Evaluation of dynamic image analysis for characterizing pharmaceutical excipient particles

International Journal of Pharmaceutics

Volumn 361, Issue 1-2, 2008, Pages 150-157

  Yu, Weili ^a   Hancock, Bruno C ^a  

^a PFIZER INC   (United States)

Author keywords

Dynamic image analysis; Laser diffraction; Microcrystalline cellulose; Particle shape; Particle size; QicPic

Indexed keywords

CELPHERE; CEOLUS; EXCIPIENT; MICROCRYSTALLINE CELLULOSE;

ANALYTIC METHOD; ARTICLE; DEVICE; EVALUATION; IMAGE ANALYSIS; INSTRUMENT; INTERMETHOD COMPARISON; PARTICLE SIZE; POROSITY; PRIORITY JOURNAL; QUANTITATIVE ANALYSIS; SCANNING ELECTRON MICROSCOPY; VALIDATION PROCESS;

CELLULOSE; CHEMISTRY, PHARMACEUTICAL; EXCIPIENTS; LASERS; MICROSCOPY, ELECTRON, SCANNING; PARTICLE SIZE; POROSITY; TECHNOLOGY, PHARMACEUTICAL;

EID: 47949085541     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2008.05.025     Document Type: Article

References (31)

1. Bao N., Shen L., Feng X., Lu X., and Yanagisawa K. Shape and size characterization of potassium titanate fibers by image analysis. J. Mater. Sci. 39 (2004) 469-476
2. Deriemaeker L., and Finsy R. Shape and size determination by laser diffraction: average aspect ratio and size distribution by volume; feasibility of data analysis by neural network. Part. Part. Syst. Charact. 22 (2005) 5-13
3. Fee J.P.H., Collier P.S., Launchbury A.P., and Clarke R.S.J. The influence of particle size on the bioavailability of inhaled temazepam. Br. J. Clin. Pharm. 33 (1992) 641-644
4. Hentschel M.L., and Page N.W. Selection of descriptors for particle shape characterization. Part. Part. Sys. Charact. 20 (2003) 25-38
5. Hintz R.J., and Johnson K.C. The effect of particle size distribution on dissolution rate and oral absorption. Int. J. Pharm. 51 (1989) 9-17
6. Jillavenkatesa A., Dapkunas S.J., and Lum L.-S.H. Particle Size Characterization (2001), U.S. Government Printing Office, Washington
7. Johnson K.C., and Swindell A.C. Guidance in the setting of drug particle size specifications to minimize variability in absorption. Pharm. Res. 13 (1996) 1795-1798
8. Kelly R.N., and Kazanjian J. Commercial reference shape standards use in the study of particle shape effect on laser diffraction particle size analysis. AAPS Pharm. Sci. Tech. 7 (2006) Article 49, 7, E1-E12
9. Köhler U., List J., and Witt W. Comparison of Laser Diffraction and Image Analysis under Identical Dispersing Conditions (2007), Partec, Nürnberg
10. Kwan A.K.H., Mora C.F., and Chan H.C. Particle shape analysis of coarse aggregates using digital image process. Cement Concrete Res. 29 (1999) 1403-1410
11. Langston P.A., and Jones T.F. Non-spherical 2-dimensional particle size analysis from chord measurements using Bayes' theorem. Part. Part. Syst. Charact. 18 (2001) 12-21
12. Li M., Wilkinson D., and Patchigolla K. Comparison of particle size distributions measured using different techniques. Particul. Sci. Technol. 23 (2005) 265-284
13. Ma Z., Merkus H.G., and Scarlett B. Extending laser diffraction for particle shape characterization: technical aspects and application. Powder Technol. 118 (2001) 180-187
14. Massol-Chaudeur S., Berthiaux H., and Dodds J.A. Experimental study of the mixing kinetics of binary pharmaceutical powder mixtures in a laboratory hoop mixer. Chem. Eng. Sci. 57 (2002) 4053-4065
15. Masuda H., and Iinoya K. Theoretical study of the scatter of experimental data due to particle-size-distribution. J. Chem. Eng. Jpn. 4 (1971) 60-66
16. Meloy T.P., and Mani B.P. Particle shape analysis and separation techniques: a critical review. J. Powder Bulk Solids Technol. 10 (1986) 15-20
17. Mullarney M.P., Hancock B.C., Carlson G.T., Ladipo D.D., and Langdon B.A. The powder flow and compact mechanical properties of sucrose and three high-intensity sweeteners used in chewable tablets. Int. J. Pharm. 257 (2003) 227-236
18. Podczeck F. A shape factor to assess the shape of particles using image analysis. Powder Technol. 93 (1997) 47-53
19. Podczeck F., and Sharma M. The influence of particle size and shape of components of binary powder mixtures on the maximum volume reduction due to packing. Int. J. Pharm. 137 (1996) 41-47
20. Rabinski G., and Thomas D. Dynamic digital image analysis: emerging technology for particle characterization. Water Sci. Technol. 50 (2004) 19-26
21. Shah K.R., Badawy S.I.F., Szemraj M.M., Gray D.B., and Hussain M.A. Assessment of segregation potential of powder blends. Pharm. Dev. Technol. 12 (2007) 457-462
22. Sommer K. 40 years of presentation particle size distribution-yet still incorrect?. Part. Part. Syst. Charact. 18 (2001) 22-25
23. Swaminathan V., and Kildsig D.O. Polydisperse powder mixtures: effect of particle size and shape on mixture stability. Drug Dev. Ind. Pharm. 28 (2002) 41-48
24. Wang W. Image analysis of particles by modified Ferret method-best-fit rectangle. Powder Technol. 165 (2006) 1-10
25. Witt W., Köhler U., and List J. Direct Imaging of Very Fast Particles Opens the Application of the Powerful (Dry) Dispersion for Size and Shape Characterization (2004), Partec, Nürnberg
26. Witt, W., Köhler, U., List, J., 2005. Experiences with dry dispersion and high-speed image analysis for size and shape characterization. Particulate Systems Analysis, Stratford-upon-Avon, UK.
27. Xu R. Particle Characterization: Light Scattering Methods (2000), Kluwer Academic Publishers, Norwell
28. Xu R., Andreina O., and Guida D. Comparison of sizing small particles using different technologies. Powder Technol. 132 (2003) 145-153
29. Yin S.X., Franchini M., Chen J., Hsieh A., Jen S., Lee T., Hussain M., and Smith R. Bioavailability enhancement of a COX-2 inhibitor, BMS-347070, from a nanocrystalline dispersion prepared by spray-drying. J. Pharm. Sci. 94 (2005) 1598-1607
30. Yu W., and Erickson K. Chord length characterization using focused beam reflectance measurement probe-methodologies and pitfalls. Powder Technol. 185 (2007) 24-30
31. Zhang Y., and Johnson K.C. Effect of drug particle size on content uniformity of low-dose solid dosage forms. Int. J. Pharm. 154 (1997) 179-183