Phys. Chem. 91:3291-3298 (1987).
3. E. W. Kaler, A. K. Murthy, B. E. Rodriguez, and J. A. Zasadzinski. Spontaneous vesicle formation in aqueous mixtures of single-tailed surfactants. Science 245:1371-1374 (1989).
4. C. Tondre and C. Caillet. Properties of the amphiphilic films in mixed cationic/anionic vesicles: a comprehensive view from a literature analysis. Adv. Colloid Interface Sci. 93:115-134 (2001).
5. E. F. Marques, O. Regev, A. Khan, M. G. Miguel, and B. Lindman. Vesicle formation and general phase behaviour in the catanionic mixture SDS-DDAB-water. The anionic-rich side. J. Phys. Chem. B. 102:6746-6758 (1998).
6. E. F. Marques. Size and stability of catanionic vesicles: Effects of formation path, sonication, and aging. Langmuir 16:4798-4807 (2000).
7. L. L. Brasher and E. W. Kaler. A small-angle neutron scattering (SANS) contrast variation investigation of aggregate composition in catanionic surfactant mixtures. Langmuir 12:6270-6276 (1996).
8. J. M. Corkill, J. F. Goodman, S. P. Harrold, and J. R. Tate. Monolayers formed by mixtures of anionic and cationic surface-active agents. Trans. Faraday Soc. 63:247-256 (1996).
9. L. E. Bromberg. Enhanced nasal retention of hydrophobically modified polyelectrolytes. J. Pharm. Pharmacol. 53:109-114 (2001).
10. J. Carlfors, K. Edsman, R. Petersson, and K. Jörnving. Rheological evaluation of Gelrite in situ gels for ophthalmic use. Eur. J. Pharm. Sci. 6:113-119 (1998).
11. G. M. Grass and J. R. Robinson. Relationship of chemical structure to corneal penetration and influence of low viscosity solution on ocular bioavailability. J. Pharm. Sci. 73:1021-1027 (1984).
12. N. A. Peppas, P. Bures, W. Leobandung, and H. Ichikawa. Hydrogels in pharmaceutical formulations. Eur. J. Pharm. Biopharm. 50:27-46 (2000).
13. M. Paulsson and K. Edsman. Controlled drug release from gels using surfactant aggregates: II. Vesicles formed from mixtures of amphiphilic drugs and oppositely charged surfactants. Pharm. Res. 18:1586-1592 (2001).
14. R. M. Minardi, P. C. Schultz, and B. Vuano. Triangular phase diagram of the catanionic system dodecyltrimethylammonium bromide-disodium dodecanephosphonate-water. Colloids Surf. A. 197:167-172 (2002).
15. C. M. Wilkinson. Extended use of, and comments on, the drop-weight (drop-volume) technique for the determination of surface and interfacial tensions. J. Colloid Interface Sci. 40:14-26 (1972).
16. M. Almgren, K. Edwards, and G. Karlsson. Cryo transmission electron microscopy of liposomes and related structures. Colloid Surf. A-Physicochem. Eng. Asp. 174:3-21 (2000).
17. L. Bohlin. New instrumentation for advanced rheometry. Suppl. Rheol. Acta. 26:161-164 (1988).
18. W. I. Higuchi. Analysis of data on the medicament release from ointments. J. Pharm. Sci. 51:802-804 (1962).
19. P. L. Ritger and N. A. Peppas. A simple equation for description of solute release I. Fickian and non-Fickian release from non-swellable devices in the form of slabs, spheres, cylinders or discs. J. Control. Release 5:23-26 (1987).
20. M. Paulsson and K. Edsman. Controlled drug release from gels using surfactant aggregates: I. Effect of lipophilic interactions for a series of uncharged substances. J. Pharm. Sci. 90:1216-1225 (2001).
21. A. Sein and J. B. F. N. Engberts. Micelle to lamellar aggregate transition of an anionic surfactant in dilute aqueous solution induced by alkali metal chloride and tetraalkylammonium chloride salts. Langmuir 11: 455-465 (1995).
22. H. Hauser, N. Gains, and M. Muller. Vesiculation of unsonicated phospholipid dispersions containing phosphatidic acid by pH adjustment: Physicochemical properties of the resulting unilamellar vesicles. Biochemistry 22:4775-4781 (1983).
23. A. T. Florence, P. Arunothayanun, S. Kiri, M. S. Bernard, and I. F. Uchegbu. Some rheological properties of nonionic surfactant vesicles and the determination of surface hydration. J. Phys. Chem. B 103:1995-2000 (1999).
24. M. Paulsson and K. Edsman. Controlled drug release from gels using lipophilic interactions of charged substances with surfactants and polymers. J. Colloid Interface Sci. 248:194-200 (2002).
25. N. W. Taylor and E. B. Bagley. Dispersions or solutions? A mechanism for certain thickening agents. J. Appl. Polym. Sci. 18:2747-2761 (1974).
26. C. Caillet, M. Hebrant, and C. Tondre, Sodium octyl sulfate/cetyltrimethylammonium bromide catanionic vesicles: Aggregate composition and probe encapsulation. Langmuir 2000:9099-9102 (2000)
27. K. Östh, M. Paulsson, E. Björk, and K. Edsman. Evaluation of controlled drug release and absorption from gels on pig nasal mucosa in a horizontal Ussing chamber. J. Control. Release 83: 377-388 (2002).