Synthesis and antimalarial activity of novel hydroxyethylamines, potential aspartyl protease inhibitors

Letters in Drug Design and Discovery

Volumn 5, Issue 3, 2008, Pages 178-181

  Cunico, Wilson ^a   Ferreira, Maria De Lourdes G ^a   Ferreira, Thaís G ^a   Penido, Carmen ^a   Henriques, Maria G M O ^a   Krettli, Luisa G ^b   Varotti, Fernando P ^b   Krettli, Antoniana U ^b  

^a INSTITUTO OSWALDO CRUZ   (Brazil)

^b FEDERAL UNIVERSITY OF MINAS GERAIS   (Brazil)

Author keywords

Antimalarial; Hydroxyethylamine; Protease inhibitors

Indexed keywords

ASPARTIC PROTEINASE INHIBITOR; ETHYLAMINE;

ANTIMALARIAL ACTIVITY; ARTICLE; CELL VIABILITY; CONTROLLED STUDY; CYTOTOXICITY; DRUG SYNTHESIS; DRUG TARGETING; HUMAN; HUMAN CELL; IC 50; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PLASMODIUM FALCIPARUM; PRIORITY JOURNAL;

EID: 42149154871     PISSN: 15701808     EISSN: None     Source Type: Journal    
DOI: 10.2174/157018008784083938     Document Type: Article

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