메뉴 건너뛰기




Volumn 9, Issue 1, 2008, Pages 154-162

Lipospheres as carriers for topical delivery of aceclofenac: Preparation, characterization and In vivo evaluation

Author keywords

Aceclofenac; Animal experiment; Entrapment; Formulation; Lipospheres; Stability; Sustained release

Indexed keywords

ACECLOFENAC; BRISTAFLAM; DRUG CARRIER; LIPID; LIPOSPHERE; PHOSPHOLIPID; UNCLASSIFIED DRUG; DICLOFENAC; DRUG DERIVATIVE; LIPOSOME; NONSTEROID ANTIINFLAMMATORY AGENT;

EID: 44849122618     PISSN: None     EISSN: 15309932     Source Type: Journal    
DOI: 10.1208/s12249-007-9028-2     Document Type: Article
Times cited : (107)

References (35)
  • 1
    • 24944588804 scopus 로고    scopus 로고
    • Saturated phospholipids promote crystallization but slow down polymorphic transitions in triglyceride nanoparticles
    • H. Bunjes, and M. H. J. Koch. Saturated phospholipids promote crystallization but slow down polymorphic transitions in triglyceride nanoparticles. J. Control. Release. 107:229-243 (2005).
    • (2005) J. Control. Release. , vol.107 , pp. 229-243
    • Bunjes, H.1    Koch, M.H.J.2
  • 3
    • 2442712381 scopus 로고    scopus 로고
    • Development of a controlled release formulation based on SLN and NLC for topical clotrimazole delivery
    • E. B. Souto, S. A. Wissing, C. M. Barbosa, and R. H. Muller. Development of a controlled release formulation based on SLN and NLC for topical clotrimazole delivery. Int. J. Pharm. 278:71-77 (2004).
    • (2004) Int. J. Pharm. , vol.278 , pp. 71-77
    • Souto, E.B.1    Wissing, S.A.2    Barbosa, C.M.3    Muller, R.H.4
  • 5
    • 0002277454 scopus 로고
    • Analgesic-antipyretics and anti-inflammatory agents: Drugs employed in the treatment of rheumatoid arthritis and gout
    • In L. S. Goodman, A. Gilman, T. W. Rall, A. S. Nies, and P. Taylor (eds.) McGraw-Hill International editions, New York, NY
    • P. A. Insel. Analgesic-antipyretics and anti-inflammatory agents: Drugs employed in the treatment of rheumatoid arthritis and gout. In L. S. Goodman, A. Gilman, T. W. Rall, A. S. Nies, and P. Taylor (eds.), The pharmacological basis of therapeutics, McGraw-Hill International editions, New York, NY, 1992, pp. 638-681.
    • (1992) The Pharmacological Basis of Therapeutics , pp. 638-681
    • Insel, P.A.1
  • 6
    • 53849103609 scopus 로고
    • Inventors. Liposphere delivery systems for local anesthetics
    • US patent 5 227 165. July 13
    • A. Domb and M. Maniar, Inventors. Liposphere delivery systems for local anesthetics. US patent 5 227 165. July 13, 1993.
    • (1993)
    • Domb, A.1    Maniar, M.2
  • 7
    • 0031847390 scopus 로고    scopus 로고
    • Liposphere local anesthetic timed-release for perineural site application
    • D. B. Masters and A. J. Domb. Liposphere local anesthetic timed-release for perineural site application. Pharm. Res. 15:1038-1045 (1998).
    • (1998) Pharm. Res. , vol.15 , pp. 1038-1045
    • Masters, D.B.1    Domb, A.J.2
  • 8
    • 33646841839 scopus 로고    scopus 로고
    • Influence of liposphere preparation on butyl-methoxydibenzoyl methane photostability
    • V. Iannuccelli, N. Sala, R. Tursilli, G. Coppi, and S. Scalia. Influence of liposphere preparation on butyl-methoxydibenzoyl methane photostability. Eur. J. Pharm. Biopharm. 63:140-145 (2006).
    • (2006) Eur. J. Pharm. Biopharm. , vol.63 , pp. 140-145
    • Iannuccelli, V.1    Sala, N.2    Tursilli, R.3    Coppi, G.4    Scalia, S.5
  • 9
    • 32944472872 scopus 로고    scopus 로고
    • Enhancement of melatonin photostability by encapsulation in lipospheres
    • R. Tursilli, A. Casolari, V. Iannuccelli, and S. Scalia. Enhancement of melatonin photostability by encapsulation in lipospheres. J. Pharm. Biomed. Anal. 40:910-914 (2006).
    • (2006) J. Pharm. Biomed. Anal. , vol.40 , pp. 910-914
    • Tursilli, R.1    Casolari, A.2    Iannuccelli, V.3    Scalia, S.4
  • 10
    • 16244375867 scopus 로고    scopus 로고
    • Effect of hexacosanol on the characteristics of novel sustained release allopurinol solid lipospheres (SLS): Factorial design application and product evaluation
    • I. El Gibaly, and S. K. Abdel-Ghaffar. Effect of hexacosanol on the characteristics of novel sustained release allopurinol solid lipospheres (SLS): Factorial design application and product evaluation. Int. J. Pharm. 294:33-51 (2005).
    • (2005) Int. J. Pharm. , vol.294 , pp. 33-51
    • El Gibaly, I.1    Abdel-Ghaffar, S.K.2
  • 11
    • 3242724894 scopus 로고    scopus 로고
    • Formulation and characterization of bupivacaine lipospheres
    • S. Toongsuwan, L. Li, B. K. Erickson, and H. Chang. Formulation and characterization of bupivacaine lipospheres. Int. J. Pharm. 280:57-65 (2004).
    • (2004) Int. J. Pharm. , vol.280 , pp. 57-65
    • Toongsuwan, S.1    Li, L.2    Erickson, B.K.3    Chang, H.4
  • 12
    • 11144326726 scopus 로고    scopus 로고
    • Anti-inflammatory effects of jojoba liquid wax in experimental models
    • R. R. Habashy, A. B. Abdel-Naim, A. E. Khalifa, and M. M. Al-Azizi. Anti-inflammatory effects of jojoba liquid wax in experimental models. Pharmacol. Res. 51:95-105 (2005).
    • (2005) Pharmacol. Res. , vol.51 , pp. 95-105
    • Habashy, R.R.1    Abdel-Naim, A.B.2    Khalifa, A.E.3    Al-Azizi, M.M.4
  • 13
    • 0042335999 scopus 로고    scopus 로고
    • Solid lipid nanoparticles and microemulsion for topical delivery of triptolide
    • Z. Mei, H. Chen, T. Weng, Y. Yang, and X. Yang. Solid lipid nanoparticles and microemulsion for topical delivery of triptolide. Eur. J. Pharm. Biopharm. 56:189-196 (2003).
    • (2003) Eur. J. Pharm. Biopharm. , vol.56 , pp. 189-196
    • Mei, Z.1    Chen, H.2    Weng, T.3    Yang, Y.4    Yang, X.5
  • 14
    • 0035821356 scopus 로고    scopus 로고
    • Development and characterization of lipid microparticles as a drug carrier for somatostatin
    • H. Reithmeier, J. Herrmann, and A. Gopferich. Development and characterization of lipid microparticles as a drug carrier for somatostatin. Int. J. Pharm. 218:133-143 (2001).
    • (2001) Int. J. Pharm. , vol.218 , pp. 133-143
    • Reithmeier, H.1    Herrmann, J.2    Gopferich, A.3
  • 15
    • 84860761485 scopus 로고
    • Characterization of Lipospheres ™-1: Effect of carrier and phospholipid on the loading of drug into the lipospheres
    • M. Maniar, D. Hannibal, S. Amselem, X. Xie, R. Burch, and A. Domb. Characterization of Lipospheres ™-1: Effect of carrier and phospholipid on the loading of drug into the lipospheres. Pharm. Res. 8 suppl.: S-185 (1991).
    • (1991) Pharm. Res. , vol.8 , Issue.SUPPL.
    • Maniar, M.1    Hannibal, D.2    Amselem, S.3    Xie, X.4    Burch, R.5    Domb, A.6
  • 16
    • 31544443007 scopus 로고    scopus 로고
    • In vitro characterization of carbamazepine-loaded precifac lipospheres
    • N. S. Barakat, and A. E. B. Yassin. In vitro characterization of carbamazepine-loaded precifac lipospheres. Drug Delivery 13:95-104 (2006).
    • (2006) Drug Delivery , vol.13 , pp. 95-104
    • Barakat, N.S.1    Yassin, A.E.B.2
  • 17
    • 0036130944 scopus 로고    scopus 로고
    • Production of lipospheres as carriers for bioactive compounds
    • R. Cortesi, E. Esposito, G. Luca, and C. Nastruzzi. Production of lipospheres as carriers for bioactive compounds. Biomaterials 23:2283-2294 (2002).
    • (2002) Biomaterials , vol.23 , pp. 2283-2294
    • Cortesi, R.1    Esposito, E.2    Luca, G.3    Nastruzzi, C.4
  • 18
    • 0025179160 scopus 로고
    • The effect of lipid composition upon the encapsulation and in vitro leakage of metaproterenol sulfate from 0.2 μm diameter, extruded, multilamellar liposomes
    • R. M. Abra, P. J. Mihalko, and H. Schreier. The effect of lipid composition upon the encapsulation and in vitro leakage of metaproterenol sulfate from 0.2 μm diameter, extruded, multilamellar liposomes. J. Control. Release. 14:71-78 (1990).
    • (1990) J. Control. Release. , vol.14 , pp. 71-78
    • Abra, R.M.1    Mihalko, P.J.2    Schreier, H.3
  • 19
    • 20444493102 scopus 로고    scopus 로고
    • Encapsulation efficiency of water-soluble and insoluble drugs in liposomes prepared by the microencapsulation vesicle method
    • T. Nii, and F. Ishii. Encapsulation efficiency of water-soluble and insoluble drugs in liposomes prepared by the microencapsulation vesicle method. Int. J. Pharm. 298:198-205 (2005).
    • (2005) Int. J. Pharm. , vol.298 , pp. 198-205
    • Nii, T.1    Ishii, F.2
  • 20
    • 12344276507 scopus 로고    scopus 로고
    • Preparation and characterization of solid lipid nanoparticles (SLN) made of cacao butter and curdlan
    • B. D. Kim, K. Na, and H. K. Choi. Preparation and characterization of solid lipid nanoparticles (SLN) made of cacao butter and curdlan. Eur. J. Pharm. Sci. 24:199-205 (2005).
    • (2005) Eur. J. Pharm. Sci. , vol.24 , pp. 199-205
    • Kim, B.D.1    Na, K.2    Choi, H.K.3
  • 21
    • 0043170806 scopus 로고    scopus 로고
    • Assessment of diclofenac permeation with different formulations: Anti-inflammatory study of a selected formula
    • E. Escribano, A. C. Calpena, J. Queralt, R. Obach, and J. Domenech. Assessment of diclofenac permeation with different formulations: anti-inflammatory study of a selected formula. Eur. J. Pharm Sci. 19:203-210 (2003).
    • (2003) Eur. J. Pharm Sci. , vol.19 , pp. 203-210
    • Escribano, E.1    Calpena, A.C.2    Queralt, J.3    Obach, R.4    Domenech, J.5
  • 22
    • 33745527085 scopus 로고    scopus 로고
    • Deet-loaded solid lipid particles for skin delivery: In vitro release and skin permeation characteristics in different vehicles
    • Y. Iscan, S. Hekimoglu, M. F. Sargon, and A. A. Hincal. Deet-loaded solid lipid particles for skin delivery: In vitro release and skin permeation characteristics in different vehicles. J. Microencapsul. 23:315-327 (2006).
    • (2006) J. Microencapsul. , vol.23 , pp. 315-327
    • Iscan, Y.1    Hekimoglu, S.2    Sargon, M.F.3    Hincal, A.A.4
  • 23
    • 1942498889 scopus 로고    scopus 로고
    • Cyclosporin nanoparticulate lipospheres for oral administration
    • T. Bekerman, J. Golenser, and A. Domb. Cyclosporin nanoparticulate lipospheres for oral administration. J. Pharm. Sci. 93:1264-1270 (2004).
    • (2004) J. Pharm. Sci. , vol.93 , pp. 1264-1270
    • Bekerman, T.1    Golenser, J.2    Domb, A.3
  • 24
    • 0037404980 scopus 로고    scopus 로고
    • The production and characteristics of solid lipid nanoparticles (SLNs)
    • D. Hou, C. Xie, K. Huang, and C. Zhu. The production and characteristics of solid lipid nanoparticles (SLNs). Biomaterials 24:1781-1785 (2003).
    • (2003) Biomaterials , vol.24 , pp. 1781-1785
    • Hou, D.1    Xie, C.2    Huang, K.3    Zhu, C.4
  • 25
    • 0041571354 scopus 로고    scopus 로고
    • S. Budavari, M. J. O'Neil, A. Smith, P. E. Heckelman, J. F. Kinneary (eds.) Whitehouse station, NJ, Merck and Co
    • S. Budavari, M. J. O'Neil, A. Smith, P. E. Heckelman, J. F. Kinneary (eds.) The Merck Index, an Encyclopedia of Chemicals, Drugs and Biologicals. Whitehouse station, NJ, Merck and Co., 1996.
    • (1996) The Merck Index, an Encyclopedia of Chemicals, Drugs and Biologicals
  • 26
    • 33746418412 scopus 로고    scopus 로고
    • Encapsulation in lipospheres of the complex between butyl methoxydibenzoylmethane and hydroxypropyl-β-cyclodextrin
    • S. Scalia, R. Tursilli, N. Sala, and V. Iannuccelli. Encapsulation in lipospheres of the complex between butyl methoxydibenzoylmethane and hydroxypropyl-β-cyclodextrin. Int. J. Pharm. 320:79-85 (2006).
    • (2006) Int. J. Pharm. , vol.320 , pp. 79-85
    • Scalia, S.1    Tursilli, R.2    Sala, N.3    Iannuccelli, V.4
  • 27
    • 0031855617 scopus 로고    scopus 로고
    • Proniosome based transdermal delivery of levonorgesterol for effective contraception
    • B. Vora, A. J. Khopade, and N. K. Jain. Proniosome based transdermal delivery of levonorgesterol for effective contraception. J. Control. Release. 54:149-165 (1998).
    • (1998) J. Control. Release. , vol.54 , pp. 149-165
    • Vora, B.1    Khopade, A.J.2    Jain, N.K.3
  • 28
    • 0000568190 scopus 로고
    • Sustained release of liposome-encapsulated gentamycin and fate of phospholipid following intramuscular injection in mice
    • H. Schreier, M. Levy, and P. Mihalko. Sustained release of liposome-encapsulated gentamycin and fate of phospholipid following intramuscular injection in mice. J. Control. Release. 5:187-192 (1987).
    • (1987) J. Control. Release. , vol.5 , pp. 187-192
    • Schreier, H.1    Levy, M.2    Mihalko, P.3
  • 29
    • 0035910870 scopus 로고    scopus 로고
    • Preparation of semisolid drug carriers for topical application based on solid lipid nanoparticles
    • A. Lippacher, R. H. Muller, and K. Mader. Preparation of semisolid drug carriers for topical application based on solid lipid nanoparticles. Int. J. Pharm. 214:9-12 (2001).
    • (2001) Int. J. Pharm. , vol.214 , pp. 9-12
    • Lippacher, A.1    Muller, R.H.2    Mader, K.3
  • 30
    • 0033975896 scopus 로고    scopus 로고
    • An investigation into the release of cefuroxime axetil from taste-masked stearic acid microspheres II. The effects of buffer composition on drug release
    • H. Robson, D. Q. M. Craig, and D. Deutsch. An investigation into the release of cefuroxime axetil from taste-masked stearic acid microspheres II. The effects of buffer composition on drug release. Int. J. Pharm. 195:137-145 (2000).
    • (2000) Int. J. Pharm. , vol.195 , pp. 137-145
    • Robson, H.1    Craig, D.Q.M.2    Deutsch, D.3
  • 31
    • 2242472082 scopus 로고    scopus 로고
    • Solid lipid nanoparticles (SLN) and nanostructured lipid carriers (NLC) in cosmetic and dermatological preparations
    • R. H. Muller, M. Radtke, and S. A. Wissing. Solid lipid nanoparticles (SLN) and nanostructured lipid carriers (NLC) in cosmetic and dermatological preparations. Adv. Drug Deliv. Rev. 54:S131-S155 (2002).
    • (2002) Adv. Drug Deliv. Rev. , vol.54
    • Muller, R.H.1    Radtke, M.2    Wissing, S.A.3
  • 32
    • 1942453805 scopus 로고    scopus 로고
    • Solid lipid nanoparticles for parentral drug delivery
    • S. A. Wissing, O. Kayser, and R. H. Muller. Solid lipid nanoparticles for parentral drug delivery. Adv. Drug Deliv. Rev. 56:1257-1272 (2004).
    • (2004) Adv. Drug Deliv. Rev. , vol.56 , pp. 1257-1272
    • Wissing, S.A.1    Kayser, O.2    Muller, R.H.3
  • 33
    • 0036008754 scopus 로고    scopus 로고
    • Semisolid SLN™ dispersions for topical application influence of formulation and production parameters on viscoelastic properties
    • A. Lippacher, R. H. Muller, and K. Mader. Semisolid SLN™ dispersions for topical application influence of formulation and production parameters on viscoelastic properties. Eur. J. Pharm. Biopharm. 53:155-160 (2002).
    • (2002) Eur. J. Pharm. Biopharm. , vol.53 , pp. 155-160
    • Lippacher, A.1    Muller, R.H.2    Mader, K.3
  • 34
    • 30844438968 scopus 로고    scopus 로고
    • A novel approach based on lipid nanoparticles (SLN ®) for topical delivery of a-lipoic acid
    • E. B. Souto, R. H. Muller, and S. Gohla. A novel approach based on lipid nanoparticles (SLN ®) for topical delivery of a-lipoic acid. J. Microencapsul. 22:581-592 (2005).
    • (2005) J. Microencapsul. , vol.22 , pp. 581-592
    • Souto, E.B.1    Muller, R.H.2    Gohla, S.3
  • 35
    • 16544392907 scopus 로고    scopus 로고
    • Tamoxifen in topical liposomes: Development, characterization and in-vitro evaluation
    • A. Bhatia, R. Kumar, and O. P. Katare. Tamoxifen in topical liposomes: development, characterization and in-vitro evaluation. J. Pharm. Pharmaceut. Sci. 7:252-259 (2004).
    • (2004) J. Pharm. Pharmaceut. Sci. , vol.7 , pp. 252-259
    • Bhatia, A.1    Kumar, R.2    Katare, O.P.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.