Synthesis of 2-alkynyl substituted 4′-thioadenosine derivatives and their binding affinities at the adenosine receptors

Archives of Pharmacal Research

Volumn 31, Issue 8, 2008, Pages 973-977

  Liang, Cheng Wu ^a,b   Choi, Won Jun ^a   Jeong, Lak Shin ^a  

^a Ewha Womans University   (South Korea)

^b JILIN MEDICAL COLLEGE   (China)

Author keywords

2 Alkynyl substituted N 6 methyl 4 thioadenosine; A 3 adenosine receptor; Binding affinity; Diazotization; Palladium catalyzed cross coupling

Indexed keywords

4'-THIOADENOSINE; ADENOSINE; ADENOSINE RECEPTOR; DRUG DERIVATIVE; DYES, REAGENTS, INDICATORS, MARKERS AND BUFFERS; NUCLEOSIDE; PALLADIUM; THIOADENOSINE;

ANIMAL; ARTICLE; CATALYSIS; CHO CELL; CRICETULUS; DRUG DESIGN; HAMSTER; HUMAN; METABOLISM; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; SYNTHESIS; ULTRAVIOLET SPECTROPHOTOMETRY;

ADENOSINE; ANIMALS; CATALYSIS; CHO CELLS; CRICETINAE; CRICETULUS; DRUG DESIGN; HUMANS; INDICATORS AND REAGENTS; MAGNETIC RESONANCE SPECTROSCOPY; PALLADIUM; RECEPTORS, PURINERGIC P1; SPECTROPHOTOMETRY, ULTRAVIOLET; THIONUCLEOSIDES;

EID: 51849143774     PISSN: 02536269     EISSN: 19763786     Source Type: Journal    
DOI: 10.1007/s12272-001-1254-x     Document Type: Article

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