Nafamostat mesilate reversibly blocks acid-sensing ion channel currents

Biochemical and Biophysical Research Communications

Volumn 363, Issue 1, 2007, Pages 203-208

  Ugawa, Shinya ^a   Ishida, Yusuke ^a   Ueda, Takashi ^a   Inoue, Kiyoshi ^a   Nagao, Masataka ^a   Shimada, Shoichi ^a  

^a NAGOYA CITY UNIVERSITY GRADUATE SCHOOL OF MEDICAL SCIENCES   (Japan)

Author keywords

6 Amidino 2 naphthol (AN); Acid sensing ion channel (ASIC); FUT 175; Inhibition; Nafamostat mesilate (NM); Oocyte electrophysiology; p Guanidinobenzoic acid (PGBA); Proton

Indexed keywords

4 GUANIDINOBENZOIC ACID; 6 AMIDINO 2 NAPHTHOL; ACID SENSING ION CHANNEL; DRUG METABOLITE; NAFAMSTAT MESILATE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; ELECTRIC CURRENT; ELECTRIC POTENTIAL; ELECTROPHYSIOLOGY; FEMALE; IC 50; NONHUMAN; NUCLEOTIDE SEQUENCE; OOCYTE; PRIORITY JOURNAL; PROTEIN EXPRESSION;

ANIMALS; CELLS, CULTURED; DOSE-RESPONSE RELATIONSHIP, DRUG; GUANIDINES; ION CHANNEL GATING; MEMBRANE POTENTIALS; MEMBRANE PROTEINS; NERVE TISSUE PROTEINS; OOCYTES; SODIUM CHANNELS; XENOPUS LAEVIS;

EID: 34548760753     PISSN: 0006291X     EISSN: 10902104     Source Type: Journal    
DOI: 10.1016/j.bbrc.2007.08.133     Document Type: Article

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