In vitro spermicidal activity of peptides from amphibian skin: Dermaseptin S4 and derivatives

Bioorganic and Medicinal Chemistry

Volumn 16, Issue 1, 2008, Pages 266-275

  Zairi, Amira ^a   Serres, Catherine ^b   Tangy, Frédéric ^c   Jouannet, Pierre ^b   Hani, Khaled ^a  

^a UNIVERSITY OF SOUSSE   (Tunisia)

^b UNIVERSITÉ PARIS DESCARTES   (France)

^c INSTITUT PASTEUR   (France)

Author keywords

Dermaseptins; Sperm motility; Spermicidal; Vaginal contraceptive

Indexed keywords

DERMASEPTIN K4S4; DERMASEPTIN K4S4[1-16]A; DERMASEPTIN K4S4[1-28]; DERMASEPTIN S4; DERMASEPTIN S4[6-28]; DERMASEPTIN S4A; NONOXINOL 9; SPERMICIDAL AGENT; UNCLASSIFIED DRUG;

AMPHIBIA; ARTICLE; CELL MEMBRANE; CONCENTRATION RESPONSE; CONTRACEPTION; CONTROLLED STUDY; DRUG CYTOTOXICITY; DRUG POTENCY; DRUG SAFETY; DRUG SCREENING; DRUG SYNTHESIS; FEMALE; FLUORESCENCE MICROSCOPY; FROG; HELA CELL; HUMAN; HUMAN CELL; IN VITRO STUDY; SEXUALLY TRANSMITTED DISEASE; SPERMATOZOON MOTILITY; STRUCTURE ACTIVITY RELATION; UNPLANNED PREGNANCY;

AMPHIBIAN PROTEINS; ANIMALS; ANTIMICROBIAL CATIONIC PEPTIDES; DOSE-RESPONSE RELATIONSHIP, DRUG; ELECTROSTATICS; FEMALE; HELA CELLS; HUMANS; MALE; PEPTIDES; RANIDAE; SKIN; SPERMATOCIDAL AGENTS; STRUCTURE-ACTIVITY RELATIONSHIP;

AMPHIBIA; ANURA;

EID: 38049091115     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2007.09.045     Document Type: Article

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