P-glycoprotein inhibition by membrane cholesterol modulation

European Journal of Pharmaceutical Sciences

Volumn 34, Issue 4-5, 2008, Pages 236-242

  Fenyvesi, Ferenc ^a   Fenyvesi, Éva ^b   Szente, Lajos ^b   Goda, Katalin ^a   Bacsó, Zsolt ^a   Bácskay, Ildikó ^a   Váradi, Judit ^a   Kiss, Tímea ^a   Molnár, Éva ^c   Janáky, Tamás ^d   Szabó Jr , Gábor ^a   Vecsernyés, Miklós ^a  

^a UNIVERSITY OF DEBRECEN   (Hungary)

^b CycloLab Cyclodextrin Research & Development Laboratory Ltd   (Hungary)

^c SOLVO BIOTECHNOLOGY   (Hungary)

^d UNIVERSITY OF SZEGED   (Hungary)

Author keywords

ATP; Cell viability; Cholesterol; Heptakis(2,6 di O methyl) cyclodextrin; P glycoprotein

Indexed keywords

ADENOSINE TRIPHOSPHATE; BETA CYCLODEXTRIN DERIVATIVE; CALCEIN; CHOLESTEROL; CYCLODEXTRIN; GLYCOPROTEIN P; HEPTAKIS(2,6 DI O METHYL)BETA CYCLODEXTRIN; MEMBRANE PROTEIN; MEROCYANINE;

ANIMAL CELL; ARTICLE; CELL MEMBRANE PERMEABILITY; CELL VIABILITY; COMPLEX FORMATION; CONTROLLED STUDY; CYTOTOXICITY; INTERNALIZATION; LIPID RAFT; LIPOPHILICITY; MEMBRANE STRUCTURE; MICROENVIRONMENT; MOUSE; MULTIDRUG RESISTANCE; NONHUMAN; PRIORITY JOURNAL; PROTEIN LOCALIZATION; STAINING;

ADENOSINE TRIPHOSPHATE; ANIMALS; CELL MEMBRANE PERMEABILITY; CELL SURVIVAL; CHOLESTEROL; CYCLODEXTRINS; DOSE-RESPONSE RELATIONSHIP, DRUG; ENDOCYTOSIS; FLUORESCEINS; MEMBRANE MICRODOMAINS; MICE; NIH 3T3 CELLS; P-GLYCOPROTEIN; TRANSFECTION;

EID: 47249099723     PISSN: 09280987     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejps.2008.04.005     Document Type: Article

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