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Volumn 361, Issue 1-2, 2008, Pages 141-149

Polymorphic control of inhalation microparticles prepared by crystallization

Author keywords

Aerosol; Antisolvent micronization; Differential scanning calorimetry; Inhalation; Polymorphism; Salmeterol xinafoate; Thermal kinetic analysis

Indexed keywords

2 PROPANOL; MACROGOL; MACROGOL 400; MACROGOL 6000; SALMETEROL XINAFOATE; SOLVENT;

EID: 47949124171     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2008.05.033     Document Type: Article
Times cited : (12)

References (45)
  • 1
    • 0342869049 scopus 로고
    • Kinetics of phase change I-general theory
    • Avrami M. Kinetics of phase change I-general theory. J. Chem. Phys. 7 (1939) 1103-1112
    • (1939) J. Chem. Phys. , vol.7 , pp. 1103-1112
    • Avrami, M.1
  • 2
    • 0001336124 scopus 로고
    • Kinetics of phase change. II. Transformation-time relations for random distribution of nuclei
    • Avrami M. Kinetics of phase change. II. Transformation-time relations for random distribution of nuclei. J. Chem. Phys. 8 (1940) 212-224
    • (1940) J. Chem. Phys. , vol.8 , pp. 212-224
    • Avrami, M.1
  • 3
    • 0346395110 scopus 로고
    • Granulation, phase change, and microstructure-kinetics of phase change III
    • Avrami M. Granulation, phase change, and microstructure-kinetics of phase change III. J. Chem. Phys. 9 (1941) 177-184
    • (1941) J. Chem. Phys. , vol.9 , pp. 177-184
    • Avrami, M.1
  • 6
    • 0344152356 scopus 로고    scopus 로고
    • Polymorph selection: challenges for the future?
    • Blagden N., and Davey R.J. Polymorph selection: challenges for the future?. Cryst. Growth Des. 3 (2003) 873-885
    • (2003) Cryst. Growth Des. , vol.3 , pp. 873-885
    • Blagden, N.1    Davey, R.J.2
  • 7
    • 0035998944 scopus 로고    scopus 로고
    • Effects of mechanical processing on phase composition
    • Brittain H.G. Effects of mechanical processing on phase composition. J. Pharm. Sci. 91 (2002) 1573-1580
    • (2002) J. Pharm. Sci. , vol.91 , pp. 1573-1580
    • Brittain, H.G.1
  • 8
    • 0018625999 scopus 로고
    • Polymorphism of pharmaceuticals and other molecular-crystals. 1. Theory of thermodynamic rules
    • Burger A., and Ramberger R. Polymorphism of pharmaceuticals and other molecular-crystals. 1. Theory of thermodynamic rules. Mikrochim. Acta 2 (1979) 259-271
    • (1979) Mikrochim. Acta , vol.2 , pp. 259-271
    • Burger, A.1    Ramberger, R.2
  • 9
    • 21344459447 scopus 로고    scopus 로고
    • Studies on the crystallinity of a pharmaceutical development drug substance
    • Byard S.J., Jackson S.L., Smail A., Bauer M., and Apperley D.C. Studies on the crystallinity of a pharmaceutical development drug substance. J. Pharm. Sci. 94 (2005) 1321-1335
    • (2005) J. Pharm. Sci. , vol.94 , pp. 1321-1335
    • Byard, S.J.1    Jackson, S.L.2    Smail, A.3    Bauer, M.4    Apperley, D.C.5
  • 10
    • 28444458504 scopus 로고    scopus 로고
    • The effect of crystal morphology and mill type on milling induced crystal disorder
    • Chikhalia V., Forbes R.T., Storey R.A., and Ticehurst M. The effect of crystal morphology and mill type on milling induced crystal disorder. Eur. J. Pharm. Sci. 27 (2006) 19-26
    • (2006) Eur. J. Pharm. Sci. , vol.27 , pp. 19-26
    • Chikhalia, V.1    Forbes, R.T.2    Storey, R.A.3    Ticehurst, M.4
  • 11
    • 20344399736 scopus 로고    scopus 로고
    • Pharmacological agents used to treat asthma
    • Chung K.F., and O'Byrne P.M. Pharmacological agents used to treat asthma. Eur. Respir. Monogr. (2003) 339-375
    • (2003) Eur. Respir. Monogr. , pp. 339-375
    • Chung, K.F.1    O'Byrne, P.M.2
  • 12
    • 33744681580 scopus 로고
    • Phase changes and chemical reactions in molecular crystals
    • Dunitz J. Phase changes and chemical reactions in molecular crystals. Acta Crystallogr. B 51 (1995) 619-631
    • (1995) Acta Crystallogr. B , vol.51 , pp. 619-631
    • Dunitz, J.1
  • 13
    • 0028018201 scopus 로고
    • Increased metastable solubility of milled griseofulvin, depending on the formation of a disordered surface structure
    • Elamin A.A., Ahlneck C., Alderborn G., and Nystrom C. Increased metastable solubility of milled griseofulvin, depending on the formation of a disordered surface structure. Int. J. Pharm. 111 (1994) 159-170
    • (1994) Int. J. Pharm. , vol.111 , pp. 159-170
    • Elamin, A.A.1    Ahlneck, C.2    Alderborn, G.3    Nystrom, C.4
  • 14
    • 0000768201 scopus 로고    scopus 로고
    • Direct methods and powder data: state of the art and perspectives
    • Giacovazzo C. Direct methods and powder data: state of the art and perspectives. Acta Crystallogr. A 52 (1996) 331-339
    • (1996) Acta Crystallogr. A , vol.52 , pp. 331-339
    • Giacovazzo, C.1
  • 15
    • 33746868980 scopus 로고    scopus 로고
    • The effects of milling on the surface properties of form I paracetamol crystals
    • Heng J.Y.Y., Thielmann F., and Williams D.R. The effects of milling on the surface properties of form I paracetamol crystals. Pharm. Res. 23 (2006) 1918-1927
    • (2006) Pharm. Res. , vol.23 , pp. 1918-1927
    • Heng, J.Y.Y.1    Thielmann, F.2    Williams, D.R.3
  • 18
    • 0037074121 scopus 로고    scopus 로고
    • The impact of low levels of amorphous material (<5%) on the blending characteristics of a direct compression formulation
    • Mackin L., Sartnurak S., Thomas I., and Moore S. The impact of low levels of amorphous material (<5%) on the blending characteristics of a direct compression formulation. Int. J. Pharm. 231 (2002) 213-226
    • (2002) Int. J. Pharm. , vol.231 , pp. 213-226
    • Mackin, L.1    Sartnurak, S.2    Thomas, I.3    Moore, S.4
  • 19
    • 0037074074 scopus 로고    scopus 로고
    • Quantification of low levels (<10%) of amorphous content in micronised active batches using dynamic vapour sorption and isothermal microcalorimetry
    • Mackin L., Zanon R., Park J.M., Foster K., Opalenik H., and Demonte M. Quantification of low levels (<10%) of amorphous content in micronised active batches using dynamic vapour sorption and isothermal microcalorimetry. Int. J. Pharm. 231 (2002) 227-236
    • (2002) Int. J. Pharm. , vol.231 , pp. 227-236
    • Mackin, L.1    Zanon, R.2    Park, J.M.3    Foster, K.4    Opalenik, H.5    Demonte, M.6
  • 20
    • 0003088993 scopus 로고    scopus 로고
    • On the determination of nucleation and growth kinetics by calorimetry
    • Michaelsen C., and Dahms M. On the determination of nucleation and growth kinetics by calorimetry. Thermochim. Acta 288 (1996) 9-27
    • (1996) Thermochim. Acta , vol.288 , pp. 9-27
    • Michaelsen, C.1    Dahms, M.2
  • 21
    • 0035897679 scopus 로고    scopus 로고
    • Theoretical approaches to physical transformations of active pharmaceutical ingredients during manufacturing processes
    • Morris K.R., Griesser U.J., Eckhardt C.J., and Stowell J.G. Theoretical approaches to physical transformations of active pharmaceutical ingredients during manufacturing processes. Adv. Drug Del. Rev. 48 (2001) 91-114
    • (2001) Adv. Drug Del. Rev. , vol.48 , pp. 91-114
    • Morris, K.R.1    Griesser, U.J.2    Eckhardt, C.J.3    Stowell, J.G.4
  • 22
    • 41549161049 scopus 로고    scopus 로고
    • Comparison of salmeterol xinafoate microparticle production by conventional and novel antisolvent crystallization
    • Murnane D., Marriott C., and Martin G.P. Comparison of salmeterol xinafoate microparticle production by conventional and novel antisolvent crystallization. Eur. J. Pharm. Biopharm. 69 (2008) 94-105
    • (2008) Eur. J. Pharm. Biopharm. , vol.69 , pp. 94-105
    • Murnane, D.1    Marriott, C.2    Martin, G.P.3
  • 23
    • 41549117146 scopus 로고    scopus 로고
    • Developing an environmentally benign process for the production of microparticles: amphiphilic crystallization
    • Murnane D., Martin G.P., and Marriott C. Developing an environmentally benign process for the production of microparticles: amphiphilic crystallization. Eur. J. Pharm. Biopharm. 69 (2008) 72-82
    • (2008) Eur. J. Pharm. Biopharm. , vol.69 , pp. 72-82
    • Murnane, D.1    Martin, G.P.2    Marriott, C.3
  • 24
    • 0037607606 scopus 로고    scopus 로고
    • Inverse gas chromatography: considerations about appropriate use for amorphous and crystalline powders
    • Planinsek O., and Buckton G. Inverse gas chromatography: considerations about appropriate use for amorphous and crystalline powders. J. Pharm. Sci. 92 (2003) 1286-1294
    • (2003) J. Pharm. Sci. , vol.92 , pp. 1286-1294
    • Planinsek, O.1    Buckton, G.2
  • 25
    • 0035117761 scopus 로고    scopus 로고
    • The influence of lung deposition on clinical response
    • Pritchard J.N. The influence of lung deposition on clinical response. J. Aerosol Med. 14 (2001) S19-S26
    • (2001) J. Aerosol Med. , vol.14
    • Pritchard, J.N.1
  • 27
    • 0344603644 scopus 로고    scopus 로고
    • Significance of controlling crystallization mechanisms and kinetics in pharmaceutical systems
    • Rodriguez-Hornedo N., and Murphy D. Significance of controlling crystallization mechanisms and kinetics in pharmaceutical systems. J. Pharm. Sci. 88 (1999) 651-660
    • (1999) J. Pharm. Sci. , vol.88 , pp. 651-660
    • Rodriguez-Hornedo, N.1    Murphy, D.2
  • 28
    • 0027642972 scopus 로고
    • Polymorphic transformations in crystal-growth
    • Sato K. Polymorphic transformations in crystal-growth. J. Phys. D: Appl. Phys. 26 (1993) B77-B84
    • (1993) J. Phys. D: Appl. Phys. , vol.26
    • Sato, K.1
  • 29
    • 33747177115 scopus 로고    scopus 로고
    • Analytical techniques for quantification of amorphous/crystalline phases in pharmaceutical solids
    • Shah B., Kakumanu V.K., and Bansal A.K. Analytical techniques for quantification of amorphous/crystalline phases in pharmaceutical solids. J. Pharm. Sci. 95 (2006) 1641-1665
    • (2006) J. Pharm. Sci. , vol.95 , pp. 1641-1665
    • Shah, B.1    Kakumanu, V.K.2    Bansal, A.K.3
  • 31
    • 0033903829 scopus 로고    scopus 로고
    • Crystallization processes in pharmaceutical technology and drug delivery design
    • Shekunov B.Y., and York P. Crystallization processes in pharmaceutical technology and drug delivery design. J. Cryst. Growth 211 (2000) 122-136
    • (2000) J. Cryst. Growth , vol.211 , pp. 122-136
    • Shekunov, B.Y.1    York, P.2
  • 32
    • 33747346761 scopus 로고    scopus 로고
    • On the misinterpretation of the correlation coefficient in pharmaceutical sciences
    • Sonnergaard J.M. On the misinterpretation of the correlation coefficient in pharmaceutical sciences. Int. J. Pharm. 321 (2006) 12-17
    • (2006) Int. J. Pharm. , vol.321 , pp. 12-17
    • Sonnergaard, J.M.1
  • 33
    • 0037838336 scopus 로고    scopus 로고
    • In vitro characterization of jet-milled and in-situ-micronized fluticasone-17-propionate
    • Steckel H., Rasenack N., Villax P., and Muller B.W. In vitro characterization of jet-milled and in-situ-micronized fluticasone-17-propionate. Int. J. Pharm. 258 (2003) 65-75
    • (2003) Int. J. Pharm. , vol.258 , pp. 65-75
    • Steckel, H.1    Rasenack, N.2    Villax, P.3    Muller, B.W.4
  • 34
    • 0013047721 scopus 로고    scopus 로고
    • A new molecular modeling approach to predict concomitant nucleation of polymorphs
    • ter Horst J.H., Kramer H.J.M., and Jansens P.J. A new molecular modeling approach to predict concomitant nucleation of polymorphs. Cryst. Growth Des. 2 (2002) 351-356
    • (2002) Cryst. Growth Des. , vol.2 , pp. 351-356
    • ter Horst, J.H.1    Kramer, H.J.M.2    Jansens, P.J.3
  • 35
    • 0034345199 scopus 로고    scopus 로고
    • Crystallisation of polymorphs: thermodynamic insight into the role of solvent
    • Threlfall T. Crystallisation of polymorphs: thermodynamic insight into the role of solvent. Org. Process Res. Dev. 4 (2000) 384-390
    • (2000) Org. Process Res. Dev. , vol.4 , pp. 384-390
    • Threlfall, T.1
  • 36
    • 0034858772 scopus 로고    scopus 로고
    • Characterization of two polymorphs of salmeterol xinafoate crystallized from supercritical fluids
    • Tong H.H., Shekunov B.Y., York P., and Chow A.H. Characterization of two polymorphs of salmeterol xinafoate crystallized from supercritical fluids. Pharm. Res. 18 (2001) 852-858
    • (2001) Pharm. Res. , vol.18 , pp. 852-858
    • Tong, H.H.1    Shekunov, B.Y.2    York, P.3    Chow, A.H.4
  • 37
    • 0036001398 scopus 로고    scopus 로고
    • Influence of polymorphism on the surface energetics of salmeterol xinafoate crystallized from supercritical fluids
    • Tong H.H.Y., Shekunov B.Y., York P., and Chow A.H.L. Influence of polymorphism on the surface energetics of salmeterol xinafoate crystallized from supercritical fluids. Pharm. Res. 19 (2002) 640-648
    • (2002) Pharm. Res. , vol.19 , pp. 640-648
    • Tong, H.H.Y.1    Shekunov, B.Y.2    York, P.3    Chow, A.H.L.4
  • 38
    • 0141567431 scopus 로고    scopus 로고
    • Thermal analysis of trace levels of polymorphic impurity in salmeterol xinafoate samples
    • Tong H.H.Y., Shekunov B.Y., York P., and Chow A.H.L. Thermal analysis of trace levels of polymorphic impurity in salmeterol xinafoate samples. Pharm. Res. 20 (2003) 1423-1429
    • (2003) Pharm. Res. , vol.20 , pp. 1423-1429
    • Tong, H.H.Y.1    Shekunov, B.Y.2    York, P.3    Chow, A.H.L.4
  • 39
    • 33645221184 scopus 로고    scopus 로고
    • Predicting the aerosol performance of dry powder inhalation formulations by interparticulate interaction analysis using inverse gas chromatography
    • Tong H.H.Y., Shekunov B.Y., York P., and Chow A.H.L. Predicting the aerosol performance of dry powder inhalation formulations by interparticulate interaction analysis using inverse gas chromatography. J. Pharm. Sci. 95 (2006) 228-233
    • (2006) J. Pharm. Sci. , vol.95 , pp. 228-233
    • Tong, H.H.Y.1    Shekunov, B.Y.2    York, P.3    Chow, A.H.L.4
  • 42
    • 0029058533 scopus 로고
    • Process-induced crystallinity changes in albuterol sulfate and its effect on powder physical stability
    • Ward G.H., and Schultz R.K. Process-induced crystallinity changes in albuterol sulfate and its effect on powder physical stability. Pharm. Res. 12 (1995) 773-779
    • (1995) Pharm. Res. , vol.12 , pp. 773-779
    • Ward, G.H.1    Schultz, R.K.2
  • 43
    • 0031733664 scopus 로고    scopus 로고
    • Characterisation of the surface energetics of milled dl-propranolol hydrochloride using inverse gas chromatography and molecular modelling
    • York P., Ticehurst M.D., Osborn J.C., Roberts R.J., and Rowe R.C. Characterisation of the surface energetics of milled dl-propranolol hydrochloride using inverse gas chromatography and molecular modelling. Int. J. Pharm. 174 (1998) 179-186
    • (1998) Int. J. Pharm. , vol.174 , pp. 179-186
    • York, P.1    Ticehurst, M.D.2    Osborn, J.C.3    Roberts, R.J.4    Rowe, R.C.5
  • 44
    • 1042298067 scopus 로고    scopus 로고
    • Phase transformation considerations during process development and manufacture of solid oral dosage forms
    • Zhang G.G.Z., Law D., Schmitt E.A., and Qiu Y. Phase transformation considerations during process development and manufacture of solid oral dosage forms. Adv. Drug Del. Rev. 56 (2004) 371-390
    • (2004) Adv. Drug Del. Rev. , vol.56 , pp. 371-390
    • Zhang, G.G.Z.1    Law, D.2    Schmitt, E.A.3    Qiu, Y.4
  • 45
    • 0037897314 scopus 로고    scopus 로고
    • Crystallization kinetics of amorphous nifedipine studied by model-fitting and model-free approaches
    • Zhou D.L., Schmitt E.A., Zhang G.G., Law D., Vyazovkin S., Wight C.A., and Grant D.J.W. Crystallization kinetics of amorphous nifedipine studied by model-fitting and model-free approaches. J. Pharm. Sci. 92 (2003) 1779-1792
    • (2003) J. Pharm. Sci. , vol.92 , pp. 1779-1792
    • Zhou, D.L.1    Schmitt, E.A.2    Zhang, G.G.3    Law, D.4    Vyazovkin, S.5    Wight, C.A.6    Grant, D.J.W.7


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