-
1
-
-
0009644628
-
Some quantitative uses of drug antagonists
-
Arunlakshana O, Schild HO (1959) Some quantitative uses of drug antagonists. Br J Pharmacol 14:48-58.
-
(1959)
Br J Pharmacol
, vol.14
, pp. 48-58
-
-
Arunlakshana, O.1
Schild, H.O.2
-
2
-
-
35349010056
-
Variation in GABRA2 predicts drinking behavior in project MATCH subjects
-
Bauer LO, Covault J, Harel O, Das S, Gelernter J, Anton R, Kranzler HR (2007) Variation in GABRA2 predicts drinking behavior in project MATCH subjects. Alcohol Clin Exp Res 31:1780-1787.
-
(2007)
Alcohol Clin Exp Res
, vol.31
, pp. 1780-1787
-
-
Bauer, L.O.1
Covault, J.2
Harel, O.3
Das, S.4
Gelernter, J.5
Anton, R.6
Kranzler, H.R.7
-
3
-
-
0031407009
-
Discriminative stimulus properties of ethanol in the rat: Differential effects of selective and nonselective benzodiazepine receptor agonists
-
Bienkowski P, Iwinska K, Stefanski R, Kostowski W (1997) Discriminative stimulus properties of ethanol in the rat: differential effects of selective and nonselective benzodiazepine receptor agonists. Pharmacol Biochem Behav 58:969-973.
-
(1997)
Pharmacol Biochem Behav
, vol.58
, pp. 969-973
-
-
Bienkowski, P.1
Iwinska, K.2
Stefanski, R.3
Kostowski, W.4
-
4
-
-
0002639656
-
Drug discrimination: Behavioral, pharmacological, and molecular mechanisms of discriminative drug effects
-
Goldman SR, Stolerman IP eds, pp, Academic Press, New York
-
Colpaert FC (1986) Drug discrimination: behavioral, pharmacological, and molecular mechanisms of discriminative drug effects, in Behavior Analysis of Drug Dependence (Goldman SR, Stolerman IP eds), pp 161-193. Academic Press, New York.
-
(1986)
Behavior Analysis of Drug Dependence
, pp. 161-193
-
-
Colpaert, F.C.1
-
5
-
-
39149145477
-
Markers in the 5'-region of GABRG1 associate to alcohol dependence and are in linkage disequilibrium with markers in the adjacent GABRA2 gene
-
Covault J, Gelernter J, Jensen K, Anton R, Kranzler HR (2008) Markers in the 5'-region of GABRG1 associate to alcohol dependence and are in linkage disequilibrium with markers in the adjacent GABRA2 gene. Neuropsycho-pharmacology 33:837-848.
-
(2008)
Neuropsycho-pharmacology
, vol.33
, pp. 837-848
-
-
Covault, J.1
Gelernter, J.2
Jensen, K.3
Anton, R.4
Kranzler, H.R.5
-
6
-
-
0000440517
-
BZ1 receptor specific ligands. Synthesis and biological properties of BCCt, a BZ1 receptor subtype specific antagonist
-
Cox ED, Hagen TJ, McKernan RM, Cook JM (1995) BZ1 receptor specific ligands. Synthesis and biological properties of BCCt, a BZ1 receptor subtype specific antagonist. Med Chem Res 5:710-718.
-
(1995)
Med Chem Res
, vol.5
, pp. 710-718
-
-
Cox, E.D.1
Hagen, T.J.2
McKernan, R.M.3
Cook, J.M.4
-
7
-
-
0022613409
-
Zolpidem, a novel nonbenzodiazepine hypnotic. I. Neuropharmacological and behavioral effects
-
Depoortere H, Zivkovic B, Lloyd KG, Sanger DJ, Perrault G, Langer SZ, Bartholini G (1986) Zolpidem, a novel nonbenzodiazepine hypnotic. I. Neuropharmacological and behavioral effects. J Pharmacol Exp Ther 237:649-658.
-
(1986)
J Pharmacol Exp Ther
, vol.237
, pp. 649-658
-
-
Depoortere, H.1
Zivkovic, B.2
Lloyd, K.G.3
Sanger, D.J.4
Perrault, G.5
Langer, S.Z.6
Bartholini, G.7
-
8
-
-
0025641577
-
Zolpidem and triazolam in humans: Behavioral and subjective effects and abuse liability
-
Evans SM, Funderburk FR, Griffiths RR (1990) Zolpidem and triazolam in humans: behavioral and subjective effects and abuse liability. J Pharmacol Exp Ther 255:1246-1255.
-
(1990)
J Pharmacol Exp Ther
, vol.255
, pp. 1246-1255
-
-
Evans, S.M.1
Funderburk, F.R.2
Griffiths, R.R.3
-
9
-
-
0030744208
-
Attenuation of the discriminative stimulus effects of ethanol by the benzodiazepine partial inverse agonist Ro 15-4513
-
Gatto GJ, Grant KA (1997) Attenuation of the discriminative stimulus effects of ethanol by the benzodiazepine partial inverse agonist Ro 15-4513. Behav Pharmacol 8:139-146.
-
(1997)
Behav Pharmacol
, vol.8
, pp. 139-146
-
-
Gatto, G.J.1
Grant, K.A.2
-
10
-
-
0032869313
-
Strategies for understanding the pharmacological effects of ethanol with drug discrimination procedures
-
Grant KA (1999) Strategies for understanding the pharmacological effects of ethanol with drug discrimination procedures. Pharmacol Biochem Behav 64:261-267.
-
(1999)
Pharmacol Biochem Behav
, vol.64
, pp. 261-267
-
-
Grant, K.A.1
-
11
-
-
0029935508
-
Ethanol-like discriminative stimulus effects of the neurosteroid 3α-hydroxy-5α- pregnan-20-one in female Macaca fascicularis monkeys
-
Grant KA, Azarov A, Bowen CA, Mirkis S, Purdy RH (1996) Ethanol-like discriminative stimulus effects of the neurosteroid 3α-hydroxy-5α- pregnan-20-one in female Macaca fascicularis monkeys. Psychopharmacology 124:340-346.
-
(1996)
Psychopharmacology
, vol.124
, pp. 340-346
-
-
Grant, K.A.1
Azarov, A.2
Bowen, C.A.3
Mirkis, S.4
Purdy, R.H.5
-
12
-
-
0031018087
-
Discriminative stimulus effects of ethanol and 3α-hydroxy-5α-pregnan-20-one in relation to menstrual cycle phase in cynomolgus monkeys (Macaca fascicularis)
-
Grant KA, Azarov A, Shively CA, Purdy RH (1997) Discriminative stimulus effects of ethanol and 3α-hydroxy-5α-pregnan-20-one in relation to menstrual cycle phase in cynomolgus monkeys (Macaca fascicularis). Psychopharmacology 130:59-68.
-
(1997)
Psychopharmacology
, vol.130
, pp. 59-68
-
-
Grant, K.A.1
Azarov, A.2
Shively, C.A.3
Purdy, R.H.4
-
15
-
-
0030024882
-
Cloning of cDNAs encoding the human γ-aminobutyric acid type A receptor α6 subunit and characterization of the pharmacology of recombinant α6-containing receptors
-
Hadingham KL, Garrett EM, Wafford KA, Bain C, Heavens RP, Sirinathsinghji Dalip JS, Whiting PJ (1996) Cloning of cDNAs encoding the human γ-aminobutyric acid type A receptor α6 subunit and characterization of the pharmacology of recombinant α6-containing receptors. Mol Pharmacol 49:253-259.
-
(1996)
Mol Pharmacol
, vol.49
, pp. 253-259
-
-
Hadingham, K.L.1
Garrett, E.M.2
Wafford, K.A.3
Bain, C.4
Heavens, R.P.5
Sirinathsinghji Dalip, J.S.6
Whiting, P.J.7
-
18
-
-
0023220764
-
Effect of an imidazobenzodiazepine, Ro15-4513, on the incoordination and hypothermia produced by ethanol and pentobarbital
-
Hoffman PL, Tabakoff B, Szabo G, Suzdak PD, Paul SM (1987) Effect of an imidazobenzodiazepine, Ro15-4513, on the incoordination and hypothermia produced by ethanol and pentobarbital. Life Sci 41:611-619.
-
(1987)
Life Sci
, vol.41
, pp. 611-619
-
-
Hoffman, P.L.1
Tabakoff, B.2
Szabo, G.3
Suzdak, P.D.4
Paul, S.M.5
-
19
-
-
0001072453
-
Discriminative stimulus effects of drugs: Relationship to potential for abuse
-
Adler MW, Cowan A eds, pp, Wiley-Liss, New York
-
Holtzman SG (1990) Discriminative stimulus effects of drugs: relationship to potential for abuse, in Modern Methods in Pharmacology, Vol. 6 (Adler MW, Cowan A eds), pp 193-210. Wiley-Liss, New York.
-
(1990)
Modern Methods in Pharmacology
, vol.6
, pp. 193-210
-
-
Holtzman, S.G.1
-
20
-
-
0345638097
-
The effects of zolpidem on motor activity, ethanol drinking and ethanol discriminative stimulus in rats
-
Jankowska E, Iwiniska K, Stefanski R, Biekowski P, Kostowski W (1996) The effects of zolpidem on motor activity, ethanol drinking and ethanol discriminative stimulus in rats. Behav Pharmacol 7:54.
-
(1996)
Behav Pharmacol
, vol.7
, pp. 54
-
-
Jankowska, E.1
Iwiniska, K.2
Stefanski, R.3
Biekowski, P.4
Kostowski, W.5
-
21
-
-
0029010943
-
International union of pharmacology committee on receptor nomenclature and drug classification. IX. Recommendations on terms and symbols in quantitative pharmacology
-
Jenkinson DH, Barnard EA, Hoyer D, Humphrey PPA, Leff P, Shankley NP (1995) International union of pharmacology committee on receptor nomenclature and drug classification. IX. Recommendations on terms and symbols in quantitative pharmacology. Pharmacol Rev 47:255-266.
-
(1995)
Pharmacol Rev
, vol.47
, pp. 255-266
-
-
Jenkinson, D.H.1
Barnard, E.A.2
Hoyer, D.3
Humphrey, P.P.A.4
Leff, P.5
Shankley, N.P.6
-
22
-
-
2342510931
-
Clinical neuropharmacology of drugs of abuse: A comparison of drug-discrimination and subject-report measures
-
Kelly TH, Stoops WW, Perry AS, Prendergast MA, Rush CR (2003) Clinical neuropharmacology of drugs of abuse: a comparison of drug-discrimination and subject-report measures. Behav Cog Neurosci Rev 2:227-260.
-
(2003)
Behav Cog Neurosci Rev
, vol.2
, pp. 227-260
-
-
Kelly, T.H.1
Stoops, W.W.2
Perry, A.S.3
Prendergast, M.A.4
Rush, C.R.5
-
24
-
-
0028338548
-
Impact of β and γ variants on ligand-binding properties of γ-aminobutyric acid type A receptors
-
Lüddens H, Seeburg PH, Korpi ER (1994) Impact of β and γ variants on ligand-binding properties of γ-aminobutyric acid type A receptors. Mol Pharmacol 45:810-814.
-
(1994)
Mol Pharmacol
, vol.45
, pp. 810-814
-
-
Lüddens, H.1
Seeburg, P.H.2
Korpi, E.R.3
-
28
-
-
0023182676
-
The effect of the imidazodiazepine Ro 15-4513 on the anticonvulsant effects of diazepam, sodium pentobarbital and ethanol
-
Nutt DJ, Lister RG (1987) The effect of the imidazodiazepine Ro 15-4513 on the anticonvulsant effects of diazepam, sodium pentobarbital and ethanol. Brain Res 413:193-196.
-
(1987)
Brain Res
, vol.413
, pp. 193-196
-
-
Nutt, D.J.1
Lister, R.G.2
-
29
-
-
0032588314
-
2 values of benzodiazepine antagonists and partial agonists in monkeys
-
2 values of benzodiazepine antagonists and partial agonists in monkeys. J Pharmacol Exp Ther 290:1222-1229.
-
(1999)
J Pharmacol Exp Ther
, vol.290
, pp. 1222-1229
-
-
Paronis, C.A.1
Bergman, J.2
-
30
-
-
0029145572
-
Ro 15-4513 selectively attenuates ethanol but not sucrose reinforced responding in a concurrent access procedure: Comparison to other drugs
-
Petry NM (1995) Ro 15-4513 selectively attenuates ethanol but not sucrose reinforced responding in a concurrent access procedure: comparison to other drugs. Psychopharmacology 121:192-203.
-
(1995)
Psychopharmacology
, vol.121
, pp. 192-203
-
-
Petry, N.M.1
-
31
-
-
19344363149
-
GABRA2 alleles moderate the subjective effects of alcohol, which are attenuated by finasteride
-
Pierucci-Lagha A, Covault J, Feinn R, Nellissery M, Hernandez-Avila C, Oncken C, Morrow AL, Kranzler HR (2005) GABRA2 alleles moderate the subjective effects of alcohol, which are attenuated by finasteride. Neuropsy-chopharmacology 30:1193-1203.
-
(2005)
Neuropsy-chopharmacology
, vol.30
, pp. 1193-1203
-
-
Pierucci-Lagha, A.1
Covault, J.2
Feinn, R.3
Nellissery, M.4
Hernandez-Avila, C.5
Oncken, C.6
Morrow, A.L.7
Kranzler, H.R.8
-
34
-
-
0032704330
-
Discriminative stimulus effects of zolpidem in squirrel monkeys: Comparison with conventional benzodiazepines and sedative-hypnotics
-
Rowlett JK, Spealman RD, Lelas S (1999) Discriminative stimulus effects of zolpidem in squirrel monkeys: comparison with conventional benzodiazepines and sedative-hypnotics. J Pharmacol Exp Ther 291: 1233-1241.
-
(1999)
J Pharmacol Exp Ther
, vol.291
, pp. 1233-1241
-
-
Rowlett, J.K.1
Spealman, R.D.2
Lelas, S.3
-
37
-
-
0034733040
-
A and α-amino-3-hydroxy-5-methylsoxazole-4-propionate receptors are differentially affected by aging in the rat hippocampus
-
A and α-amino-3-hydroxy-5-methylsoxazole-4-propionate receptors are differentially affected by aging in the rat hippocampus. J Biol Chem 275:19585-19593.
-
(2000)
J Biol Chem
, vol.275
, pp. 19585-19593
-
-
Ruano, D.1
Araujo, F.2
Revilla, E.3
Vela, J.4
Bergis, O.5
Vitorica, J.6
-
38
-
-
0030823552
-
The effects of new hypnotic drugs in rats trained to discriminate ethanol
-
Sanger DJ (1997) The effects of new hypnotic drugs in rats trained to discriminate ethanol. Behav Pharmacol 8:287-292.
-
(1997)
Behav Pharmacol
, vol.8
, pp. 287-292
-
-
Sanger, D.J.1
-
39
-
-
0037072577
-
A receptor subtypes
-
A receptor subtypes. Eur J Pharmacol 451:103-110.
-
(2002)
Eur J Pharmacol
, vol.451
, pp. 103-110
-
-
Sanna, E.1
Busonero, F.2
Talani, G.3
Carta, M.4
Massa, F.5
Peis, M.6
Maciocco, E.7
Biggio, G.8
-
40
-
-
2942648336
-
Discriminative stimulus effects of ethanol in mice lacking the c-aminobutyric acid type A receptor δ subunit
-
Shannon EE, Shelton KL, Vivian JA, Yount I, Morgan AR, Homanics GE, Grant KA (2004) Discriminative stimulus effects of ethanol in mice lacking the c-aminobutyric acid type A receptor δ subunit. Alcohol Clin Exp Res 28:906-913.
-
(2004)
Alcohol Clin Exp Res
, vol.28
, pp. 906-913
-
-
Shannon, E.E.1
Shelton, K.L.2
Vivian, J.A.3
Yount, I.4
Morgan, A.R.5
Homanics, G.E.6
Grant, K.A.7
-
41
-
-
0035192581
-
Effects of naltrexone and Ro 15-4513 on a multiple schedule of ethanol and tang self-administration
-
Shelton KL, Grant KA (2001) Effects of naltrexone and Ro 15-4513 on a multiple schedule of ethanol and tang self-administration. Alcohol Clin Exp Res 25:1576-1585.
-
(2001)
Alcohol Clin Exp Res
, vol.25
, pp. 1576-1585
-
-
Shelton, K.L.1
Grant, K.A.2
-
42
-
-
0028981088
-
A receptor subtypes
-
A receptor subtypes. Pharmacol Rev 47:181-234.
-
(1995)
Pharmacol Rev
, vol.47
, pp. 181-234
-
-
Sieghart, W.1
-
43
-
-
0035039871
-
36Cl ion flux
-
36Cl ion flux. Mol Pharmacol 59:1108-1118.
-
(2001)
Mol Pharmacol
, vol.59
, pp. 1108-1118
-
-
Smith, A.J.1
Alder, L.2
Silk, J.3
Adkins, C.4
Fletcher, A.E.5
Scales, T.6
Kerby, J.7
Marshall, G.8
Wafford, K.A.9
McKernan, R.M.10
Atack, J.R.11
-
44
-
-
33947433399
-
Using drug-discrimination techniques to study the abuse-related effects of psycho-active drugs in rats
-
Solinas M, Panlilio LV, Justinova Z, Yasar S, Goldberg S (2006) Using drug-discrimination techniques to study the abuse-related effects of psycho-active drugs in rats. Nat Protoc 1:1194-1206.
-
(2006)
Nat Protoc
, vol.1
, pp. 1194-1206
-
-
Solinas, M.1
Panlilio, L.V.2
Justinova, Z.3
Yasar, S.4
Goldberg, S.5
-
45
-
-
0023042881
-
A selective imidazobenzodiazepine antagonist of ethanol in the rat
-
Suzdak PD, Glowa JR, Crawley JN, Schwartz RD, Skolnick P, Paul SM (1986) A selective imidazobenzodiazepine antagonist of ethanol in the rat. Science 234:1243-1247.
-
(1986)
Science
, vol.234
, pp. 1243-1247
-
-
Suzdak, P.D.1
Glowa, J.R.2
Crawley, J.N.3
Schwartz, R.D.4
Skolnick, P.5
Paul, S.M.6
-
46
-
-
0018655874
-
2 and receptor differentiation: A statistical analysis of competitive antagonism
-
2 and receptor differentiation: a statistical analysis of competitive antagonism. Life Sci 25:637-654.
-
(1979)
Life Sci
, vol.25
, pp. 637-654
-
-
Tallarida, F.J.1
Cowan, A.2
Adler, M.W.3
-
47
-
-
0036020326
-
Characterization of the discriminative stimulus effects of N-methyl-D- aspartate ligands under different ethanol training conditions in the cynomolgus monkey (Macaca fascicularis)
-
Vivian JA, Waters CA, Szeliga KT, Jordan K, Grant KA (2002) Characterization of the discriminative stimulus effects of N-methyl-D- aspartate ligands under different ethanol training conditions in the cynomolgus monkey (Macaca fascicularis). Psychopharmacology 162:273-281.
-
(2002)
Psychopharmacology
, vol.162
, pp. 273-281
-
-
Vivian, J.A.1
Waters, C.A.2
Szeliga, K.T.3
Jordan, K.4
Grant, K.A.5
-
48
-
-
0026722810
-
Influences of gender, gonadectomy, and estrous cycle on GABA/BZ receptors and benzodiazepine responses in rats
-
Wilson MA (1992) Influences of gender, gonadectomy, and estrous cycle on GABA/BZ receptors and benzodiazepine responses in rats. Brain Res Bull 29:165-172.
-
(1992)
Brain Res Bull
, vol.29
, pp. 165-172
-
-
Wilson, M.A.1
|