Initial synthesis of UK-427,857 (Maraviroc)

Tetrahedron Letters

Volumn 46, Issue 30, 2005, Pages 5005-5007

  Price, David A ^a   Gayton, Simon ^a   Selby, Matthew D ^a   Ahman, Jens ^a   Haycock Lewandowski, Sarah ^a   Stammen, Blanda L ^a   Warren, Andrew ^a  

^a PFIZER GLOBAL RESEARCH AND DEVELOPMENT   (United Kingdom)

Author keywords

Amide; Fluorination; Heterocycles; Triazoles; Tropane

Indexed keywords

4,4 DIFLUOROCYCLOHEXANOIC ACID; AMIDE; MARAVIROC; POLYMER; REAGENT; UNCLASSIFIED DRUG;

ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS;

EID: 20544475634     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2005.05.082     Document Type: Article

References (15)

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14. ® catalogue number 800369.
15. 5O requires C, 67.75; H, 8.06; N, 13.54; Found C, 67.77; H, 8.00; N, 13.64.