Application of the BD ACTOne™ technology for the high-throughput screening of Gs-coupled receptor antagonists

Journal of Biomolecular Screening

Volumn 12, Issue 8, 2007, Pages 1068-1073

  Visegrády, András ^a   Boros, András ^a   Némethy, Zsolt ^a   Kiss, Béla ^a   Keseru, György M ^a  

^a GEDEON RICHTER LTD   (Hungary)

Author keywords

cAMP; Cyclic nucleotide gated channel; G protein coupled receptor; High throughput screening; Peptide parathyroid hormone 2 receptor

Indexed keywords

CALCIUM; G PROTEIN COUPLED RECEPTOR; PARATHYROID HORMONE RECEPTOR 2; STIMULATORY GUANINE NUCLEOTIDE BINDING PROTEIN;

ARTICLE; BIOSENSOR; CALCIUM TRANSPORT; CELL MEMBRANE DEPOLARIZATION; CELL STRAIN HEK293; CONTROLLED STUDY; DRUG DETERMINATION; HIGH THROUGHPUT SCREENING; HUMAN; HUMAN CELL; ISOTOPE LABELING; PRIORITY JOURNAL; SCREENING TEST;

CALCIUM; CELL LINE; CYCLIC AMP; CYCLIC NUCLEOTIDE-GATED CATION CHANNELS; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG EVALUATION, PRECLINICAL; FLUORESCENCE; GTP-BINDING PROTEIN ALPHA SUBUNITS, GS; HUMANS; MEMBRANE POTENTIALS; NEUROPEPTIDES; RECEPTOR, PARATHYROID HORMONE, TYPE 1; RECEPTORS, G-PROTEIN-COUPLED; SIGNAL TRANSDUCTION;

EID: 36549045575     PISSN: 10870571     EISSN: 1552454X     Source Type: Journal    
DOI: 10.1177/1087057107309035     Document Type: Article

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