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Volumn 25, Issue 1, 2008, Pages 31-45

Diclofenac sodium loaded-cellulose acetate butyrate: Effect of processing variables on microparticles properties, drug release kinetics and ulcerogenic activity

Author keywords

Cellulose acetate butyrate; Encapsulation efficiency; Gastric lesion; Solvent evaporation method; Sustained release microparticles

Indexed keywords

ALCOHOL; CELLABURATE; DICLOFENAC; EUDRAGIT; PHOSPHATE; POLYMER; SURFACTANT;

EID: 38049129387     PISSN: 02652048     EISSN: 14645246     Source Type: Journal    
DOI: 10.1080/02652040701747928     Document Type: Article
Times cited : (33)

References (44)
  • 1
    • 0022639470 scopus 로고
    • Some factors affecting the miroencapsultion of pharmaceuticals with cellulose acetate phthalate
    • Beyger, JW and Nairn, JG (1986) Some factors affecting the miroencapsultion of pharmaceuticals with cellulose acetate phthalate. J Pharm Sci, 75, pp. 573-578.
    • (1986) J Pharm Sci , vol.75 , pp. 573-578
    • Beyger, J.W.1    Nairn, J.G.2
  • 3
    • 0037006611 scopus 로고    scopus 로고
    • Preparation and characterization of fentanyl-loaded PLGA microspheres: In vitro release profiles
    • Choi, HS, Seo, SA, Khang, G., Rhee, JM and Lee, HB (2002) Preparation and characterization of fentanyl-loaded PLGA microspheres: In vitro release profiles. Int J Pharm, 234, pp. 195-203.
    • (2002) Int J Pharm , vol.234 , pp. 195-203
    • Choi, H.S.1    Seo, S.A.2    Khang, G.3    Rhee, J.M.4    Lee, H.B.5
  • 4
    • 0037320895 scopus 로고    scopus 로고
    • Preparation and in vitro evaluation of modified release ketoprofen microsponges
    • Çomoǧlu, T., Gönül, N. and Baykara, T. (2003) Preparation and in vitro evaluation of modified release ketoprofen microsponges. Il Farmaco, 58, pp. 101-106.
    • (2003) Il Farmaco , vol.58 , pp. 101-106
    • Çomoǧlu, T.1    Gönül, N.2    Baykara, T.3
  • 5
    • 0023935380 scopus 로고
    • Side-effects of non-steroidal anti-inflammatory drugs
    • Cooke, PM (1988) Side-effects of non-steroidal anti-inflammatory drugs. Med J Aust, 148, pp. 248-251.
    • (1988) Med J Aust , vol.148 , pp. 248-251
    • Cooke, P.M.1
  • 6
    • 0035073301 scopus 로고    scopus 로고
    • Modeling and comparison of dissolution profiles
    • Costa, P. and Lobo, JMS (2001) Modeling and comparison of dissolution profiles. Eur J Pharm Sci, 13, pp. 123-133.
    • (2001) Eur J Pharm Sci , vol.13 , pp. 123-133
    • Costa, P.1    Lobo, J.M.S.2
  • 9
    • 38049163768 scopus 로고
    • Side effects of drugs: Anti-inflammatory and antipyretic analgesics and drugs used in gout
    • Elsevier, Amsterdam
    • Favero, A Del (1988) Side effects of drugs: Anti-inflammatory and antipyretic analgesics and drugs used in gout, Ann. 12, p. 80. Elsevier, Amsterdam
    • (1988) Ann. , vol.12 , pp. 80
    • Del Favero, A.1
  • 10
    • 0036200418 scopus 로고    scopus 로고
    • A tunable hydrogel for encapsulation and controlled release of bioactive proteins
    • Delgado, M., Spanka, C., Kerwin, LD, Wentworth Jr, P. and Janda, KD (2002) A tunable hydrogel for encapsulation and controlled release of bioactive proteins. Biomacromolecules, 3, pp. 262-271.
    • (2002) Biomacromolecules , vol.3 , pp. 262-271
    • Delgado, M.1    Spanka, C.2    Kerwin, L.D.3    Wentworth Jr., P.4    Janda, K.D.5
  • 12
    • 0003428589 scopus 로고    scopus 로고
    • FDA Guidance for Industry. Food and Drug Administration, Center for Drug Evaluation and Research, Rockville, MD
    • FDA Guidance for Industry. (1997) Dissolution testing of immediate release solid and dosage forms, Food and Drug Administration, Center for Drug Evaluation and Research, Rockville, MD
    • (1997) Dissolution Testing of Immediate Release Solid and Dosage Forms
  • 13
    • 0026608368 scopus 로고
    • Biopharmaceutical comparison of oral multiple-unit and single-unit sustained release dosage forms
    • Follonier, N. and Doelker, E. (1992) Biopharmaceutical comparison of oral multiple-unit and single-unit sustained release dosage forms. STP Pharma Sci, 2, pp. 141-158.
    • (1992) STP Pharma Sci , vol.2 , pp. 141-158
    • Follonier, N.1    Doelker, E.2
  • 14
    • 0026366263 scopus 로고
    • Inhibition of gastric-secretion by a water extract from Baccharis-Triptera
    • Gamberini, MT, Skorupa, LA, Souccar, C. and Lapa, AJ (1991) Inhibition of gastric-secretion by a water extract from Baccharis-Triptera. Mem Inst Oswaldo Cruz, 86, pp. 137-139.
    • (1991) Mem Inst Oswaldo Cruz , vol.86 , pp. 137-139
    • Gamberini, M.T.1    Skorupa, L.A.2    Souccar, C.3    Lapa, A.J.4
  • 16
    • 0032967523 scopus 로고    scopus 로고
    • Formulation design and optimization of modified-release microspheres of diclofenac sodium
    • Gohel, MC and Amin, AF (1999) Formulation design and optimization of modified-release microspheres of diclofenac sodium. Drug Dev Ind Pharm, 25, pp. 247-251.
    • (1999) Drug Dev Ind Pharm , vol.25 , pp. 247-251
    • Gohel, M.C.1    Amin, A.F.2
  • 17
    • 0031837762 scopus 로고    scopus 로고
    • Biodegradable, somatostatin acetate containing microspheres prepared by various aqueous and non-aqueous solvent evaporation methods
    • Hermann, J. and Bodmeier, R. (1998) Biodegradable, somatostatin acetate containing microspheres prepared by various aqueous and non-aqueous solvent evaporation methods. Eur J Pharm Biopharm, 45:1, pp. 75-82.
    • (1998) Eur J Pharm Biopharm , vol.45 , Issue.1 , pp. 75-82
    • Hermann, J.1    Bodmeier, R.2
  • 18
    • 0001817527 scopus 로고
    • Factors influencing the dispersion of drug powder as aerosols
    • Hickey, A., Concessio, N., Ort, M. and Platz, R. (1994) Factors influencing the dispersion of drug powder as aerosols. Pharm Tech
    • (1994) Pharm Tech
    • Hickey, A.1    Concessio, N.2    Ort, M.3    Platz, R.4
  • 19
    • 0035292910 scopus 로고    scopus 로고
    • Influence of physicochemical properties of dissolution of drugs in the gastrointestinal tract
    • Hörter, D. and Dressman, JB (2001) Influence of physicochemical properties of dissolution of drugs in the gastrointestinal tract. Adv Drug Del Rev, 46, pp. 75-87.
    • (2001) Adv Drug Del Rev , vol.46 , pp. 75-87
    • Hörter, D.1    Dressman, J.B.2
  • 20
    • 0034380586 scopus 로고    scopus 로고
    • Preparation and characterization of PLGA microparticles for the sustained release of AZT
    • Khang, G., Lee, JH, Lee, JW, Cho, JC and Lee, HB (2000) Preparation and characterization of PLGA microparticles for the sustained release of AZT. Korea Polym J, 8, pp. 80-88.
    • (2000) Korea Polym J , vol.8 , pp. 80-88
    • Khang, G.1    Lee, J.H.2    Lee, J.W.3    Cho, J.C.4    Lee, H.B.5
  • 21
    • 0033029061 scopus 로고    scopus 로고
    • Long-circulating multiple-emulsion system for improved delivery of an anticancer agent
    • Khopade, AJ and Jain, NK (1999) Long-circulating multiple-emulsion system for improved delivery of an anticancer agent. Drug Del, 6, pp. 107-110.
    • (1999) Drug Del , vol.6 , pp. 107-110
    • Khopade, A.J.1    Jain, N.K.2
  • 22
    • 0029099021 scopus 로고
    • Preparation and characterization of cytarabine-loaded w/o/w multiple emulsions
    • Kim, CK, Kim, SC, Shin, HJ, Kim, KM, Oh, KH, Lee, YB and Oh, JJ (1995) Preparation and characterization of cytarabine-loaded w/o/w multiple emulsions. Int J Pharm, 124, pp. 61-67.
    • (1995) Int J Pharm , vol.124 , pp. 61-67
    • Kim, C.K.1    Kim, S.C.2    Shin, H.J.3    Kim, K.M.4    Oh, K.H.5    Lee, Y.B.6    Oh, J.J.7
  • 24
    • 0032509838 scopus 로고    scopus 로고
    • Oil-water-oil multiple emulsion for prolonged delivery of hydrocortisone after topical application: Comparison with simple emulsions
    • Laugel, C., Baillet, A., Piemi, MP Youenang, Marty, JP and Ferrier, D. (1998) Oil-water-oil multiple emulsion for prolonged delivery of hydrocortisone after topical application: Comparison with simple emulsions. Int J Pharm, 160, pp. 109-117.
    • (1998) Int J Pharm , vol.160 , pp. 109-117
    • Laugel, C.1    Baillet, A.2    Youenang Piemi, M.P.3    Marty, J.P.4    Ferrier, D.5
  • 25
    • 0036371181 scopus 로고    scopus 로고
    • Spray-drying of proteins
    • Lee, G. (2002) Spray-drying of proteins. Pharm Biotechnol, 13, pp. 135-158.
    • (2002) Pharm Biotechnol , vol.13 , pp. 135-158
    • Lee, G.1
  • 27
    • 0031808578 scopus 로고    scopus 로고
    • Evaluation of a novel phase separation technique for the encapsulation of water-soluble drug in biodegradable polymer
    • Mandal, TK (1998) Evaluation of a novel phase separation technique for the encapsulation of water-soluble drug in biodegradable polymer. Drug Dev Ind Pharm, 24, pp. 623-639.
    • (1998) Drug Dev Ind Pharm , vol.24 , pp. 623-639
    • Mandal, T.K.1
  • 28
    • 18744395801 scopus 로고    scopus 로고
    • Effect of preparation temperature in solvent evaporation process on Eudragit RS microspheres properties
    • Mateovi-Rojnik, T., Frlan, R., Bogataj, M., Bukovec, P. and Mrhar, A. (2005) Effect of preparation temperature in solvent evaporation process on Eudragit RS microspheres properties. Chem Pharm Bull, 53, pp. 143-146.
    • (2005) Chem Pharm Bull , vol.53 , pp. 143-146
    • Mateovi-Rojnik, T.1    Frlan, R.2    Bogataj, M.3    Bukovec, P.4    Mrhar, A.5
  • 29
    • 2342652446 scopus 로고    scopus 로고
    • Mathematical comparison of dissolution profiles
    • Moore, JW and Flanner, HH (1996) Mathematical comparison of dissolution profiles. Pharm Tech, 20, pp. 64-74.
    • (1996) Pharm Tech , vol.20 , pp. 64-74
    • Moore, J.W.1    Flanner, H.H.2
  • 30
    • 0032851413 scopus 로고    scopus 로고
    • Preparation of poly (Dl-lactibe-co-glycolide) nanoparticles by modified spontaneous emulsification solvent diffusion method
    • Murakami, H., Kobayashi, M., Takeuchi, H. and Kawashima, Y. (1999) Preparation of poly (Dl-lactibe-co-glycolide) nanoparticles by modified spontaneous emulsification solvent diffusion method. Int J Pharm, 187, pp. 143-152.
    • (1999) Int J Pharm , vol.187 , pp. 143-152
    • Murakami, H.1    Kobayashi, M.2    Takeuchi, H.3    Kawashima, Y.4
  • 31
    • 0033989236 scopus 로고    scopus 로고
    • Further application of a modified spontaneous emulsification solvent diffusion method to various types of PLGA and PLA polymer for preparation of nanoparticles
    • Murakami, H., Kobayashi, M., Takeuchi, H. and Kawashima, Y. (2000) Further application of a modified spontaneous emulsification solvent diffusion method to various types of PLGA and PLA polymer for preparation of nanoparticles. Powder Tech, 107, pp. 137-143.
    • (2000) Powder Tech , vol.107 , pp. 137-143
    • Murakami, H.1    Kobayashi, M.2    Takeuchi, H.3    Kawashima, Y.4
  • 32
    • 22244451672 scopus 로고    scopus 로고
    • Preparation and in vitro evaluation of propylthiouracil microspheres made of Eudragit RL100 and cellulose acetate butyrate polymers using the emulsion-solvent evaporation method
    • Obeidat, WM and Price, JC (2005) Preparation and in vitro evaluation of propylthiouracil microspheres made of Eudragit RL100 and cellulose acetate butyrate polymers using the emulsion-solvent evaporation method. J Microencapsulation, 22, pp. 281-289.
    • (2005) J Microencapsulation , vol.22 , pp. 281-289
    • Obeidat, W.M.1    Price, J.C.2
  • 33
    • 0035821402 scopus 로고    scopus 로고
    • Microencapsulation of ibuprofen and Eudragit RS® 100 by the emulsion solvent diffusion technique
    • Perumal, D. (2001) Microencapsulation of ibuprofen and Eudragit RS® 100 by the emulsion solvent diffusion technique. Int J Pharm, 218, pp. 1-11.
    • (2001) Int J Pharm , vol.218 , pp. 1-11
    • Perumal, D.1
  • 34
    • 0018292487 scopus 로고
    • Cytoprotection by prostaglandins
    • Robert, A. (1979) Cytoprotection by prostaglandins. Gastroenterology, 77, pp. 761-767.
    • (1979) Gastroenterology , vol.77 , pp. 761-767
    • Robert, A.1
  • 36
    • 0025729451 scopus 로고
    • Phase diagram studies for microencapsulation of pharmaceutics using cellulose acetate trimellitate
    • Sanghvi, SP and Nairn, JG (1991) Phase diagram studies for microencapsulation of pharmaceutics using cellulose acetate trimellitate. J Pharm Sci, 80, pp. 394-398.
    • (1991) J Pharm Sci , vol.80 , pp. 394-398
    • Sanghvi, S.P.1    Nairn, J.G.2
  • 37
    • 0031667838 scopus 로고    scopus 로고
    • Influence of additives on the release profile of nifedipine from poly (DL-lactide-co-glycolide) microspheres
    • Sansdrap, P. and Moës, AJ (1998) Influence of additives on the release profile of nifedipine from poly (DL-lactide-co-glycolide) microspheres. J Microencapsulation, 15, pp. 545-553.
    • (1998) J Microencapsulation , vol.15 , pp. 545-553
    • Sansdrap, P.1    Moës, A.J.2
  • 39
    • 15244341414 scopus 로고    scopus 로고
    • Effects of viscosity and concentration of wall former, emulsifier and pore-inducer on the properties of amoxicillin microcapsule prepared by emulsion solvent evaporation
    • Song, M., Li, N., Sun, S., Tiedt, LR, Liebenberg, W. and deVillirs, MM (2005) Effects of viscosity and concentration of wall former, emulsifier and pore-inducer on the properties of amoxicillin microcapsule prepared by emulsion solvent evaporation. IL Farmaco, 60, pp. 261-267.
    • (2005) IL Farmaco , vol.60 , pp. 261-267
    • Song, M.1    Li, N.2    Sun, S.3    Tiedt, L.R.4    Liebenberg, W.5    deVillirs, M.M.6
  • 40
    • 38049152435 scopus 로고
    • United State Pharmacopeial 23 Convention, Inc.,, USP, Rockville, MD
    • The United State Pharmacopoeia 23 (1995) United State Pharmacopeial Convention, Inc.,, USP, Rockville, MD
    • (1995) The United State Pharmacopoeia
  • 41
    • 0023976547 scopus 로고
    • Diclofenac sodium, a reappraisal of its pharmacodynamic and pharmacokinetic properties, and therapeutic efficacy
    • Todd, PA and Sorkin, EM (1988) Diclofenac sodium, a reappraisal of its pharmacodynamic and pharmacokinetic properties, and therapeutic efficacy. Drugs, 35, pp. 244-285.
    • (1988) Drugs , vol.35 , pp. 244-285
    • Todd, P.A.1    Sorkin, E.M.2
  • 42
    • 0032990165 scopus 로고    scopus 로고
    • Modification of release rate of cyclosporine a from poly (L-lactic acid) microspheres by fatty acid esters and in vivo evaluation of the microspheres
    • Urata, T., Arimori, K. and Nakano, H. (1999) Modification of release rate of cyclosporine a from poly (L-lactic acid) microspheres by fatty acid esters and in vivo evaluation of the microspheres. J Control Rel, 58, pp. 133-141.
    • (1999) J Control Rel , vol.58 , pp. 133-141
    • Urata, T.1    Arimori, K.2    Nakano, H.3
  • 44
    • 0035901708 scopus 로고    scopus 로고
    • Polymer particle erosion controlling drug release: I. Factors influencing drug release and characterization of the release mechanism
    • Zuleger, S. and Lippold, BC (2001) Polymer particle erosion controlling drug release: I. Factors influencing drug release and characterization of the release mechanism. Int J Pharm, 217, pp. 139-152.
    • (2001) Int J Pharm , vol.217 , pp. 139-152
    • Zuleger, S.1    Lippold, B.C.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.