Stimulation of Na+/Cl-coupled opioid peptide transport system in SK-N-SH cells by L-kyotorphin, an endogenous substrate for H+-coupled peptide transporter PEPT2

Drug Metabolism and Pharmacokinetics

Volumn 23, Issue 4, 2008, Pages 254-262

  Thakkar, Santoshanand V ^a   Miyauchi, Seiji ^a   Prasad, Puttur D ^a   Ganapathy, Vadivel ^a  

^a MEDICAL COLLEGE OF GEORGIA   (United States)

Author keywords

Kyotorphin; Opioid peptide transport; Opioidergic neurotransmission; PEPT2; SK N SH cell line; Stereospecificity

Indexed keywords

CHLORIDE ION; DELTORPHIN; KYOTORPHIN; OPIATE PEPTIDE; PEPTIDE TRANSPORTER 2; SODIUM ION; CHLORIDE; COTRANSPORTER; DELTORPHIN II, ALA(2); DELTORPHIN II, ALA(2)-; ENDORPHIN; GLYCYL GLYCYL PHENYLALANINAMIDE; GLYCYL-GLYCYL-PHENYLALANINAMIDE; HYDROGEN COUPLED OLIGOPEPTIDE TRANSPORTER PEPT2; HYDROGEN-COUPLED OLIGOPEPTIDE TRANSPORTER PEPT2; OLIGOPEPTIDE; SODIUM;

ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; HUMAN; HUMAN CELL; NERVE CELL; NEUROTRANSMISSION; NONHUMAN; PROTEIN EXPRESSION; PROTEIN TRANSPORT; STEREOSPECIFICITY; ANIMAL; CELL LINE; DOSE RESPONSE; DRUG EFFECT; METABOLISM; PHYSIOLOGY; STEREOISOMERISM; TRANSPORT AT THE CELLULAR LEVEL; XENOPUS LAEVIS;

ANIMALS; BIOLOGICAL TRANSPORT; CELL LINE; CHLORIDES; DOSE-RESPONSE RELATIONSHIP, DRUG; ENDORPHINS; HUMANS; OLIGOPEPTIDES; OPIOID PEPTIDES; SODIUM; STEREOISOMERISM; SYMPORTERS; XENOPUS LAEVIS;

EID: 56149085072     PISSN: 13474367     EISSN: 18800920     Source Type: Journal    
DOI: 10.2133/dmpk.23.254     Document Type: Article

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