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Volumn 31, Issue 10, 2007, Pages 78-88

Strategy for the prediction and selection of drug substance salt forms

Author keywords

[No Author keywords available]

Indexed keywords

ACIDS; IONIZATION;

EID: 53649083004     PISSN: 15432521     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review
Times cited : (3)

References (16)
  • 2
    • 0001056344 scopus 로고    scopus 로고
    • Preparation of Water-Soluble Compounds Through Salt Formation
    • C.G. Wermuth, Ed, Academic Press, New York, NY
    • B.D. Anderson and K.P. Flora, "Preparation of Water-Soluble Compounds Through Salt Formation," in The Practice of Medicinal Chemistry, C.G. Wermuth, Ed. (Academic Press, New York, NY, 1996), pp. 739-754.
    • (1996) The Practice of Medicinal Chemistry , pp. 739-754
    • Anderson, B.D.1    Flora, K.P.2
  • 4
    • 53649084710 scopus 로고    scopus 로고
    • L.D. Bighley, S.M. Berge, and D.C. Monkhouse, Salt Forms of Drugs and Absorption, in Encyclopedia of Pharmaceutical Technology, J. Swarbrick and J.C. Boylan JC, Eds. (Marcel Dekker, New York, NY, 1995), pp. 453-499.
    • L.D. Bighley, S.M. Berge, and D.C. Monkhouse, "Salt Forms of Drugs and Absorption," in Encyclopedia of Pharmaceutical Technology, J. Swarbrick and J.C. Boylan JC, Eds. (Marcel Dekker, New York, NY, 1995), pp. 453-499.
  • 5
    • 1642457350 scopus 로고    scopus 로고
    • An Automated Approach to Salt Selection for New Unique Trazodone Salts
    • E.C. Ware and D.R. Lu, "An Automated Approach to Salt Selection for New Unique Trazodone Salts," Pharm. Res. 21 (1), 177-184 (2004).
    • (2004) Pharm. Res , vol.21 , Issue.1 , pp. 177-184
    • Ware, E.C.1    Lu, D.R.2
  • 6
    • 27944487022 scopus 로고    scopus 로고
    • Occurrence of Pharmaceutically Acceptable Anions and Cations in the Cambridge Structural Database
    • D.A. Haynes, W. Jones, and W.D.S. Motherwell, "Occurrence of Pharmaceutically Acceptable Anions and Cations in the Cambridge Structural Database," J. Pharm. Sci. 94 (10), 2111-2120 (2005).
    • (2005) J. Pharm. Sci , vol.94 , Issue.10 , pp. 2111-2120
    • Haynes, D.A.1    Jones, W.2    Motherwell, W.D.S.3
  • 7
    • 0023032232 scopus 로고
    • Salt Selection for Basic Drugs
    • P.L. Gould, "Salt Selection for Basic Drugs," Int. J. Pharm. 33 (1-2), 201-217 (1986).
    • (1986) Int. J. Pharm , vol.33 , Issue.1-2 , pp. 201-217
    • Gould, P.L.1
  • 8
    • 0028219710 scopus 로고
    • An Integrated Approach to the Selection of Optimal Salt Form for a New Drug Candidate
    • K.R. Morris et al., "An Integrated Approach to the Selection of Optimal Salt Form for a New Drug Candidate," Int. J. Pharm. 105 (2), 209-217 (1994).
    • (1994) Int. J. Pharm , vol.105 , Issue.2 , pp. 209-217
    • Morris, K.R.1
  • 9
    • 0031806352 scopus 로고    scopus 로고
    • In Situ Salt Screening - A Useful Technique for Discovery Support and Preformulation Studies
    • W-Q. Tong and G. Whitesell, "In Situ Salt Screening - A Useful Technique for Discovery Support and Preformulation Studies," Pharm. Dev. Tech. 3 (2), 215-223 (1998).
    • (1998) Pharm. Dev. Tech , vol.3 , Issue.2 , pp. 215-223
    • Tong, W.-Q.1    Whitesell, G.2
  • 10
    • 0033671441 scopus 로고    scopus 로고
    • General Equations for In Situ Salt Screening of Multibasic Drugs in Multiprotic Acids
    • M. Sacchetti, "General Equations for In Situ Salt Screening of Multibasic Drugs in Multiprotic Acids," Pharm. Dev. Tech. 5 (4), 579-582 (2000).
    • (2000) Pharm. Dev. Tech , vol.5 , Issue.4 , pp. 579-582
    • Sacchetti, M.1
  • 11
    • 0034345216 scopus 로고    scopus 로고
    • Salt Selection and Optimization Procedures for Pharmaceutical New Chemical Entities
    • R.J.Bastin, M.J. Bowker, and B.J. Slater, "Salt Selection and Optimization Procedures for Pharmaceutical New Chemical Entities," Org. Proc. Res. Dev. 4 (5), 427-435 (2000).
    • (2000) Org. Proc. Res. Dev , vol.4 , Issue.5 , pp. 427-435
    • Bastin, R.J.1    Bowker, M.J.2    Slater, B.J.3
  • 12
    • 1042284960 scopus 로고    scopus 로고
    • Salt-Selection Strategies
    • P.H. Stahl and C.G. Wermuth, Eds, Wiley-VCH, Weinheim, Germany
    • A.T.M. Serajuddin and M. Pudipeddi, "Salt-Selection Strategies," in Handbook of Pharmaceutical Salts, P.H. Stahl and C.G. Wermuth, Eds. (Wiley-VCH, Weinheim, Germany, 2002), pp. 135-160.
    • (2002) Handbook of Pharmaceutical Salts , pp. 135-160
    • Serajuddin, A.T.M.1    Pudipeddi, M.2
  • 13
    • 1042284962 scopus 로고    scopus 로고
    • A Procedure for Salt Selection and Optimization
    • P.H. Stahl and C.G. Wermuth, Eds, Wiley-VCH, Weinheim, Germany
    • M.J. Bowker, "A Procedure for Salt Selection and Optimization," in Handbook of Pharmaceutical Salts, P.H. Stahl and C.G. Wermuth, Eds. (Wiley-VCH, Weinheim, Germany, 2002), pp. 161-189.
    • (2002) Handbook of Pharmaceutical Salts , pp. 161-189
    • Bowker, M.J.1
  • 14
    • 33750904749 scopus 로고    scopus 로고
    • R.B. Hammond et al., Grid-Based Molecular Modeling for Pharmaceutical Salt Screening: Case Example of 3,4,5,7,8,9-hexahydro-2H- pyrimido-(1,2-a)-primidinium acetate, J. Pharm. Sci. 95 (11), 2361-2372 (2006).
    • R.B. Hammond et al., "Grid-Based Molecular Modeling for Pharmaceutical Salt Screening: Case Example of 3,4,5,7,8,9-hexahydro-2H- pyrimido-(1,2-a)-primidinium acetate," J. Pharm. Sci. 95 (11), 2361-2372 (2006).
  • 15
    • 53649097470 scopus 로고    scopus 로고
    • Lange's Handbook of Chemistry, J.A. Dean, Ed. (McGraw-Hill, New York, NY, 12th edition, 1979), pp. 5-7.
    • Lange's Handbook of Chemistry, J.A. Dean, Ed. (McGraw-Hill, New York, NY, 12th edition, 1979), pp. 5-7.
  • 16
    • 0011223331 scopus 로고    scopus 로고
    • Ibuprofen
    • H.G. Brittain, Ed, Academic Press, San Diego, CA
    • J.D Higgins et al., "Ibuprofen," in Analytical Profiles of Drug Substances and Excipients, vol. 27, H.G. Brittain, Ed. (Academic Press, San Diego, CA, 2001), pp. 265-300.
    • (2001) Analytical Profiles of Drug Substances and Excipients , vol.27 , pp. 265-300
    • Higgins, J.D.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.