Novel aryloxy-8-azabicyclo[3.2.1]oct-3-enes with 5-HT transporter and 5-HT 1A affinity

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 21, 2004, Pages 5281-5284

  Gilbert, Adam M ^a   Coleman, Thomas ^a   Kodah, Jason ^a   Mewshaw, Richard E ^a   Scerni, Rosemary ^a   Schechter, Lee E ^a   Smith, Deborah L ^a   Andree, Terrance H ^a  

^a PFIZER INC   (United States)

Author keywords

Serotonin 1A receptor; Serotonin transporter

Indexed keywords

ALKANE; ALKENE DERIVATIVE; HETEROCYCLIC COMPOUND; SEROTONIN; SEROTONIN 1A ANTAGONIST; SEROTONIN 1A RECEPTOR;

ARTICLE; BINDING AFFINITY; RECEPTOR AFFINITY;

ANIMALS; BICYCLO COMPOUNDS, HETEROCYCLIC; CHO CELLS; CRICETINAE; CRICETULUS; HUMANS; MEMBRANE GLYCOPROTEINS; MEMBRANE TRANSPORT PROTEINS; NERVE TISSUE PROTEINS; RADIOLIGAND ASSAY; RECEPTOR, SEROTONIN, 5-HT1A; SEROTONIN PLASMA MEMBRANE TRANSPORT PROTEINS; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 5344267450     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.08.030     Document Type: Article

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