Inhibition of ryanodine receptors by 4-(2-aminopropyl)-3,5-dichloro-N,N- dimethylaniline (FLA 365) in canine pulmonary arterial smooth muscle cells

Journal of Pharmacology and Experimental Therapeutics

Volumn 323, Issue 1, 2007, Pages 381-390

  Ostrovskaya, Olga ^a,e   Goyal, Ravi ^a   Osman, Noah ^a,b   McAllister, Claire E ^c   Pessah, Isaac N ^d   Hume, Joseph R ^c   Wilson, Sean M ^a,b,f  

^a UNIVERSITY OF MISSISSIPPI   (United States)

^b UNIVERSITY OF MISSISSIPPI   (United States)

^c UNIVERSITY OF NEVADA SCHOOL OF MEDICINE   (United States)

^d UNIVERSITY OF CALIFORNIA   (United States)

^e UNIVERSITY OF TENNESSEE HEALTH SCIENCE CENTER   (United States)

^f UNIVERSITY OF MISSISSIPPI   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2,6 DICHLORO 4 DIMETHYLAMINOAMPHETAMINE; BARIUM; CAFFEINE; CALCIUM; CALCIUM CHANNEL L TYPE; CARBACHOL; CYCLOPIAZONIC ACID; FURA 2; INOSITOL 1,4,5 TRISPHOSPHATE RECEPTOR; RYANODINE; RYANODINE RECEPTOR; SEROTONIN;

ANIMAL CELL; ARTICLE; CALCIUM TRANSPORT; CELL STRAIN HEK293; CONTROLLED STUDY; DOG; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; GENE EXPRESSION; HEART MUSCLE; HUMAN; HUMAN CELL; IC 50; MEMBRANE CONDUCTANCE; MEMBRANE CURRENT; NONHUMAN; PRIORITY JOURNAL; PULMONARY ARTERY; SARCOPLASMIC RETICULUM; SMOOTH MUSCLE FIBER; VOLTAGE CLAMP;

ANIMALS; BARIUM; CAFFEINE; CALCIUM CHANNEL BLOCKERS; CALCIUM SIGNALING; CELL LINE; DOGS; DOSE-RESPONSE RELATIONSHIP, DRUG; ELECTROPHYSIOLOGY; FEMALE; INDOLES; MALE; MUSCLE, SMOOTH, VASCULAR; MYOCYTES, SMOOTH MUSCLE; PHENETHYLAMINES; PULMONARY ARTERY; RYANODINE; RYANODINE RECEPTOR CALCIUM RELEASE CHANNEL;

EID: 34548835267     PISSN: 00223565     EISSN: 15210103     Source Type: Journal    
DOI: 10.1124/jpet.107.122119     Document Type: Article

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