Inhibition of sodium channel gating by trapping the domain II voltage sensor with protoxin II

Molecular Pharmacology

Volumn 73, Issue 3, 2008, Pages 1020-1028

  Sokolov, Stanislav ^a   Kraus, Richard L ^b   Scheuer, Todd ^a   Catterall, William A ^a  

^a UNIVERSITY OF WASHINGTON SCHOOL OF MEDICINE   (United States)

^b MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ARGININE; GLUTAMINE; ION CHANNEL; PROTOXIN; SODIUM CHANNEL; TRANSMEMBRANE CONDUCTANCE REGULATOR; VOLTAGE GATED SODIUM CHANNEL;

ARTICLE; BINDING SITE; BRAIN; CHANNEL GATING; GENE MUTATION; MEMBRANE STEADY POTENTIAL; PRIORITY JOURNAL; SODIUM CONDUCTANCE;

ANIMALS; BINDING SITES; DATA INTERPRETATION, STATISTICAL; ELECTROPHYSIOLOGY; FEMALE; INHIBITORY CONCENTRATION 50; ION CHANNEL GATING; KINETICS; MICROELECTRODES; OOCYTES; PATCH-CLAMP TECHNIQUES; PROTEIN STRUCTURE, TERTIARY; SCORPION VENOMS; SODIUM CHANNEL BLOCKERS; SODIUM CHANNELS; XENOPUS LAEVIS;

EID: 40849142344     PISSN: 0026895X     EISSN: 15210111     Source Type: Journal    
DOI: 10.1124/mol.107.041046     Document Type: Article

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