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Volumn 69, Issue 2, 2008, Pages 597-604

Transdermal and dermal delivery of adefovir: Effects of pH and permeation enhancers

Author keywords

Acyclic nucleoside phosphonates; Adefovir; Permeation enhancer; Skin absorption; Transdermal drug delivery

Indexed keywords

ADEFOVIR; CARBAMIC ACID DERIVATIVE; LAUROCAPRAM; LAURYL ALCOHOL; PROPIONIC ACID DERIVATIVE;

EID: 43249128108     PISSN: 09396411     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejpb.2007.12.005     Document Type: Article
Times cited : (39)

References (37)
  • 1
    • 7744241924 scopus 로고    scopus 로고
    • Adefovir dipivoxil: review of a novel acyclic nucleoside analogue
    • Danta M., and Dusheiko G. Adefovir dipivoxil: review of a novel acyclic nucleoside analogue. Int. J. Clin. Pract. 58 (2004) 877-886
    • (2004) Int. J. Clin. Pract. , vol.58 , pp. 877-886
    • Danta, M.1    Dusheiko, G.2
  • 2
    • 0345138983 scopus 로고    scopus 로고
    • Phosphonomethoxyalkyl analogs of nucleotides
    • Holy A. Phosphonomethoxyalkyl analogs of nucleotides. Curr. Pharm. Des. 9 (2003) 2567-2592
    • (2003) Curr. Pharm. Des. , vol.9 , pp. 2567-2592
    • Holy, A.1
  • 3
    • 1242308254 scopus 로고    scopus 로고
    • Current status and future potential of transdermal drug delivery
    • Prausnitz M.R., Mitragotri S., and Langer R. Current status and future potential of transdermal drug delivery. Nat. Rev. Drug Discov. 3 (2004) 115-124
    • (2004) Nat. Rev. Drug Discov. , vol.3 , pp. 115-124
    • Prausnitz, M.R.1    Mitragotri, S.2    Langer, R.3
  • 5
    • 0034008388 scopus 로고    scopus 로고
    • Cytotoxicity of antiviral nucleotides adefovir and cidofovir is induced by the expression of human renal organic anion transporter 1
    • Ho E.S., Lin D.C., Mendel D.B., and Cihlar T. Cytotoxicity of antiviral nucleotides adefovir and cidofovir is induced by the expression of human renal organic anion transporter 1. J. Am. Soc. Nephrol. 11 (2000) 383-393
    • (2000) J. Am. Soc. Nephrol. , vol.11 , pp. 383-393
    • Ho, E.S.1    Lin, D.C.2    Mendel, D.B.3    Cihlar, T.4
  • 6
    • 17844373273 scopus 로고    scopus 로고
    • Transdermal drug delivery: penetration enhancement techniques
    • Benson H.A. Transdermal drug delivery: penetration enhancement techniques. Curr. Drug Deliv. 2 (2005) 23-33
    • (2005) Curr. Drug Deliv. , vol.2 , pp. 23-33
    • Benson, H.A.1
  • 8
    • 23844512530 scopus 로고    scopus 로고
    • Amphiphilic transdermal permeation enhancers: structure-activity relationships
    • Vávrová K., Zbytovská J., and Hrabálek A. Amphiphilic transdermal permeation enhancers: structure-activity relationships. Curr. Med. Chem. 12 (2005) 2273-2291
    • (2005) Curr. Med. Chem. , vol.12 , pp. 2273-2291
    • Vávrová, K.1    Zbytovská, J.2    Hrabálek, A.3
  • 9
    • 0029036834 scopus 로고
    • Optimization of in vitro flux through hairless mouse skin of cidofovir, a potent nucleotide analog
    • Aspe E., Guy R.H., Lee W.A., Kennedy J.A., Visor G.C., and Ennis R.D. Optimization of in vitro flux through hairless mouse skin of cidofovir, a potent nucleotide analog. J. Pharm. Sci. 84 (1995) 750-754
    • (1995) J. Pharm. Sci. , vol.84 , pp. 750-754
    • Aspe, E.1    Guy, R.H.2    Lee, W.A.3    Kennedy, J.A.4    Visor, G.C.5    Ennis, R.D.6
  • 10
    • 0028107422 scopus 로고
    • Oral, subcutaneous, and intramuscular bioavailabilities of the antiviral nucleotide analog 9-(2-phosphonylmethoxyethyl) adenine in cynomolgus monkeys
    • Cundy K.C., Shaw J.P., and Lee W.A. Oral, subcutaneous, and intramuscular bioavailabilities of the antiviral nucleotide analog 9-(2-phosphonylmethoxyethyl) adenine in cynomolgus monkeys. Antimicrob. Agents Chemother. 38 (1994) 365-368
    • (1994) Antimicrob. Agents Chemother. , vol.38 , pp. 365-368
    • Cundy, K.C.1    Shaw, J.P.2    Lee, W.A.3
  • 11
    • 0037205832 scopus 로고    scopus 로고
    • Determination of cidofovir in both skin layers and percutaneous penetration samples by HPLC
    • Santoyo S., de Jalon E.G., Campanero M.A., and Ygartua P. Determination of cidofovir in both skin layers and percutaneous penetration samples by HPLC. J. Pharm. Biomed. Anal. 29 (2002) 819-826
    • (2002) J. Pharm. Biomed. Anal. , vol.29 , pp. 819-826
    • Santoyo, S.1    de Jalon, E.G.2    Campanero, M.A.3    Ygartua, P.4
  • 13
    • 34250020296 scopus 로고    scopus 로고
    • HPLC method for determination of transdermal and dermal delivery of adefovir (PMEA)
    • Vávrová K., Lorencová K., Klimentová J., Novotný J., and Hrabálek A. HPLC method for determination of transdermal and dermal delivery of adefovir (PMEA). J. Chrom. B 853 (2007) 198-203
    • (2007) J. Chrom. B , vol.853 , pp. 198-203
    • Vávrová, K.1    Lorencová, K.2    Klimentová, J.3    Novotný, J.4    Hrabálek, A.5
  • 14
    • 0001153009 scopus 로고
    • Acyclic nucleotide analogs. 3. Synthesis of 9-(2-phosphonylmethoxyethyl)adenine and related-compounds
    • Holy A., and Rosenberg I. Acyclic nucleotide analogs. 3. Synthesis of 9-(2-phosphonylmethoxyethyl)adenine and related-compounds. Collect. Czech. Chem. Commun. 52 (1987) 2801-2809
    • (1987) Collect. Czech. Chem. Commun. , vol.52 , pp. 2801-2809
    • Holy, A.1    Rosenberg, I.2
  • 15
    • 0019940117 scopus 로고
    • Enhanced percutaneous penetration with 1-dodecylazacycloheptan-2-one
    • Stoughton R.B. Enhanced percutaneous penetration with 1-dodecylazacycloheptan-2-one. Arch. Dermatol. 118 (1982) 474-477
    • (1982) Arch. Dermatol. , vol.118 , pp. 474-477
    • Stoughton, R.B.1
  • 16
    • 0027524981 scopus 로고
    • Synthesis and enhancing effect of dodecyl 2-(N,N-dimethylamino)propionate on the transepidermal delivery of indomethacin, clonidine, and hydrocortisone
    • Buyuktimkin S., Buyuktimkin N., and Rytting J.H. Synthesis and enhancing effect of dodecyl 2-(N,N-dimethylamino)propionate on the transepidermal delivery of indomethacin, clonidine, and hydrocortisone. Pharm. Res. 10 (1993) 1632-1637
    • (1993) Pharm. Res. , vol.10 , pp. 1632-1637
    • Buyuktimkin, S.1    Buyuktimkin, N.2    Rytting, J.H.3
  • 17
    • 0027337992 scopus 로고
    • Epsilon-aminocaproic acid esters as transdermal penetration enhancing agents
    • Doležal P., Hrabálek A., and Semecký V. Epsilon-aminocaproic acid esters as transdermal penetration enhancing agents. Pharm. Res. 10 (1993) 1015-1019
    • (1993) Pharm. Res. , vol.10 , pp. 1015-1019
    • Doležal, P.1    Hrabálek, A.2    Semecký, V.3
  • 18
    • 33646889983 scopus 로고    scopus 로고
    • Synthesis and enhancing effect of transkarbam 12 on the transdermal delivery of theophylline, clotrimazole, flobufen, and griseofulvin
    • Hrabálek A., Doležal P., Vávrová K., Zbytovská J., Holas T., Klimentová J., and Novotný J. Synthesis and enhancing effect of transkarbam 12 on the transdermal delivery of theophylline, clotrimazole, flobufen, and griseofulvin. Pharm. Res. 23 (2006) 912-919
    • (2006) Pharm. Res. , vol.23 , pp. 912-919
    • Hrabálek, A.1    Doležal, P.2    Vávrová, K.3    Zbytovská, J.4    Holas, T.5    Klimentová, J.6    Novotný, J.7
  • 19
    • 43249114575 scopus 로고    scopus 로고
    • Percutaneous Absorption: Drugs, Cosmetics, Mechanisms, Methods
    • Bronaugh R.L., and Maibach H.I. Percutaneous Absorption: Drugs, Cosmetics, Mechanisms, Methods. Informa Healthcare (2005) 696
    • (2005) Informa Healthcare , pp. 696
    • Bronaugh, R.L.1    Maibach, H.I.2
  • 20
    • 0016610679 scopus 로고
    • Percutaneous absorption on the relevance of in vitro data
    • Franz T.J. Percutaneous absorption on the relevance of in vitro data. J. Invest. Dermatol. 64 (1975) 190-195
    • (1975) J. Invest. Dermatol. , vol.64 , pp. 190-195
    • Franz, T.J.1
  • 22
    • 0014587011 scopus 로고
    • The effect of perfusion rate on in vitro percutaneous penetration
    • Crutcher W., and Maibach H.I. The effect of perfusion rate on in vitro percutaneous penetration. J. Invest. Dermatol. 53 (1969) 264-269
    • (1969) J. Invest. Dermatol. , vol.53 , pp. 264-269
    • Crutcher, W.1    Maibach, H.I.2
  • 24
    • 33745278513 scopus 로고    scopus 로고
    • Enhancement of transdermal delivery of 6-beta-naltrexol via a codrug linked to hydroxybupropion
    • Kiptoo P.K., Hamad M.O., Crooks P.A., and Stinchcomb A.L. Enhancement of transdermal delivery of 6-beta-naltrexol via a codrug linked to hydroxybupropion. J. Control. Release 113 (2006) 137-145
    • (2006) J. Control. Release , vol.113 , pp. 137-145
    • Kiptoo, P.K.1    Hamad, M.O.2    Crooks, P.A.3    Stinchcomb, A.L.4
  • 25
    • 0002246502 scopus 로고
    • Preparation of isolated sheets of human stratum corneum
    • Kligman A.M., and Christophers E. Preparation of isolated sheets of human stratum corneum. Arch. Dermatol. 88 (1963) 709-712
    • (1963) Arch. Dermatol. , vol.88 , pp. 709-712
    • Kligman, A.M.1    Christophers, E.2
  • 26
    • 0036295388 scopus 로고    scopus 로고
    • Raman spectroscopy study of acid-base and structural properties of 9-[2-(phosphonomethoxy)ethyl]adenine in aqueous solutions
    • Kopecky Jr. V., Mojzes P., Burda J.V., and Dostal L. Raman spectroscopy study of acid-base and structural properties of 9-[2-(phosphonomethoxy)ethyl]adenine in aqueous solutions. Biopolymers 67 (2002) 285-288
    • (2002) Biopolymers , vol.67 , pp. 285-288
    • Kopecky Jr., V.1    Mojzes, P.2    Burda, J.V.3    Dostal, L.4
  • 27
    • 42449085801 scopus 로고    scopus 로고
    • J. Levin, H.I. Maibach, Human skin buffering capacity: an overview, Skin Res. Technol, in press, doi:10.1111/j.1600-0846.2007.00271.x.
    • J. Levin, H.I. Maibach, Human skin buffering capacity: an overview, Skin Res. Technol, in press, doi:10.1111/j.1600-0846.2007.00271.x.
  • 28
    • 0000413401 scopus 로고    scopus 로고
    • Solution properties of antiviral adenine-nucleotide analogues. The acid-base properties of 9-[2-(phosphonomethoxy)ethyl]adenine (PMEA) and of its N1, N3 and N7 deaza derivatives in aqueous solution
    • Blindauer C.A., Holy A., Dvorakova H., and Sigel H. Solution properties of antiviral adenine-nucleotide analogues. The acid-base properties of 9-[2-(phosphonomethoxy)ethyl]adenine (PMEA) and of its N1, N3 and N7 deaza derivatives in aqueous solution. J. Chem. Soc., Perkin Trans. 2 (1997) 2353-2363
    • (1997) J. Chem. Soc., Perkin Trans. , vol.2 , pp. 2353-2363
    • Blindauer, C.A.1    Holy, A.2    Dvorakova, H.3    Sigel, H.4
  • 29
    • 0037237566 scopus 로고    scopus 로고
    • pH profiles in human skin: influence of two in vitro test systems for drug delivery testing
    • Wagner H., Kostka K.H., Lehr C.M., and Schaefer U.F. pH profiles in human skin: influence of two in vitro test systems for drug delivery testing. Eur. J. Pharm. Biopharm. 55 (2003) 57-65
    • (2003) Eur. J. Pharm. Biopharm. , vol.55 , pp. 57-65
    • Wagner, H.1    Kostka, K.H.2    Lehr, C.M.3    Schaefer, U.F.4
  • 30
    • 33750085043 scopus 로고    scopus 로고
    • Synthesis and transdermal permeation-enhancing activity of carbonate and carbamate analogs of Transkarbam 12
    • Holas T., Vávrová K., Ši{dotless}́ma M., Klimentová J., and Hrabálek A. Synthesis and transdermal permeation-enhancing activity of carbonate and carbamate analogs of Transkarbam 12. Bioorg. Med. Chem. 14 (2006) 7671-7680
    • (2006) Bioorg. Med. Chem. , vol.14 , pp. 7671-7680
    • Holas, T.1    Vávrová, K.2    Šíma, M.3    Klimentová, J.4    Hrabálek, A.5
  • 33
    • 0024587772 scopus 로고
    • Efficacy of phosphonylmethoxyalkyl derivatives of adenine in experimental herpes simplex virus and vaccinia virus infections in vivo
    • De Clercq E., Holy A., and Rosenberg I. Efficacy of phosphonylmethoxyalkyl derivatives of adenine in experimental herpes simplex virus and vaccinia virus infections in vivo. Antimicrob. Agents Chemother. 33 (1989) 185-191
    • (1989) Antimicrob. Agents Chemother. , vol.33 , pp. 185-191
    • De Clercq, E.1    Holy, A.2    Rosenberg, I.3
  • 34
    • 9444293982 scopus 로고    scopus 로고
    • Potent inhibition of human immunodeficiency virus and herpes simplex virus type 1 by 9-(2-phosphonylmethoxyethyl)adenine in primary macrophages is determined by drug metabolism, nucleotide pools, and cytokines
    • Perno C.F., Balestra E., Aquaro S., Panti S., Cenci A., Lazzarino G., Tavazzi B., Di Pierro D., Balzarini J., and Calio R. Potent inhibition of human immunodeficiency virus and herpes simplex virus type 1 by 9-(2-phosphonylmethoxyethyl)adenine in primary macrophages is determined by drug metabolism, nucleotide pools, and cytokines. Mol. Pharmacol. 50 (1996) 359-366
    • (1996) Mol. Pharmacol. , vol.50 , pp. 359-366
    • Perno, C.F.1    Balestra, E.2    Aquaro, S.3    Panti, S.4    Cenci, A.5    Lazzarino, G.6    Tavazzi, B.7    Di Pierro, D.8    Balzarini, J.9    Calio, R.10
  • 35
    • 0028884262 scopus 로고
    • Antiviral activity of selected acyclic nucleoside analogues against human herpesvirus 6
    • Reymen D., Naesens L., Balzarini J., Holy A., Dvorakova H., and De Clercq E. Antiviral activity of selected acyclic nucleoside analogues against human herpesvirus 6. Antivir. Res. 28 (1995) 343-357
    • (1995) Antivir. Res. , vol.28 , pp. 343-357
    • Reymen, D.1    Naesens, L.2    Balzarini, J.3    Holy, A.4    Dvorakova, H.5    De Clercq, E.6
  • 36
    • 0028873448 scopus 로고
    • Influence of propylene glycol as cosolvent on mechanism of drug transport from hydrogels
    • Bendas B., Schmalfuss U., and Neubert R. Influence of propylene glycol as cosolvent on mechanism of drug transport from hydrogels. Int. J. Pharm. 116 (1995) 19-30
    • (1995) Int. J. Pharm. , vol.116 , pp. 19-30
    • Bendas, B.1    Schmalfuss, U.2    Neubert, R.3
  • 37
    • 37349074682 scopus 로고    scopus 로고
    • Probing the permeation enhancement of mefenamic acid by ethanol across full-thickness skin, heat-separated epidermal membrane and heat-separated dermal membrane
    • Heard C.M., and Screen C. Probing the permeation enhancement of mefenamic acid by ethanol across full-thickness skin, heat-separated epidermal membrane and heat-separated dermal membrane. Int. J. Pharm. 349 (2008) 323-325
    • (2008) Int. J. Pharm. , vol.349 , pp. 323-325
    • Heard, C.M.1    Screen, C.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.