SCOPUS 정보 검색 플랫폼

Volumn 47, Issue 19, 2004, Pages 4642-4644

Potent and orally bioavailable non-peptide antagonists at the human bradykinin B1 receptor based on a 2-alkylamino-5-sulfamoylbenzamide core

(15) Ritchie, Timothy J a Dziadulewicz, Edward K a Culshaw, Andrew J a Müller, Werner b Burgess, Gillian M c Bloomfield, Graham C d Drake, Gillian S a Dunstan, Andrew R d Beattie, David d Hughes, Glyn A a Ganju, Pam a McIntyre, Peter a Bevan, Stuart J a Davis, Clare a Yaqoob, Mohammed a

a Novartis Inst for Medical Sciences (United Kingdom)

b NOVARTIS PHARMA AG (Switzerland)

c PFIZER GLOBAL RESEARCH AND DEVELOPMENT (United Kingdom)

d NOVARTIS HORSHAM RESEARCH CENTRE (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

5 SULFAMOYLBENZAMIDE DERIVATIVE; AMINE; AMINO ACID; ANILINE; BENZAMIDE DERIVATIVE; BRADYKININ B1 RECEPTOR; BRADYKININ B1 RECEPTOR ANTAGONIST; ISONIPECOTIC ACID; SULFONAMIDE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; BINDING AFFINITY; CELL STRAIN COS7; CONTROLLED STUDY; DRUG BIOAVAILABILITY; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; HYDROPHOBICITY; HYPERALGESIA; INFLAMMATION; NONHUMAN; RAT; TISSUE INJURY;

ADMINISTRATION, ORAL; AMINES; AMINO ACIDS; ANTHRANILIC ACIDS; BIOLOGICAL AVAILABILITY; CARBOXYLIC ACIDS; HUMANS; MOLECULAR STRUCTURE; PEPTIDES; RECEPTOR, BRADYKININ B1;

EID: 4444315533 PISSN: 00222623 EISSN: None Source Type: Journal
DOI: 10.1021/jm049747g Document Type: Article

Times cited : (30)

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