The therapeutic index of locally acting inhaled drugs as a function of their fine particle mass and particle size distribution - A literature review

Current Drug Delivery

Volumn 5, Issue 2, 2008, Pages 142-147

  Weda, Marjolein ^a   Zanen, Pieter ^b   De Boer, Anne H ^c   Barends, Dirk M ^a   Frijlink, Henderik W ^c  

^a NATIONAL INSTITUTE FOR PUBLIC HEALTH AND THE ENVIRONMENT   (Netherlands)

^b Heart Lung Center Utrecht   (Netherlands)

^c UNIVERSITY OF GRONINGEN   (Netherlands)

Author keywords

Adverse drug reactions; Efficacy; Fine particle mass; Inhaled drugs; Particle size distribution; Therapeutic index

Indexed keywords

BECLOMETASONE DIPROPIONATE; BRONCHODILATING AGENT; CORTICOSTEROID; FLUORINATED HYDROCARBON; IPRATROPIUM BROMIDE; SALBUTAMOL;

AEROSOL; CANDIDIASIS; DRUG ABSORPTION; DRUG DISTRIBUTION; DRUG DOSE INCREASE; DRUG EFFICACY; FINGER TREMOR; HUMAN; LUNG; LUNG DIFFUSION; PARTICLE SIZE; PRIORITY JOURNAL; REVIEW; SINGLE DRUG DOSE;

ADMINISTRATION, INHALATION; AEROSOLS; BRONCHODILATOR AGENTS; DELAYED-ACTION PREPARATIONS; DOSE-RESPONSE RELATIONSHIP, DRUG; GLUCOCORTICOIDS; HUMANS; PARTICLE SIZE; TISSUE DISTRIBUTION;

EID: 42149116307     PISSN: 15672018     EISSN: None     Source Type: Journal    
DOI: 10.2174/156720108783954897     Document Type: Review

References (37)

1. Melchor, R.; Biddiscome, M.F.; Mak, V.H.; Short, M.D.; Spiro, S.G. Thorax, 1993, 48, 506.
2. Weda, M.; Zanen, P.; de Boer, A.H.; Barends, D.M.; Frijlink, H.W. Int. J. Pharm., 2002, 249, 247.
3. Weda, M.; Zanen, P.; de Boer, A.H.; Barends, D.M.; Frijlink, H.W. Int. J. Pharm., 2004, 287, 79.
4. Findeisen, W. Phlügers Arch. Ges. Physiol., 1935, 236, 367.
5. Heyder, J.; Gebhart, J.; Rudolf, G.; Schiller, C.F.; Stahlhofen, W. J. Aerosol Sci., 1986, 17, 811.
6. Newman, S.P. J. Aerosol Med., 1998, 11(Suppl.1), S97.
7. Silkstone, V.L.; Dennis, J.H.; Pieron, C.A.; Chrystyn, H. J. Aerosol Med., 2002, 15, 251.
8. Gabrio, B.J.; Stein, S.W.; Velasquez, D.J. Int.J. Pharm., 1999, 186, 3.
9. Barnes, P.J.; Basbaum, C.B.; Nadel, J.A. Am. Rev. Respir. Dis., 1983, 127, 758.
10. Carstairs, J.R.; Nimmo, A.J.; Barnes, P.J. Am. Rev. Respir. Dis., 1985, 132, 541.
11. Adcock, I.M.; Gilbey, T.; Gelder, C.M.; Chung, K.F.; Barnes, P.J. Am. J. Respir. Crit. Care Med., 1996, 154, 771.
12. Lipworth, B.J.; Lee, D.K.; Anhoj, J.; Bisgaard, H. Br. J. Clin. Pharmacol., 2002, 54, 544.
13. Aswania, O.; Chrystyn, H. Biopharm. Drug Dispos., 2002, 23, 159.
14. Le Brun, P.P.; de Boer, A.H.; Mannes, G.P.; de Fraîture, D.M.; Brimicombe, R.W.; Touw, D.J.; Vinks, A.A.; Frijlink, H.W.; Heijerman, H.G. Eur. J. Pharm. Biopharm., 2002, 54, 25.
15. Hochhaus, G.; Möllmann, H. Int. J. Clin. Pharmacol. Ther. Toxicol., 1992, 30, 342.
16. Derendorf, H.; Hochhaus, G.; Möllmann, H. J. Aerosol Med., 2001, 14(Suppl 1), S9.
17. Bondesson, E.; Bengtsson, T.; Borgström, L.; Nilsson, L.E.; Norrgren, K.; Olsson, B.; Svensson, M.; Wollmer, P. Int. J. Pharm., 2003, 258, 227.
18. Dahlström, K.; Thorsson, L.; Larsson, P.; Nikander, K. Ann. Allergy Asthma Immunol., 2003, 90, 226.
19. Harding, S.M. Resp. Med., 1990, 84(Suppl.A), 25.
20. Toogood, J.H.; Lefcoe, N.M.; Haines, D.S.; Jennings, B.; Errington, N.; Baksh, L.; Chuang, L. J. Allergy Clin. Immunol., 1977, 59, 298.
21. Srichana, T.; Suedee, R.; Muanpanarai, D.; Tanmanee, N. J. Pharm. Sci., 2005, 94, 220.
22. Newnham, D.M.; Lipworth, B.J. Thorax, 1994, 49, 762.
23. Johnson, M.A.; Newman, S.P.; Bloom, R.; Talaee, N.; Clarke, S.W. Chest, 1989, 96, 6.
24. Usmani, O.S.; Biddiscombe, M.F.; Nightingale, J.A.; Underwood, S.R.; Barnes, P.J J. Appl. Physiol., 2003, 95, 2106.
25. Zanen, P.; Go, T.L.; Lammers, J-W.J. Int. J. Pharm., 1994, 107, 211.
26. Zanen, P.; Go, T.L.; Lammers, J-W.J. Thorax, 1996, 51, 977.
27. Zanen, P.; Go, T.L.; Lammers, J-W.J. Int. J. Pharm., 1995, 114, 111.
28. Leach, C.L.; Davidson, P.J.; Boudreau, R.J. Eur. Respir. J., 1998, 12, 1346.
29. Busse, W.W.; Brazinsky, S.; Jacobson, K.; Stricker, W.; Schmitt, K.; Vanden Burgt, J.; Donnell, D.; Hannon, S.; Colice, G.L. J. Allergy Clin. Immunol., 1999, 140, 1215.
30. Woodcock, A.; Acerbi, D.; Poli, G. Resp. Med., 2002, 96(Suppl D), S9.
31. Harrison, L.I.; Colice, G.L.; Donnell, D.; Soria, I.; Dockhorn, R. J. Pharm. Pharmacol., 1999, 51, 263.
32. Richards, J.; Hirst, P.; Pitcairn, G.; Mahashabde, S.; Abramowitz, W.; Nolting, A. J. Aerosol Med., 2001, 14, 197.
33. Corren, J.; Nelson, H.; Greos, L.S.; Bensch, G.; Goldstein, M.; Wu, J.; Wang, S.; Newman, K. Ann. Allergy Asthma Immunol., 2001, 87, 405.
34. Kelly, H.W. Ann. Pharmacother., 1998, 32, 220.
35. Dickens, G.R.; Wermeling, D.P.; Matheny, C.J.; John, W.; Abramowitz, W.; Sista, S.M.; Foster, T.; Choudhury, S. Ann. Allergy Asthma Immunol., 2000, 84, 528.
36. Nolting, A.; Sista, S.; Abramowitz, W. J. Pharm. Sci., 2001, 91(2), 424.
37. Martin, R.J.; Szefler, S.J.; Chinchilli, V.M.; Kraft, M.; Dolovich, M.; Boushey, H.A.; Cherniack, R.M.; Craig, T.J.; Drazen, J.M.; Fagan, J.K.; Fahy, J.V.; Fish, J.E.; Ford, J.G.; Israel, E.; Kunselman, S.J.; Lazarus, S.C.; Lemanske, R.F.; Peters, S.P.; Christine, A. Am. J. Respir. Crit. Care Med., 2002, 165, 1377.