메뉴 건너뛰기




Volumn 586, Issue 11, 2008, Pages 2743-2752

Cyclothiazide: A subunit-specific inhibitor of GABAC receptors

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOBUTYRIC ACID C RECEPTOR; CYCLOTHIAZIDE; RECEPTOR SUBUNIT; 4 AMINOBUTYRIC ACID A RECEPTOR; PROLINE; SERINE;

EID: 44449168726     PISSN: 00223751     EISSN: 14697793     Source Type: Journal    
DOI: 10.1113/jphysiol.2008.153346     Document Type: Article
Times cited : (11)

References (29)
  • 1
    • 0014094028 scopus 로고
    • The antihypertensive effect of cyclothiazide, a double blind study
    • Antlitz AM & Valle NG (1967). The antihypertensive effect of cyclothiazide, a double blind study. Curr Ther Res Clin Exp 9, 288-292.
    • (1967) Curr Ther Res Clin Exp , vol.9 , pp. 288-292
    • Antlitz, A.M.1    Valle, N.G.2
  • 2
    • 0033137017 scopus 로고    scopus 로고
    • A novel presynaptic inhibitory mechanism underlies paired pulse depression at a fast central synapse
    • Bellingham MC & Walmsley B (1999). A novel presynaptic inhibitory mechanism underlies paired pulse depression at a fast central synapse. Neuron 23, 159-170.
    • (1999) Neuron , vol.23 , pp. 159-170
    • Bellingham, M.C.1    Walmsley, B.2
  • 3
    • 0027140862 scopus 로고
    • Modulation of AMPA/kainate receptors by analogues of diazoxide and cyclothiazide in thin slices of rat hippocampus
    • Bertolino M, Baraldi M, Parenti C, Braghiroli D, DiBella M, Vicini S & Costa E (1993). Modulation of AMPA/kainate receptors by analogues of diazoxide and cyclothiazide in thin slices of rat hippocampus. Receptors Channels 1, 267-278.
    • (1993) Receptors Channels , vol.1 , pp. 267-278
    • Bertolino, M.1    Baraldi, M.2    Parenti, C.3    Braghiroli, D.4    DiBella, M.5    Vicini, S.6    Costa, E.7
  • 4
    • 0242363125 scopus 로고    scopus 로고
    • Cyclothiazide potently inhibits γ-aminobutyric acid type A receptors in addition to enhancing glutamate responses
    • Deng L & Chen G (2003). Cyclothiazide potently inhibits γ-aminobutyric acid type A receptors in addition to enhancing glutamate responses. Proc Natl Acad Sci U S A 100, 13025-13029.
    • (2003) Proc Natl Acad Sci U S A , vol.100 , pp. 13025-13029
    • Deng, L.1    Chen, G.2
  • 5
    • 0028792374 scopus 로고
    • Asynchronous release of synaptic vesicles determines the time course of the AMPA receptor-mediated EPSC
    • Diamond JS & Jahr CE (1995). Asynchronous release of synaptic vesicles determines the time course of the AMPA receptor-mediated EPSC. Neuron 15, 1097-1107.
    • (1995) Neuron , vol.15 , pp. 1097-1107
    • Diamond, J.S.1    Jahr, C.E.2
  • 7
    • 0030540969 scopus 로고    scopus 로고
    • Use-dependent and use-independent blocking actions of picrotoxin and zinc at the GABA C receptor in retinal horizontal cells
    • Dong CJ & Werblin FS (1996). Use-dependent and use-independent blocking actions of picrotoxin and zinc at the GABA C receptor in retinal horizontal cells. Vision Res 36, 3997-4005.
    • (1996) Vision Res , vol.36 , pp. 3997-4005
    • Dong, C.J.1    Werblin, F.S.2
  • 8
    • 0032587999 scopus 로고    scopus 로고
    • C receptor ρ subunits are heterogeneously expressed in the human CNS and form homo- and heterooligomers with distinct physical properties
    • C receptor ρ subunits are heterogeneously expressed in the human CNS and form homo- and heterooligomers with distinct physical properties. Eur J Neurosci 11, 41-50.
    • (1999) Eur J Neurosci , vol.11 , pp. 41-50
    • Enz, R.1    Cutting, G.R.2
  • 9
    • 0029990678 scopus 로고    scopus 로고
    • New developments in the molecular pharmacology of alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionate and kainate receptors
    • Fletcher EJ & Lodge D (1996). New developments in the molecular pharmacology of alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionate and kainate receptors. Pharmacol Ther 70, 65-89.
    • (1996) Pharmacol Ther , vol.70 , pp. 65-89
    • Fletcher, E.J.1    Lodge, D.2
  • 10
    • 34250018794 scopus 로고    scopus 로고
    • A receptors exhibit two distinct and separable agonist affinities
    • A receptors exhibit two distinct and separable agonist affinities. J Physiol 581, 1001-1018.
    • (2007) J Physiol , vol.581 , pp. 1001-1018
    • Hadley, S.H.1    Amin, J.2
  • 11
    • 0035369889 scopus 로고    scopus 로고
    • Mechanisms underlying presynaptic facilitatory effect of cyclothiazide at the calyx of Held of juvenile rats
    • Ishikawa T & Takahashi T (2001). Mechanisms underlying presynaptic facilitatory effect of cyclothiazide at the calyx of Held of juvenile rats. J Physiol 533, 423-431.
    • (2001) J Physiol , vol.533 , pp. 423-431
    • Ishikawa, T.1    Takahashi, T.2
  • 12
    • 34047216195 scopus 로고    scopus 로고
    • Targeting AMPA receptor gating processes with allosteric modulators and mutations
    • Mitchell NA & Fleck MW (2007). Targeting AMPA receptor gating processes with allosteric modulators and mutations. Biophys J 92, 2392-2402.
    • (2007) Biophys J , vol.92 , pp. 2392-2402
    • Mitchell, N.A.1    Fleck, M.W.2
  • 13
    • 0028935086 scopus 로고
    • Structural determinants of allosteric regulation in alternatively spliced AMPA receptors
    • Partin KM, Bowie D & Mayer ML (1995). Structural determinants of allosteric regulation in alternatively spliced AMPA receptors. Neuron 14, 833-843.
    • (1995) Neuron , vol.14 , pp. 833-843
    • Partin, K.M.1    Bowie, D.2    Mayer, M.L.3
  • 14
    • 0029862192 scopus 로고    scopus 로고
    • AMPA receptor flip/flop mutants affecting deactivation, desensitization, and modulation by cyclothiazide, aniracetam, and thiocyanate
    • Partin KM, Fleck MW & Mayer ML (1996). AMPA receptor flip/flop mutants affecting deactivation, desensitization, and modulation by cyclothiazide, aniracetam, and thiocyanate. J Neurosci 16, 6634-6647.
    • (1996) J Neurosci , vol.16 , pp. 6634-6647
    • Partin, K.M.1    Fleck, M.W.2    Mayer, M.L.3
  • 15
    • 0027715150 scopus 로고
    • Selective modulation of desensitization at AMPA versus kainate receptors by cyclothiazide and concanavalin A
    • Partin KM, Patneau DK, Winters CA, Mayer ML & Buonanno A (1993). Selective modulation of desensitization at AMPA versus kainate receptors by cyclothiazide and concanavalin A. Neuron 11, 1069-1082.
    • (1993) Neuron , vol.11 , pp. 1069-1082
    • Partin, K.M.1    Patneau, D.K.2    Winters, C.A.3    Mayer, M.L.4    Buonanno, A.5
  • 16
    • 0031782676 scopus 로고    scopus 로고
    • Molecular and pharmacological properties of GABA-ρ subunits from white perch retina
    • Qian H, Dowling JE & Ripps H (1998). Molecular and pharmacological properties of GABA-ρ subunits from white perch retina. J Neurobiol 37, 305-320.
    • (1998) J Neurobiol , vol.37 , pp. 305-320
    • Qian, H.1    Dowling, J.E.2    Ripps, H.3
  • 19
    • 0035542638 scopus 로고    scopus 로고
    • C receptors of retinal neurons
    • In ed. Kolb H, Ripps H & Wu S, Elsevier Science B.V. Amsterdam, The Netherlands
    • C receptors of retinal neurons. In Progress in Brain Research, ed. Kolb H, Ripps H & Wu S, pp. 295-308. Elsevier Science B.V. Amsterdam, The Netherlands.
    • (2001) Progress in Brain Research , pp. 295-308
    • Qian, H.1    Ripps, H.2
  • 20
    • 34547876902 scopus 로고    scopus 로고
    • Streptozotocin-induced diabetes modulates GABA receptor activity of rat retinal neurons
    • Ramsey DJ, Ripps H & Qian H (2007). Streptozotocin-induced diabetes modulates GABA receptor activity of rat retinal neurons. Exp Eye Res 85, 413-422.
    • (2007) Exp Eye Res , vol.85 , pp. 413-422
    • Ramsey, D.J.1    Ripps, H.2    Qian, H.3
  • 21
    • 0036460422 scopus 로고    scopus 로고
    • Expression and dendritic mRNA localization of GABA C receptor ρ1 and ρ2 subunits in developing rat brain and spinal cord
    • Rozzo A, Armellin M, Franzot J, Chiaruttini C, Nistri A & Tongiorgi E (2002). Expression and dendritic mRNA localization of GABA C receptor ρ1 and ρ2 subunits in developing rat brain and spinal cord. Eur J Neurosci 15, 1747-1758.
    • (2002) Eur J Neurosci , vol.15 , pp. 1747-1758
    • Rozzo, A.1    Armellin, M.2    Franzot, J.3    Chiaruttini, C.4    Nistri, A.5    Tongiorgi, E.6
  • 23
    • 0027210626 scopus 로고
    • Desensitization of AMPA receptors upon multiquantal neurotransmitter release
    • Trussell LO, Zhang S & Raman IM (1993). Desensitization of AMPA receptors upon multiquantal neurotransmitter release. Neuron 10, 1185-1196.
    • (1993) Neuron , vol.10 , pp. 1185-1196
    • Trussell, L.O.1    Zhang, S.2    Raman, I.M.3
  • 24
    • 0029610075 scopus 로고
    • A single amino acid in γ-aminobutyric acid ρ1 receptors affects competitive and noncompetitive components of picrotoxin inhibition
    • Wang TL, Hackam AS, Guggino WB & Cutting GR (1995). A single amino acid in γ-aminobutyric acid ρ1 receptors affects competitive and noncompetitive components of picrotoxin inhibition. Proc Natl Acad Sci U S A 92, 11751-11755.
    • (1995) Proc Natl Acad Sci U S A , vol.92 , pp. 11751-11755
    • Wang, T.L.1    Hackam, A.S.2    Guggino, W.B.3    Cutting, G.R.4
  • 26
    • 0027209412 scopus 로고
    • Benzothiadiazides inhibit rapid glutamate receptor desensitization and enhance glutamatergic synaptic currents
    • Yamada KA & Tang CM (1993). Benzothiadiazides inhibit rapid glutamate receptor desensitization and enhance glutamatergic synaptic currents. J Neurosci 13, 3904-3915.
    • (1993) J Neurosci , vol.13 , pp. 3904-3915
    • Yamada, K.A.1    Tang, C.M.2
  • 28
    • 0029417199 scopus 로고
    • Cloning of a γ-aminobutyric acid type C receptor subunit in rat retina with a methionine residue critical for picrotoxinin channel block
    • Zhang D, Pan ZH, Zhang X, Brideau AD & Lipton SA (1995). Cloning of a γ-aminobutyric acid type C receptor subunit in rat retina with a methionine residue critical for picrotoxinin channel block. Proc Natl Acad Sci U S A 92, 11756-11760.
    • (1995) Proc Natl Acad Sci U S A , vol.92 , pp. 11756-11760
    • Zhang, D.1    Pan, Z.H.2    Zhang, X.3    Brideau, A.D.4    Lipton, S.A.5
  • 29
    • 34247394266 scopus 로고    scopus 로고
    • A single amino acid in the second transmembrane domain of GABA ρ receptors regulates channel conductance
    • Zhu Y, Ripps H & Qian H (2007). A single amino acid in the second transmembrane domain of GABA ρ receptors regulates channel conductance. Neurosci Lett 418, 205-209.
    • (2007) Neurosci Lett , vol.418 , pp. 205-209
    • Zhu, Y.1    Ripps, H.2    Qian, H.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.