The prediction of the dissolution rate constant by mixing rules: The study of acetaminophen batches

Drug Development and Industrial Pharmacy

Volumn 34, Issue 5, 2008, Pages 522-535

  Lee, Tu ^a   Hou, Hung Ju ^a   Hsieh, Hsiang Yu ^a   Su, Yan Chan ^a   Wang, Yeh Wen ^a   Hsu, Fu Bin ^a  

^a NATIONAL CENTRAL UNIVERSITY   (Taiwan)

Author keywords

Acetaminophen; Dissolution rate constant; Mixing rules

Indexed keywords

PARACETAMOL;

ARTICLE; BATCH PROCESS; DRUG FORMULATION; DRUG GRANULATION; DRUG GRANULE; DRUG MANUFACTURE; DRUG SOLUBILITY; PARTICLE SIZE; PREDICTION;

ACETAMINOPHEN; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; CALORIMETRY, DIFFERENTIAL SCANNING; CHEMISTRY, PHARMACEUTICAL; MICROSCOPY, ELECTRON, SCANNING; PARTICLE SIZE; POWDERS; SOLUBILITY; SPECTROPHOTOMETRY, ULTRAVIOLET;

EID: 45849133068     PISSN: 03639045     EISSN: 15205762     Source Type: Journal    
DOI: 10.1080/03639040701744194     Document Type: Article

References (21)

1. Braga, D., & Grepioni, F. (2005). Making crystals from crystals: A green route to crystal engineering and polymorphism. Chem. Commun., 29, 3635-3645.
2. Bryn, S., Morris, K., & Comella, S. (2005). Reducing time to market with a science-based product management strategy. Pharm. Tech., 46-56.
3. Cao, Q. R., Choi, Y. W., Cui, J. H., & Lee, B. J. (2005). Formulation, release, characteristics and bioavailability of novel monolithic hydroxypropylmethylcellulose matrix tablets containing acetaminophen. J. Control. Release, 108, 351-361.
4. Ebube, N. K., Hikal, A. H., Wyandt, C. M., Beer, D. C., Miller, L. G., & Jones, A. B. (1997). Effect of drug, formulation and process variables on granulation and compaction characteristics of heterogeneous matrices. Part 1: HMPC and HPC systems. Int. J. Pharm., 156, 49-57.
5. Habib, M. J., Venkataram, S., & Delwar Hussain, M. (2001). Fundamentals of solid dispersions. In M. J. Habib (Ed.), Pharmaceutical solid dispersion technology (pp. 7-35). Lancaster, PA: Technomic.
6. Hashin, Z., & Shtrikman, S. (1963). Conductivity of polycrystals. Phys. Rev., 130, 129-133.
7. Jørgensen, K., & Christensen, F. N. (1996). Shape modelling of dissolution profiles by non-integer kinetic orders. Int. J. Pharm., 143, 223-232.
8. Keleb, E. I., Vermeire, A., Vervaet, C., & Remon, J. P. (2004). Extrusion granulation and high shear granulation of different grades of lactose and high dosed drugs: A comparative study. Drug Dev. Ind. Pharm., 30, 679-691.
9. Lee, T., & Hsu, F. B. (2007). A cross-performance relationship between Carr's index and dissolution rate constant: The study of acetaminophen batches. Drug Dev. Ind. Pharm., 33, 1273-1284.
10. Lee, T., Hung, S. T., & Kuo, C. S. (2006). Polymorph farming of acetaminophen and sulfathiazole on a chip. Pharm. Res., 23, 2542-2555.
11. Lee, T., Kuo, C. S., & Chen, Y. H. (2006). Solubility, polymorphism, crystallinity, and crystal habit of acetaminophen and ibuprofen by initial solvent screening. Pharm. Tech., 30, 72-92.
12. Lee, T., & Lee, J. (2003). Particle attrition by particle-surface friction in dryers. Pharm. Tech., 27, 64-72.
13. Looyenga, H. (1965). Dielectric constants of heterogeneous mixtures. Physica, 31, 401-406.
14. Maxwell, J. C. (1904). A treatise on electricity and magnetism (Vol. 1, p. 440). Oxford, UK: Clarendon Press.
15. Railkar, A. M., & Schwartz, J. B. (2001). Use of a moist granulation technique (MGT) to develop controlled-release dosage forms of acetaminophen. Drug Dev. Ind. Pharm., 27, 337-343.
16. Randall, C. A., Miyazaki, S., More, K. L., Bhalla, A. S., & Newnham, R. E. (1992). Structural property relationships in dielectrophoretically assembled BaTiO3 nanocomposites. Mater. Lett., 15, 26-30.
17. Simpson, G. (1974). The dielectric constants of a ferroelectric ceramic. Ferroelectrics, 6, 283-288.
18. Sorasuchart, W., Wardrop, J., & Ayres, J. W. (1999). Drug release from spray layered and coated drug-containing beads: Effects of pH and comparison of different dissolution methods. Drug Dev. Ind. Pharm., 25, 1093-1098.
19. Torquato, S. (1991). Random heterogeneous media: Microstructure and improved bounds on effective properties. Appl. Mech. Rev., 44, 37-73.
20. Van den Dries, K., & Vromans, H. (2003). Experimental and modelistic approach to explain granulate inhomogeneity through preferential growth. Eur. J. Pharm. Sci., 20, 409-417.
21. Wade, A., & Weller, P. J. (1994) Handbook of pharmaceutical excipients (2nd ed., pp. 392-399). Washington, DC: American Pharmaceutical Association.