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Volumn 32, Issue 10, 2007, Pages 587-593

Advances in triazole antimicrobial agents

Author keywords

Antibacterial; Antifungal; Antituberculotic; Antiviral; Triazole

Indexed keywords

1 [2 (2,4 DIFLUOROPHENYL) 2 HYDROXY 1 METHYL 3 (1H 1,2,4 TRIAZOL 1 YL)PROPYL] 3 [4 (1H TETRAZOL 1 YL)PHENYL] 2 IMIDAZOLIDINONE; 2 [2 (2,4 DIFLUOROPHENYL) 2 HYDROXY 1 METHYL 3 (1H 1,2,4 TRIAZOL 1 YL)PROPYL] 4 [4 (2,2,3,3 TETRAFLUOROPROPOXY)PHENYL] 1,2,4 TRIAZOL 3(2H) ONE; 4 [4 [4 [2 (2,4 DIFLUOROPHENYL) 2 HYDROXY 1 METHYL 3 (1H 1,2,4 TRIAZOL 1 YL)PROPYL] 1 PIPERAZINYL]PHENYL] 2,4 DIHYDRO 2 [4 (TRIFLUOROMETHOXY)BENZYL] 1,2,4 TRIAZOL 3 ONE; 4 [4 [5 [2 (2,4 DIFLUOROPHENYL) 2 HYDROXY 1 METHYL 3 (1H 1,2,4, TRIAZOL 1 YL)PROPYLTHIO] 1,3 DIOXAN 2 YL] 1,3 BUTADIENYL] 3 FLUOROBENZONITIRLE; ALBACONAZOLE; ALPHA (4 CHLOROPHENYL) ALPHA (1 CYCLOPROPYL 1 METHYLETHYL) 1H 1,2,4 TRIAZOLE 1 ETHANOL; ANTIINFECTIVE AGENT; AZOLINE; ELECTRAZOLE; GENACONAZOLE; KP 103; POSACONAZOLE; SCH 50001; SCH 50002; SCH 51048; SCH 59884; T 8581; TRIAZOLE; TUBERCULOSTATIC AGENT; UNCLASSIFIED DRUG;

EID: 37049002838     PISSN: 10018689     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review
Times cited : (31)

References (30)
  • 1
    • 4644262187 scopus 로고    scopus 로고
    • Newer systemic antifungal agents pharmacokinetics, safety and efficacy [J]
    • Boucher H W, Groll A H, Chiou C C, et al. Newer systemic antifungal agents pharmacokinetics, safety and efficacy [J]. Drugs, 2004,64(18):1997-2020.
    • (2004) Drugs , vol.64 , Issue.18 , pp. 1997-2020
    • Boucher, H.W.1    Groll, A.H.2    Chiou, C.C.3
  • 2
    • 37049006430 scopus 로고    scopus 로고
    • Chinese source
    • Chinese source
  • 3
    • 37049034400 scopus 로고    scopus 로고
    • Chinese source
    • Chinese source
  • 4
    • 27744582591 scopus 로고    scopus 로고
    • Hydroxylated analogues of the orally active broad spectrum antifungal, Sch 51048 (1), and the discovery of posaconazole [Sch 56592; 2 or (S,S)-5] [J]
    • Bennett F, Saksena A K, Lovey RG, et al. Hydroxylated analogues of the orally active broad spectrum antifungal, Sch 51048 (1), and the discovery of posaconazole [Sch 56592; 2 or (S,S)-5] [J]. Bioorg Med Chem Lett, 2006, 16(1):186-190.
    • (2006) Bioorg Med Chem Lett , vol.16 , Issue.1 , pp. 186-190
    • Bennett, F.1    Saksena, A.K.2    Lovey, R.G.3
  • 5
    • 37049007125 scopus 로고    scopus 로고
    • Parang K, Sardari S. Azole derivatives and methods for making the same: WO2005/006860 A2 [P]. 2005-01-27
    • Parang K, Sardari S. Azole derivatives and methods for making the same: WO2005/006860 A2 [P]. 2005-01-27
  • 6
    • 0036301181 scopus 로고    scopus 로고
    • The discovery and process development of a commercial route to the water soluble prodrug, Fosfluconazole [J]
    • Bentley A, Butters M, Green S P, et al. The discovery and process development of a commercial route to the water soluble prodrug, Fosfluconazole [J]. Org Proc Res Dev, 2002,6(2):109-112.
    • (2002) Org Proc Res Dev , vol.6 , Issue.2 , pp. 109-112
    • Bentley, A.1    Butters, M.2    Green, S.P.3
  • 7
    • 37049019420 scopus 로고    scopus 로고
    • Synthesis and antifungal activity of novel soluble gluco-fluconazole triazolium [J]
    • Zhou C H, Bai X, Li T Q, et al. Synthesis and antifungal activity of novel soluble gluco-fluconazole triazolium [J]. Chin J Org Chem, 2005,25(Suppl):574.
    • (2005) Chin J Org Chem , vol.25 , Issue.SUPPL. , pp. 574
    • Zhou, C.H.1    Bai, X.2    Li, T.Q.3
  • 8
    • 16244418371 scopus 로고    scopus 로고
    • Comparative efficacies of tAK-187, a long-lasting ergosterol biosynthesis inhibitor, and benznidazole in preventing cardiac damage in a murine model of chagas' disease [J]
    • Corrales M, Cardozo R, Segura M A, et al. Comparative efficacies of tAK-187, a long-lasting ergosterol biosynthesis inhibitor, and benznidazole in preventing cardiac damage in a murine model of chagas' disease [J]. Antimicrob Agents Chemother, 2005,49(4):1556-1560.
    • (2005) Antimicrob Agents Chemother , vol.49 , Issue.4 , pp. 1556-1560
    • Corrales, M.1    Cardozo, R.2    Segura, M.A.3
  • 9
    • 0038440789 scopus 로고    scopus 로고
    • Efficacy of albaconazole (UR-9825) in treatment of disseminated scedosporium prolificans infection in rabbits [J]
    • Capilla J, Yustes C, Mayayo E, et al. Efficacy of albaconazole (UR-9825) in treatment of disseminated scedosporium prolificans infection in rabbits [J]. Antimicrob Agents Chemother, 2003,47(6):1948-1951.
    • (2003) Antimicrob Agents Chemother , vol.47 , Issue.6 , pp. 1948-1951
    • Capilla, J.1    Yustes, C.2    Mayayo, E.3
  • 10
    • 0034425534 scopus 로고    scopus 로고
    • Efficacies of two new antifungal agents, the triazole ravuconazole and the echinocandin LY-303366, in an experimental model of invasive aspergillosis [J]
    • Roberts J, Schock K, Marino S, et al. Efficacies of two new antifungal agents, the triazole ravuconazole and the echinocandin LY-303366, in an experimental model of invasive aspergillosis [J]. Antimicrob Agents Chemother, 2000,44(12):3381-3388.
    • (2000) Antimicrob Agents Chemother , vol.44 , Issue.12 , pp. 3381-3388
    • Roberts, J.1    Schock, K.2    Marino, S.3
  • 11
    • 0036146358 scopus 로고    scopus 로고
    • In vitro and in vivo activities of CS-758 (R-120758), a new triazole antifungal agent [J]
    • Kamai Y, Harasaki T, Fukuoka T, et al. In vitro and in vivo activities of CS-758 (R-120758), a new triazole antifungal agent [J]. Antimicrob Agents Chemother, 2002,46 (2):367-370.
    • (2002) Antimicrob Agents Chemother , vol.46 , Issue.2 , pp. 367-370
    • Kamai, Y.1    Harasaki, T.2    Fukuoka, T.3
  • 12
    • 0037447868 scopus 로고    scopus 로고
    • Synthesis and antimycotic activity of N-azolyl-2,4-dihydroxythiobenzamides [J]
    • Matysiak J, Niewiadomy A. Synthesis and antimycotic activity of N-azolyl-2,4-dihydroxythiobenzamides [J]. Bioorg Med Chem, 2003,11(10):2285-2291.
    • (2003) Bioorg Med Chem , vol.11 , Issue.10 , pp. 2285-2291
    • Matysiak, J.1    Niewiadomy, A.2
  • 13
    • 0038309147 scopus 로고    scopus 로고
    • 1.2,4-Triazolo mercapto and aminonitriles as potent antifungal agents [J]
    • Collin X, Sauleau A, Coulon J. 1.2,4-Triazolo mercapto and aminonitriles as potent antifungal agents [J]. Bioorg Med Chem Lett, 2003,13(15):2601-2605.
    • (2003) Bioorg Med Chem Lett , vol.13 , Issue.15 , pp. 2601-2605
    • Collin, X.1    Sauleau, A.2    Coulon, J.3
  • 14
    • 3042759522 scopus 로고    scopus 로고
    • (E)- and (Z)-1,2,4-Triazolylchromanone oxime ethers as conformationally constrained antifungals [J]
    • Emami S, Falahati M, Banifatemi A, et al. (E)- and (Z)-1,2,4-Triazolylchromanone oxime ethers as conformationally constrained antifungals [J]. Bioorg Med Chem, 2004,12(15):3971-3976.
    • (2004) Bioorg Med Chem , vol.12 , Issue.15 , pp. 3971-3976
    • Emami, S.1    Falahati, M.2    Banifatemi, A.3
  • 15
    • 37049005093 scopus 로고    scopus 로고
    • Chinese source
    • Chinese source
  • 16
    • 13444257877 scopus 로고    scopus 로고
    • An efficient entry to new sugar modified ketolide antibiotics [J]
    • Romero A, Chang-Hsing L, Yu-Hung C, et al. An efficient entry to new sugar modified ketolide antibiotics [J]. Tetrahedron Lett, 2005,46(9):1483-1487.
    • (2005) Tetrahedron Lett , vol.46 , Issue.9 , pp. 1483-1487
    • Romero, A.1    Chang-Hsing, L.2    Yu-Hung, C.3
  • 17
    • 3042544160 scopus 로고    scopus 로고
    • Synthesis and antibacterial activity of 5-substttuted oxazolidinones [J]
    • Phillips O A, Udo E E, Ali A A M, et al. Synthesis and antibacterial activity of 5-substttuted oxazolidinones [J]. Bioorg Med Chem, 2003,11(1):35-41.
    • (2003) Bioorg Med Chem , vol.11 , Issue.1 , pp. 35-41
    • Phillips, O.A.1    Udo, E.E.2    Ali, A.A.M.3
  • 18
    • 0033694468 scopus 로고    scopus 로고
    • Synthesis and antimicrobial activities of some 3-arylamino-5-[2-(substituted1-imidazolyl)ethyl]-1,2,4-triazole derivatives [J]
    • Demirayak S, Benkli K, Guuven K. Synthesis and antimicrobial activities of some 3-arylamino-5-[2-(substituted1-imidazolyl)ethyl]-1,2,4-triazole derivatives [J]. Eur J Med Chem, 2000,35(11):1037-1040.
    • (2000) Eur J Med Chem , vol.35 , Issue.11 , pp. 1037-1040
    • Demirayak, S.1    Benkli, K.2    Guuven, K.3
  • 19
    • 19544394603 scopus 로고    scopus 로고
    • Turan-Zitouni G, Kaplakcikli Z A, Yildiz M T, et al. Synthesis and antimicrobial activity of 4-phenyl/cyclohexyl-5-(1-phenoxyethyl)-3-[N-(2- thiazolyl)acetamido] thio-4H-1,2,4- triazole derivatives [J]. Eur J Med Chem, 2005,40(6):607-613.
    • Turan-Zitouni G, Kaplakcikli Z A, Yildiz M T, et al. Synthesis and antimicrobial activity of 4-phenyl/cyclohexyl-5-(1-phenoxyethyl)-3-[N-(2- thiazolyl)acetamido] thio-4H-1,2,4- triazole derivatives [J]. Eur J Med Chem, 2005,40(6):607-613.
  • 20
    • 28444465911 scopus 로고    scopus 로고
    • Yang J G, Pan F Y, Shao H. Synthesis, crystal structure and antibacterial activities of 3-[3-methyl-(2-thienyl)methylenehydrazinocarbonyl]-(1H)-1,2,4- triazol [J]. Chin J Struct Chem, 2005,11(24):1286-1289.
    • Yang J G, Pan F Y, Shao H. Synthesis, crystal structure and antibacterial activities of 3-[3-methyl-(2-thienyl)methylenehydrazinocarbonyl]-(1H)-1,2,4- triazol [J]. Chin J Struct Chem, 2005,11(24):1286-1289.
  • 21
    • 0033834164 scopus 로고    scopus 로고
    • Novel synthetic approach for antifungal and antibacterial organotin compounds [J]
    • Kidwai M, Dave B, Misra P, et al. Novel synthetic approach for antifungal and antibacterial organotin compounds [J]. Inorg Chem Commun, 2000,3(9):465-468.
    • (2000) Inorg Chem Commun , vol.3 , Issue.9 , pp. 465-468
    • Kidwai, M.1    Dave, B.2    Misra, P.3
  • 22
    • 8444243711 scopus 로고    scopus 로고
    • Synthesis and antimycobacterial activity of pyridylmethylsulfanyl and naphthylmethylsulfanyl derivatives of benzazoles, 1,2,4-triazole, and pyridine-2-carbothioamide/-2-carbonitrile [J]
    • Zahajská L, Klimesová V, Koci J, et al. Synthesis and antimycobacterial activity of pyridylmethylsulfanyl and naphthylmethylsulfanyl derivatives of benzazoles, 1,2,4-triazole, and pyridine-2-carbothioamide/-2-carbonitrile [J]. Arch Pharm, 2004,337(10):549-555.
    • (2004) Arch Pharm , vol.337 , Issue.10 , pp. 549-555
    • Zahajská, L.1    Klimesová, V.2    Koci, J.3
  • 23
    • 22844446396 scopus 로고    scopus 로고
    • Thiourea, triazole and thiadiazine compounds and their metal complexes as antifungal agents [J]
    • Rodriguez-Fernández E, Manzano J L, Benito J J, et al. Thiourea, triazole and thiadiazine compounds and their metal complexes as antifungal agents [J]. J Inorg Biochem, 2005,99(8):1558-1572.
    • (2005) J Inorg Biochem , vol.99 , Issue.8 , pp. 1558-1572
    • Rodriguez-Fernández, E.1    Manzano, J.L.2    Benito, J.J.3
  • 24
    • 22044444255 scopus 로고    scopus 로고
    • Studies on pyrazine derivatives. 38. Synthesis, reactions, and tuberculostatic activity of pyrazinyl-substituted derivatives of hydrazinocarbodithioic acid [J]
    • Foks H, Trapkowska I, Janowiec M, et al. Studies on pyrazine derivatives. 38. Synthesis, reactions, and tuberculostatic activity of pyrazinyl-substituted derivatives of hydrazinocarbodithioic acid [J]. Chem Heterocycl Compd, 2004,40(9):1185-1194.
    • (2004) Chem Heterocycl Compd , vol.40 , Issue.9 , pp. 1185-1194
    • Foks, H.1    Trapkowska, I.2    Janowiec, M.3
  • 25
    • 0035753788 scopus 로고    scopus 로고
    • Inhibition of the helicase activity of HCV NTPase/helicase by 1-beta-D-ribofuranosyl-1,2,4-triazole-3- carboxamide-5′-triphosphate (ribavirin-TP) [J]
    • Borowski P, Lang M, Niebuhr A, et al. Inhibition of the helicase activity of HCV NTPase/helicase by 1-beta-D-ribofuranosyl-1,2,4-triazole-3- carboxamide-5′-triphosphate (ribavirin-TP) [J]. Acta Biochim Pol, 2001,48 (3):739-744.
    • (2001) Acta Biochim Pol , vol.48 , Issue.3 , pp. 739-744
    • Borowski, P.1    Lang, M.2    Niebuhr, A.3
  • 26
    • 32344433894 scopus 로고    scopus 로고
    • Synthesis of cyclopentenyl carbocyclic nucleosides as potential antiviral agents against orthopoxviruses and SARS [J]
    • Cho J H, Bernard D L, Sidwell R W, et al. Synthesis of cyclopentenyl carbocyclic nucleosides as potential antiviral agents against orthopoxviruses and SARS [J]. J Med Chem, 2006,49(3):1140-1148.
    • (2006) J Med Chem , vol.49 , Issue.3 , pp. 1140-1148
    • Cho, J.H.1    Bernard, D.L.2    Sidwell, R.W.3
  • 27
    • 4544287480 scopus 로고    scopus 로고
    • Recent advances in 4′-thionucleosides as potential antiviral and antitumor agents [J]
    • Gunaga P, Moon H R, Choi WJ, et al. Recent advances in 4′-thionucleosides as potential antiviral and antitumor agents [J]. Curr Med Chem, 2004,11(10):2585-2637.
    • (2004) Curr Med Chem , vol.11 , Issue.10 , pp. 2585-2637
    • Gunaga, P.1    Moon, H.R.2    Choi, W.J.3
  • 28
    • 26044483537 scopus 로고    scopus 로고
    • Synthesis and biological activity of 1H-benzotriazole and 1H-benzimidazole analogues - inhibitors of the NTpase/helicase of HCV and of some related Flaviviridae [J]
    • Bretner M, Baier A, Kopanska K, et al. Synthesis and biological activity of 1H-benzotriazole and 1H-benzimidazole analogues - inhibitors of the NTpase/helicase of HCV and of some related Flaviviridae [J]. Antiviral Chem Chemother, 2005,16(5):315-326.
    • (2005) Antiviral Chem Chemother , vol.16 , Issue.5 , pp. 315-326
    • Bretner, M.1    Baier, A.2    Kopanska, K.3
  • 29
    • 20544475634 scopus 로고    scopus 로고
    • Initial synthesis of UK-427, 857 (Maraviroc) [J]
    • Price D A, Gayton S, Selby M D, et al. Initial synthesis of UK-427, 857 (Maraviroc) [J]. Tetrahedron Lett, 2005,46(30):5005-5007.
    • (2005) Tetrahedron Lett , vol.46 , Issue.30 , pp. 5005-5007
    • Price, D.A.1    Gayton, S.2    Selby, M.D.3
  • 30
    • 2342561153 scopus 로고    scopus 로고
    • Rational design and synthesis of novel dimeric diketoacid-containing inhibitors of HIV-1 integrase : Implication for binding to two metal ions on the active site of integrase [J]
    • Long Y Q, Jiang X H, Dayam R, et al. Rational design and synthesis of novel dimeric diketoacid-containing inhibitors of HIV-1 integrase : implication for binding to two metal ions on the active site of integrase [J]. J Med Chem, 2004,47(10):2561-2573.
    • (2004) J Med Chem , vol.47 , Issue.10 , pp. 2561-2573
    • Long, Y.Q.1    Jiang, X.H.2    Dayam, R.3


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