SCOPUS 정보 검색 플랫폼

Volumn 6, Issue 22, 2008, Pages 4108-4119

Effects of C-17 heterocyclic substituents on the anticancer activity of 2-ethylestra-1,3,5(10)-triene-3-O-sulfamates: Synthesis, in vitro evaluation and computational modelling

(10) Jourdan, Fabrice a Bubert, Christian a Leese, Mathew P a Smith, Andrew a Ferrandis, Eric b Regis Lydi, Sandra b Newman, Simon P c Purohit, Atul c Reed, Michael J c Potter, Barry V L a

a University of Bath (United Kingdom)

b Institut de Recherche Henri Beaufour (France)

c ST MARY S HOSPITAL (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

BINDING ENERGY; BINDING SITES; CELLS; NITROGEN COMPOUNDS; TUMORS;

ACTIVE COMPOUNDS; ANTICANCER ACTIVITIES; BOND ACCEPTORS; CANCER CELLS; COLCHICINE BINDINGS; COMPUTATIONAL MODELLING; DIFFERENT MODES; ELECTRON DENSITIES; HETEROCYCLIC RINGS; IN VITRO; IN VITRO ACTIVITIES; IN-VIVO; OPTIMAL ACTIVITIES; OXAZOLE; POTENT ACTIVITIES; PROLIFERATIVE ACTIVITIES; PROSTATE CANCER CELLS; SULFAMATE; SULFAMATES; TUMOURS;

COMPLEXATION;

ANTINEOPLASTIC AGENT; HETEROCYCLIC COMPOUND; SULFAMIC ACID; SULFONIC ACID DERIVATIVE; TUBULIN;

ARTICLE; BINDING SITE; CELL PROLIFERATION; CHEMICAL STRUCTURE; CHEMISTRY; COMPUTER SIMULATION; DRUG EFFECT; ELECTRON; HUMAN; HYDROGEN BOND; METABOLISM; SYNTHESIS; TUMOR CELL LINE;

ANTINEOPLASTIC AGENTS; BINDING SITES; CELL LINE, TUMOR; CELL PROLIFERATION; COMPUTER SIMULATION; ELECTRONS; HETEROCYCLIC COMPOUNDS; HUMANS; HYDROGEN BONDING; MODELS, MOLECULAR; SULFONIC ACIDS; TUBULIN;

EID: 55549129602 PISSN: 14770520 EISSN: None Source Type: Journal
DOI: 10.1039/b810300c Document Type: Article

Times cited : (33)

References (30)

1
- 2442442849
- -3138
- M. P. Leese S. P. Newman A. Purohit M. J. Reed B. V. L. Potter Bioorg. Med. Chem. Lett. 2004 14 3135 3138
- (2004) Bioorg. Med. Chem. Lett. , vol.14 , pp. 3135
- Leese, M.P.¹ Newman, S.P.² Purohit, A.³ Reed, M.J.⁴ Potter, B.V.L.⁵

2
- 41649119942
- -1308
- M. P. Leese F. L. Jourdan K. Gaukroger M. F. Mahon S. P. Newman P. A. Foster C. Stengel S. Regis-Lydi E. Ferrandis A. D. Fiore G. De Simone C. T. Supuran A. Purohit M. J. Reed B. V. L. Potter J. Med. Chem. 2008 51 1295 1308
- (2008) J. Med. Chem. , vol.51 , pp. 1295
- Leese, M.P.¹ Jourdan, F.L.² Gaukroger, K.³ Mahon, M.F.⁴ Newman, S.P.⁵ Foster, P.A.⁶ Stengel, C.⁷ Regis-Lydi, S.⁸ Ferrandis, E.⁹ Fiore, A.D.¹⁰ De Simone, G.¹¹ Supuran, C.T.¹² Purohit, A.¹³ Reed, M.J.¹⁴ Potter, B.V.L.¹⁵

3
- 33845953699
- -7696
- M. P. Leese B. Leblond A. Smith S. P. Newman A. Di Fiore G. De Simone C. T. Supuran A. Purohit M. J. Reed B. V. L. Potter J. Med. Chem. 2006 49 7683 7696
- (2006) J. Med. Chem. , vol.49 , pp. 7683
- Leese, M.P.¹ Leblond, B.² Smith, A.³ Newman, S.P.⁴ Di Fiore, A.⁵ De Simone, G.⁶ Supuran, C.T.⁷ Purohit, A.⁸ Reed, M.J.⁹ Potter, B.V.L.¹⁰

4
- 23444441492
- -5256
- M. P. Leese H. A. Hejaz M. F. Mahon S. P. Newman A. Purohit M. J. Reed B. V. L. Potter J. Med. Chem. 2005 48 5243 5256
- (2005) J. Med. Chem. , vol.48 , pp. 5243
- Leese, M.P.¹ Hejaz, H.A.² Mahon, M.F.³ Newman, S.P.⁴ Purohit, A.⁵ Reed, M.J.⁶ Potter, B.V.L.⁷

5
- 18144419334
- -251
- M. P. Leese B. Leblond S. P. Newman A. Purohit M. J. Reed B. V. L. Potter J. Steroid Biochem. Mol. Biol. 2005 94 239 251
- (2005) J. Steroid Biochem. Mol. Biol. , vol.94 , pp. 239
- Leese, M.P.¹ Leblond, B.² Newman, S.P.³ Purohit, A.⁴ Reed, M.J.⁵ Potter, B.V.L.⁶

6
- 0033956376
- -589
- A. Purohit H. A. Hejaz L. Walden L. Carthy-Morrogh G. Packham B. V. L. Potter M. J. Reed Int. J. Cancer 2000 85 584 589
- (2000) Int. J. Cancer , vol.85 , pp. 584
- Purohit, A.¹ Hejaz, H.A.² Walden, L.³ Carthy-Morrogh, L.⁴ Packham, G.⁵ Potter, B.V.L.⁶ Reed, M.J.⁷

7
- 0034307330
- -5450
- L. MacCarthy-Morrogh P. A. Townsend A. Purohit H. A. M. Hejaz B. V. L. Potter M. J. Reed G. Packham Cancer Res. 2000 60 5441 5450
- (2000) Cancer Res. , vol.60 , pp. 5441
- MacCarthy-Morrogh, L.¹ Townsend, P.A.² Purohit, A.³ Hejaz, H.A.M.⁴ Potter, B.V.L.⁵ Reed, M.J.⁶ Packham, G.⁷

8
- 1542510122
- -540
- S. P. Newman M. P. Leese A. Purohit D. R. James C. E. Rennie B. V. L. Potter M. J. Reed Int. J. Cancer 2004 109 533 540
- (2004) Int. J. Cancer , vol.109 , pp. 533
- Newman, S.P.¹ Leese, M.P.² Purohit, A.³ James, D.R.⁴ Rennie, C.E.⁵ Potter, B.V.L.⁶ Reed, M.J.⁷

9
- 34247604099
- -1376
- S. K. Chander P. A. Foster M. P. Leese S. P. Newman B. V. L. Potter A. Purohit M. J. Reed Br. J. Cancer 2007 96 1368 1376
- (2007) Br. J. Cancer , vol.96 , pp. 1368
- Chander, S.K.¹ Foster, P.A.² Leese, M.P.³ Newman, S.P.⁴ Potter, B.V.L.⁵ Purohit, A.⁶ Reed, M.J.⁷

10
- 1642319678
- -937
- C. R. Ireson S. K. Chander A. Purohit S. Perera S. P. Newman D. Parish M. P. Leese A. C. Smith B. V. L. Potter M. J. Reed Br. J. Cancer 2004 90 932 937
- (2004) Br. J. Cancer , vol.90 , pp. 932
- Ireson, C.R.¹ Chander, S.K.² Purohit, A.³ Perera, S.⁴ Newman, S.P.⁵ Parish, D.⁶ Leese, M.P.⁷ Smith, A.C.⁸ Potter, B.V.L.⁹ Reed, M.J.¹⁰

11
- 35748981525
- -2809
- G. Kesisis H. Broxterman G. Giaccone Curr. Pharm. Des. 2007 13 2795 2809
- (2007) Curr. Pharm. Des. , vol.13 , pp. 2795
- Kesisis, G.¹ Broxterman, H.² Giaccone, G.³

12
- 0028220858
- -239
- T. Fotsis Y. Zhang M. S. Pepper H. Adlercreutz R. Montesano P. P. Nawroth L. Schweigerer Nature 1994 368 237 239
- (1994) Nature , vol.368 , pp. 237
- Fotsis, T.¹ Zhang, Y.² Pepper, M.S.³ Adlercreutz, H.⁴ Montesano, R.⁵ Nawroth, P.P.⁶ Schweigerer, L.⁷

13
- 0028331925
- -3968
- R. J. D'Amato C. M. Lin E. Flynn J. Folkman E. Hamel Proc. Natl. Acad. Sci. U. S. A. 1994 91 3964 3968
- (1994) Proc. Natl. Acad. Sci. U. S. A. , vol.91 , pp. 3964
- D'Amato, R.J.¹ Lin, C.M.² Flynn, E.³ Folkman, J.⁴ Hamel, E.⁵

14
- 3242808959
- -332
- L. Wood M. P. Leese A. Mouzakiti A. Purohit B. V. L. Potter M. J. Reed G. Packham Apoptosis 2004 9 323 332
- (2004) Apoptosis , vol.9 , pp. 323
- Wood, L.¹ Leese, M.P.² Mouzakiti, A.³ Purohit, A.⁴ Potter, B.V.L.⁵ Reed, M.J.⁶ Packham, G.⁷

15
- 31544434859
- -330
- S. P. Newman C. R. Ireson H. J. Tutill J. M. Day M. F. Parsons M. P. Leese B. V. L. Potter M. J. Reed A. Purohit Cancer Res. 2006 66 324 330
- (2006) Cancer Res. , vol.66 , pp. 324
- Newman, S.P.¹ Ireson, C.R.² Tutill, H.J.³ Day, J.M.⁴ Parsons, M.F.⁵ Leese, M.P.⁶ Potter, B.V.L.⁷ Reed, M.J.⁸ Purohit, A.⁹

16
- 0037904915
- -914
- Y. T. Ho A. Purohit N. Vicker S. P. Newman J. J. Robinson M. P. Leese D. Ganeshapillai L. W. Woo B. V. L. Potter M. J. Reed Biochem. Biophys. Res. Commun. 2003 305 909 914
- (2003) Biochem. Biophys. Res. Commun. , vol.305 , pp. 909
- Ho, Y.T.¹ Purohit, A.² Vicker, N.³ Newman, S.P.⁴ Robinson, J.J.⁵ Leese, M.P.⁶ Ganeshapillai, D.⁷ Woo, L.W.⁸ Potter, B.V.L.⁹ Reed, M.J.¹⁰

17
- 0029620774
- -403
- W. Elger S. Schwarz A. Hedden G. Reddersen B. Schneider J. Steroid Biochem. Mol. Biol. 1995 55 395 403
- (1995) J. Steroid Biochem. Mol. Biol. , vol.55 , pp. 395
- Elger, W.¹ Schwarz, S.² Hedden, A.³ Reddersen, G.⁴ Schneider, B.⁵

18
- 42549148009
- -463
- J. Y. Winum M. Rami A. Scozzafava J. L. Montero C. Supuran Med. Res. Rev. 2008 28 445 463
- (2008) Med. Res. Rev. , vol.28 , pp. 445
- Winum, J.Y.¹ Rami, M.² Scozzafava, A.³ Montero, J.L.⁴ Supuran, C.⁵

19
- 37049031003
- -1682
- S. P. Newman P. A. Foster Y. T. Ho J. M. Day B. Raobaikady P. G. Kasprzyk M. P. Leese B. V. L. Potter M. J. Reed A. Purohit Br. J. Cancer 2007 97 1673 1682
- (2007) Br. J. Cancer , vol.97 , pp. 1673
- Newman, S.P.¹ Foster, P.A.² Ho, Y.T.³ Day, J.M.⁴ Raobaikady, B.⁵ Kasprzyk, P.G.⁶ Leese, M.P.⁷ Potter, B.V.L.⁸ Reed, M.J.⁹ Purohit, A.¹⁰

20
- 38949192004
- -606
- S. P. Newman P. A. Foster C. Stengel J. M. Day Y. T. Ho J. G. Judde M. Lassalle G. Prévost M. P. Leese B. V. L. Potter M. J. Reed A. Purohit Clin. Cancer Res. 2008 14 597 606
- (2008) Clin. Cancer Res. , vol.14 , pp. 597
- Newman, S.P.¹ Foster, P.A.² Stengel, C.³ Day, J.M.⁴ Ho, Y.T.⁵ Judde, J.G.⁶ Lassalle, M.⁷ Prévost, G.⁸ Leese, M.P.⁹ Potter, B.V.L.¹⁰ Reed, M.J.¹¹ Purohit, A.¹²

21
- 0034596449
- -7051
- M. Okada S. Iwashita N. Koizumi Tetrahedron Lett. 2000 41 7047 7051
- (2000) Tetrahedron Lett. , vol.41 , pp. 7047
- Okada, M.¹ Iwashita, S.² Koizumi, N.³

22
- 84949695566
- -564
- S. Ohira Synth. Commun. 1989 19 561 564
- (1989) Synth. Commun. , vol.19 , pp. 561
- Ohira, S.¹

23
- 0027366650
- -3250
- G. D. Diana D. Cutcliffe D. L. Volkots J. P. Mallamo T. R. Bailey N. Vescio R. C. Oglesby T. J. Nitz J. Wetzel V. Giranda J. Med. Chem. 1993 36 3240 3250
- (1993) J. Med. Chem. , vol.36 , pp. 3240
- Diana, G.D.¹ Cutcliffe, D.² Volkots, D.L.³ Mallamo, J.P.⁴ Bailey, T.R.⁵ Vescio, N.⁶ Oglesby, R.C.⁷ Nitz, T.J.⁸ Wetzel, J.⁹ Giranda, V.¹⁰

24
- 37049116588
- SYBYL 7.0, Tripos Inc., 1699 South Hanley Rd., St. Louis, Missouri, 63144, USA. Ref Type: Generic -1666
- R. K. Bartlett I. R. Humphrey J. Chem. Soc. C 1967 1664 1666
- (1967) J. Chem. Soc. C , pp. 1664
- Bartlett, R.K.¹ Humphrey, I.R.²

25
- 33744994054
- Planaria Software LLC, Seattle, WA
- ArgusLab 4.0.1, Mark A. Thompson, Planaria Software LLC, Seattle, WA http://www.Arguslab.Com
- ArgusLab 4.0.1
- Thompson Mark, A.¹

26
- 0027055934
- -4794
- Y. S. Lo J. C. Nolan T. H. Maren W. J. Welstead, Jr. D. F. Gripshover D. A. Shamblee J. Med. Chem. 1992 35 4790 4794
- (1992) J. Med. Chem. , vol.35 , pp. 4790
- Lo, Y.S.¹ Nolan, J.C.² Maren, T.H.³ Welstead Jr. W., J.⁴ Gripshover, D.F.⁵ Shamblee, D.A.⁶

27
- 1642401199
- -202
- R. B. Ravelli B. Gigant P. A. Curmi I. Jourdain S. Lachkar A. Sobel M. Knossow Nature 2004 428 198 202
- (2004) Nature , vol.428 , pp. 198
- Ravelli, R.B.¹ Gigant, B.² Curmi, P.A.³ Jourdain, I.⁴ Lachkar, S.⁵ Sobel, A.⁶ Knossow, M.⁷

28
- 84926319125
- -1341
- R. Appel G. Berger Chem. Ber. 1958 91 1339 1341
- (1958) Chem. Ber. , vol.91 , pp. 1339
- Appel, R.¹ Berger, G.²

29
- 0029876168
- -88
- L. W. Woo M. Lightowler A. Purohit M. J. Reed B. V. L. Potter J. Steroid Biochem. Mol. Biol. 1996 57 79 88
- (1996) J. Steroid Biochem. Mol. Biol. , vol.57 , pp. 79
- Woo, L.W.¹ Lightowler, M.² Purohit, A.³ Reed, M.J.⁴ Potter, B.V.L.⁵

30
- 34548498111
- -4443
- C. Bubert M. P. Leese M. F. Mahon E. Ferrandis S. Regis-Lydi P. G. Kasprzyk S. P. Newman Y. T. Ho A. Purohit M. J. Reed B. V. L. Potter J. Med. Chem. 2007 50 4431 4443
- (2007) J. Med. Chem. , vol.50 , pp. 4431
- Bubert, C.¹ Leese, M.P.² Mahon, M.F.³ Ferrandis, E.⁴ Regis-Lydi, S.⁵ Kasprzyk, P.G.⁶ Newman, S.P.⁷ Ho, Y.T.⁸ Purohit, A.⁹ Reed, M.J.¹⁰ Potter, B.V.L.¹¹

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