-
1
-
-
0343029631
-
Chemistry and antitumor activities of camptothecins
-
Potmesil M, Kohn KW, editors, New York: Oxford University Press. pp
-
Wall ME, Wani MC. 1991. Chemistry and antitumor activities of camptothecins. In: Potmesil M, Kohn KW, editors. DNA topoisomerases in cancer. New York: Oxford University Press. pp 93-102.
-
(1991)
DNA topoisomerases in cancer
, pp. 93-102
-
-
Wall, M.E.1
Wani, M.C.2
-
2
-
-
0012345706
-
Twenty years later: Review of clinical trials with camptothecin sodium (NSC-100880)
-
Potmesil M, Pinedo H, editors, Boca Raton: CRC Press. p
-
Muggia FM. 1995. Twenty years later: Review of clinical trials with camptothecin sodium (NSC-100880). In: Potmesil M, Pinedo H, editors. Camptothecins: New anticancer agents. Boca Raton: CRC Press. p 44.
-
(1995)
Camptothecins: New anticancer agents
, pp. 44
-
-
Muggia, F.M.1
-
3
-
-
0032169909
-
Camptothecins: A review of their development and schedules of administration
-
O'Leary J, Muggian FM. 1998. Camptothecins: A review of their development and schedules of administration. Eur J Cancer 34:1500-1508.
-
(1998)
Eur J Cancer
, vol.34
, pp. 1500-1508
-
-
O'Leary, J.1
Muggian, F.M.2
-
4
-
-
0014895176
-
Preliminary pharmacological and clinical evaluation of camptothecin sodium (NCS 100880)
-
Gottlieb JA, Guarino AM, Call JB, Block JB. 1970. Preliminary pharmacological and clinical evaluation of camptothecin sodium (NCS 100880). Cancer Chemother Rep 54:461-470.
-
(1970)
Cancer Chemother Rep
, vol.54
, pp. 461-470
-
-
Gottlieb, J.A.1
Guarino, A.M.2
Call, J.B.3
Block, J.B.4
-
5
-
-
0018901322
-
Plant antitumor agents. 18. Synthesis and biological activity of camptothecin analogs
-
Wani MC, Ronman PE, Lindley JT, Wall ME. 1980. Plant antitumor agents. 18. Synthesis and biological activity of camptothecin analogs. J Med Chem 23:554-560.
-
(1980)
J Med Chem
, vol.23
, pp. 554-560
-
-
Wani, M.C.1
Ronman, P.E.2
Lindley, J.T.3
Wall, M.E.4
-
6
-
-
0024560495
-
Structure-activity study of the actions of camptothecin derivatives on mammalian topoisomerase I: Evidence for a specific receptor site and a relation to antitumor activity
-
Jaxel C, Kohn KW, Wani MC, Wall ME, Pommier Y. 1989. Structure-activity study of the actions of camptothecin derivatives on mammalian topoisomerase I: Evidence for a specific receptor site and a relation to antitumor activity. Cancer Res 49:1465-1469.
-
(1989)
Cancer Res
, vol.49
, pp. 1465-1469
-
-
Jaxel, C.1
Kohn, K.W.2
Wani, M.C.3
Wall, M.E.4
Pommier, Y.5
-
8
-
-
0031573854
-
Formulation study for the antitumor drug camptothecin: Liposomes, micellar solutions and a microemulsion
-
Cortesi R, Esposito E, Maietti A, Menegatti E, Nastruzzi C. 1997. Formulation study for the antitumor drug camptothecin: Liposomes, micellar solutions and a microemulsion. Int J Pharm 159:95-103.
-
(1997)
Int J Pharm
, vol.159
, pp. 95-103
-
-
Cortesi, R.1
Esposito, E.2
Maietti, A.3
Menegatti, E.4
Nastruzzi, C.5
-
9
-
-
33750065726
-
Camptothecin in sterically stabilized phospholipid micelles: A novel nanomedicine
-
Koo MO, Rubinstein I, Onyuksel HJ. 2006. Camptothecin in sterically stabilized phospholipid micelles: A novel nanomedicine. Nanosci Nanotechnol 6:2996-3000.
-
(2006)
Nanosci Nanotechnol
, vol.6
, pp. 2996-3000
-
-
Koo, M.O.1
Rubinstein, I.2
Onyuksel, H.J.3
-
10
-
-
0028264207
-
Stabilization of topotecan in low pH liposomes composed of distearoylphosphatidylcholine
-
Burke TG, Gao X. 1994. Stabilization of topotecan in low pH liposomes composed of distearoylphosphatidylcholine. J Pharm Sci 7:967-969.
-
(1994)
J Pharm Sci
, vol.7
, pp. 967-969
-
-
Burke, T.G.1
Gao, X.2
-
11
-
-
0035816198
-
The highly lipophilic DNA topoisomerase I inhibitor DB-67 displays elevated lactone levels in human blood and potent anticancer activity
-
Bom D, Curran DP, Zhang J, Zimmer SG, Bevins R, Kruszewski S, Howe JN, Bingcang A, Latus LJ, Burke TG. 2001. The highly lipophilic DNA topoisomerase I inhibitor DB-67 displays elevated lactone levels in human blood and potent anticancer activity. J Control Release 74:325-333.
-
(2001)
J Control Release
, vol.74
, pp. 325-333
-
-
Bom, D.1
Curran, D.P.2
Zhang, J.3
Zimmer, S.G.4
Bevins, R.5
Kruszewski, S.6
Howe, J.N.7
Bingcang, A.8
Latus, L.J.9
Burke, T.G.10
-
12
-
-
0036803284
-
Camptothecin delivery methods
-
Hatefi A, Amsden B. 2002. Camptothecin delivery methods. Pharm Res 19:1389-1399.
-
(2002)
Pharm Res
, vol.19
, pp. 1389-1399
-
-
Hatefi, A.1
Amsden, B.2
-
15
-
-
0030891273
-
Simple and versatile high-performance liquid chromatographic method for the simultaneous quantitation of the lactone and carboxylate forms of camptothecin anticancer drugs
-
Warner DL, Burke TG. 1997. Simple and versatile high-performance liquid chromatographic method for the simultaneous quantitation of the lactone and carboxylate forms of camptothecin anticancer drugs. J Chromatogr B Biomed Sci Appl 691:161-171.
-
(1997)
J Chromatogr B Biomed Sci Appl
, vol.691
, pp. 161-171
-
-
Warner, D.L.1
Burke, T.G.2
-
16
-
-
0032523144
-
Spectroscopic and biochemical characterisation of self-aggregates formed by antitumor drugs of the camptothecin family: Their possible role in the unique mode of drug action
-
Nabiev I, Fleury F, Kudelina I, Pommier Y, Charton F, Riou JF, Alix AJP, Manfait M. 1998. Spectroscopic and biochemical characterisation of self-aggregates formed by antitumor drugs of the camptothecin family: Their possible role in the unique mode of drug action. Biochem Pharmacol 55:1163-1174.
-
(1998)
Biochem Pharmacol
, vol.55
, pp. 1163-1174
-
-
Nabiev, I.1
Fleury, F.2
Kudelina, I.3
Pommier, Y.4
Charton, F.5
Riou, J.F.6
Alix, A.J.P.7
Manfait, M.8
-
17
-
-
0037018966
-
Preformulation studies of a novel camptothecin anticancer agent, CKD-602: Physicochemical characterization and hydrolytic equilibrium kinetics
-
Kim JH, Lee SK, Lim JL, Shin HJ, Hong C. 2002. Preformulation studies of a novel camptothecin anticancer agent, CKD-602: Physicochemical characterization and hydrolytic equilibrium kinetics. Int J Pharm 239:207-211.
-
(2002)
Int J Pharm
, vol.239
, pp. 207-211
-
-
Kim, J.H.1
Lee, S.K.2
Lim, J.L.3
Shin, H.J.4
Hong, C.5
-
18
-
-
21844480086
-
pH-dependent association of SN-38 with lipid bilayers of a novel liposomal formulation
-
Peikov V, Ugwu S, Parmar M, Zhang A, Ahmad I. 2005. pH-dependent association of SN-38 with lipid bilayers of a novel liposomal formulation. Int J Pharm 299:92-99.
-
(2005)
Int J Pharm
, vol.299
, pp. 92-99
-
-
Peikov, V.1
Ugwu, S.2
Parmar, M.3
Zhang, A.4
Ahmad, I.5
-
19
-
-
0015239588
-
Microviscosity and order in the hydrocarbon region of micelles and membranes determined with fluorescent probe. I. Synthetic micelles
-
Shinitzky M, Dianoux AC, Gitler C, Weber G. 1971. Microviscosity and order in the hydrocarbon region of micelles and membranes determined with fluorescent probe. I. Synthetic micelles. Biochemistry 10:2106-2113.
-
(1971)
Biochemistry
, vol.10
, pp. 2106-2113
-
-
Shinitzky, M.1
Dianoux, A.C.2
Gitler, C.3
Weber, G.4
-
20
-
-
0018378035
-
Light-scattering effects in the measurement of membrane microviscosity with diphenylhexatriene
-
Lentz BR, Moore BM, Barrow DA. 1979. Light-scattering effects in the measurement of membrane microviscosity with diphenylhexatriene. Biophys J 25:489-494.
-
(1979)
Biophys J
, vol.25
, pp. 489-494
-
-
Lentz, B.R.1
Moore, B.M.2
Barrow, D.A.3
-
21
-
-
0021983692
-
Structural basis of anthracycline selectivity for unilamellar phosphatidylcholine vesicles: An equilibrium binding stud
-
Burke TG, Tritton TR. 1985. Structural basis of anthracycline selectivity for unilamellar phosphatidylcholine vesicles: An equilibrium binding stud. Biochemistry 24:1768-1776.
-
(1985)
Biochemistry
, vol.24
, pp. 1768-1776
-
-
Burke, T.G.1
Tritton, T.R.2
-
22
-
-
0026641763
-
Liposomal stabilization of camptothecin's lactone ring
-
Burke TG, Staubus AE, Mishra AK. 1992. Liposomal stabilization of camptothecin's lactone ring. J Am Chem Soc 114:8318-8319.
-
(1992)
J Am Chem Soc
, vol.114
, pp. 8318-8319
-
-
Burke, T.G.1
Staubus, A.E.2
Mishra, A.K.3
-
23
-
-
0027930186
-
Differential interactions of camptothecin lactone and carboxylate forms with human blood components
-
Mi Z, Burke GT. 1994. Differential interactions of camptothecin lactone and carboxylate forms with human blood components. Biochemistry 33:10325-10336.
-
(1994)
Biochemistry
, vol.33
, pp. 10325-10336
-
-
Mi, Z.1
Burke, G.T.2
-
24
-
-
0027276081
-
Lipid bilayer partitioning and stability of camptothecin drugs
-
Burke TG, Mishra KA, Wani MC, Wall ME. 1993. Lipid bilayer partitioning and stability of camptothecin drugs. Biochemistry 32:5352-5364.
-
(1993)
Biochemistry
, vol.32
, pp. 5352-5364
-
-
Burke, T.G.1
Mishra, K.A.2
Wani, M.C.3
Wall, M.E.4
-
25
-
-
0032473430
-
Kinetics of lactone hydrolysis in antitumor drugs of camptothecin series as studied by fluorescence spectroscopy
-
Chourpa I, Millot JM, Sockalingum GD, Riou JF, Manfait M. 1998. Kinetics of lactone hydrolysis in antitumor drugs of camptothecin series as studied by fluorescence spectroscopy. Biochim Biophys Acta 1379:353-366.
-
(1998)
Biochim Biophys Acta
, vol.1379
, pp. 353-366
-
-
Chourpa, I.1
Millot, J.M.2
Sockalingum, G.D.3
Riou, J.F.4
Manfait, M.5
-
26
-
-
23144434579
-
A method to determine the incorporation capacity of camptothecin liposomes
-
Saetern AM, Flaten GE, Brand M. 2004. A method to determine the incorporation capacity of camptothecin liposomes. AAPS Pharm Sci Tech 5:40.
-
(2004)
AAPS Pharm Sci Tech
, vol.5
, pp. 40
-
-
Saetern, A.M.1
Flaten, G.E.2
Brand, M.3
-
27
-
-
0035343249
-
Interaction of topotecan, DNA topoisomerase I inhibitor, with double-stranded polydeoxyribonucleotides 1. Topotecan dimerization in solution
-
Strel'tsov SA, Grokhovskii SL, Kudelina IA, Oleinikov VA, Zhuze AL. 2001. Interaction of topotecan, DNA topoisomerase I inhibitor, with double-stranded polydeoxyribonucleotides 1. Topotecan dimerization in solution. Mol Biol 35:432-441.
-
(2001)
Mol Biol
, vol.35
, pp. 432-441
-
-
Strel'tsov, S.A.1
Grokhovskii, S.L.2
Kudelina, I.A.3
Oleinikov, V.A.4
Zhuze, A.L.5
-
28
-
-
0027096415
-
A kinetic and mechanictic study of the hydrolysis of camptothecin and some analogues
-
Fassberg J, Stella JV. 1992. A kinetic and mechanictic study of the hydrolysis of camptothecin and some analogues. J Pharm Sci 81:676-684.
-
(1992)
J Pharm Sci
, vol.81
, pp. 676-684
-
-
Fassberg, J.1
Stella, J.V.2
-
29
-
-
27644501575
-
New hints on the pH-driven tautomeric equilibria of the topotecan anticancer drug in aqueous solutions from an integrated spectroscopic and quantum-mechanical approach
-
Sanna N, Chillemi G, Grandi A, Castelli S, Desideri A, Barone VJ. 2005. New hints on the pH-driven tautomeric equilibria of the topotecan anticancer drug in aqueous solutions from an integrated spectroscopic and quantum-mechanical approach. Am Chem Soc 127:15429-15436.
-
(2005)
Am Chem Soc
, vol.127
, pp. 15429-15436
-
-
Sanna, N.1
Chillemi, G.2
Grandi, A.3
Castelli, S.4
Desideri, A.5
Barone, V.J.6
-
30
-
-
0031024171
-
Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings
-
Lipinski CA, Lombardo F, Dominy BW, Feeney PJ. 1997. Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings. Adv Drug Deliv Rev 23:3-25.
-
(1997)
Adv Drug Deliv Rev
, vol.23
, pp. 3-25
-
-
Lipinski, C.A.1
Lombardo, F.2
Dominy, B.W.3
Feeney, P.J.4
-
31
-
-
0019840171
-
Correlation of water solubility with octanol-water partition coefficient: A response
-
Yalkowsky SH, Valvani SC. 1981. Correlation of water solubility with octanol-water partition coefficient: A response. J Pharm Sci 70:1177-1178.
-
(1981)
J Pharm Sci
, vol.70
, pp. 1177-1178
-
-
Yalkowsky, S.H.1
Valvani, S.C.2
-
32
-
-
85031381167
-
-
Yalkowsky SH. 1999. Solubility and solubilization in aqueous media, New York, New York.
-
Yalkowsky SH. 1999. Solubility and solubilization in aqueous media, New York, New York.
-
-
-
-
33
-
-
0020599769
-
Solubility and partitioning VI: Octanol solubility and octanol-water partition coefficients
-
Yalkowsky SH, Valvani SC, Roseman TJ. 1983. Solubility and partitioning VI: Octanol solubility and octanol-water partition coefficients. J Pharm Sci 72:866-870.
-
(1983)
J Pharm Sci
, vol.72
, pp. 866-870
-
-
Yalkowsky, S.H.1
Valvani, S.C.2
Roseman, T.J.3
-
34
-
-
4744376004
-
Excited-state proton transfer reactions of 10-hydroxycamptothecin
-
Solntsev KM, Sullivan EN, Tolbert LM, Ashkenazi S, Leidderman P, Huppert D. 2004. Excited-state proton transfer reactions of 10-hydroxycamptothecin. J Am Chem Soc 126:12701-12708.
-
(2004)
J Am Chem Soc
, vol.126
, pp. 12701-12708
-
-
Solntsev, K.M.1
Sullivan, E.N.2
Tolbert, L.M.3
Ashkenazi, S.4
Leidderman, P.5
Huppert, D.6
-
35
-
-
0026099599
-
Synthesis of water soluble (aminoaklyl) camptothecin analogues: Inhibition of topoisomerase I and antitumor activity
-
Kingsbury W, Boehm J, Jakas D, Holden K, Hecht S, Gallgher G, Caranfa M, McCabe F, Faucette L, Johnson R, Hertzberg R. 1991. Synthesis of water soluble (aminoaklyl) camptothecin analogues: Inhibition of topoisomerase I and antitumor activity. J Med Chem 34:98-107.
-
(1991)
J Med Chem
, vol.34
, pp. 98-107
-
-
Kingsbury, W.1
Boehm, J.2
Jakas, D.3
Holden, K.4
Hecht, S.5
Gallgher, G.6
Caranfa, M.7
McCabe, F.8
Faucette, L.9
Johnson, R.10
Hertzberg, R.11
-
36
-
-
0037343958
-
Derivatives of camptothecin as albumin-binding prodrugs: Synthesis and antitumor efficacy
-
Warnecke A, Kratz F. 2003. Derivatives of camptothecin as albumin-binding prodrugs: Synthesis and antitumor efficacy. Bioconjugate Chem 14:377-387.
-
(2003)
Bioconjugate Chem
, vol.14
, pp. 377-387
-
-
Warnecke, A.1
Kratz, F.2
-
37
-
-
0011071824
-
Formation and properties of 1000-A-diameter, single-bilayer phospholipid vesicles
-
Enoch GH, Strittmatter P. 1979. Formation and properties of 1000-A-diameter, single-bilayer phospholipid vesicles. Proc Natl Acad Sci USA 76:145-149.
-
(1979)
Proc Natl Acad Sci USA
, vol.76
, pp. 145-149
-
-
Enoch, G.H.1
Strittmatter, P.2
-
38
-
-
33750087849
-
Incorporation of camptothecin into N-phthaloyl chitosan-g-mPEG self-assembly micellar system
-
Opanasopit P, Ngawhirunpat T, Chaidedgumjorn A, Rojanarata T, Apirakaramwong A, Phongying S, Choochottiros C, Chirachanchai S. 2006. Incorporation of camptothecin into N-phthaloyl chitosan-g-mPEG self-assembly micellar system. Eur J Pharm Biopharm 64:269-276.
-
(2006)
Eur J Pharm Biopharm
, vol.64
, pp. 269-276
-
-
Opanasopit, P.1
Ngawhirunpat, T.2
Chaidedgumjorn, A.3
Rojanarata, T.4
Apirakaramwong, A.5
Phongying, S.6
Choochottiros, C.7
Chirachanchai, S.8
-
39
-
-
19444377195
-
Influence of serum and albumins from different species on stability of camptothecin loaded micelles
-
Opanasopit P, Yokoyama M, Watanabe M, Kawano K, Maitani Y, Okano T. 2005. Influence of serum and albumins from different species on stability of camptothecin loaded micelles. J Control Release 104:313-321.
-
(2005)
J Control Release
, vol.104
, pp. 313-321
-
-
Opanasopit, P.1
Yokoyama, M.2
Watanabe, M.3
Kawano, K.4
Maitani, Y.5
Okano, T.6
|